AR018994A1 - TIAZOLIDINDIONA COMPOUNDS, A PROCESS FOR PREPARATION, PHARMACEUTICAL COMPOSITION THAT INCLUDES THEM AND THE USE OF THEM FOR THE MANUFACTURE OF A MEDICINAL PRODUCT - Google Patents
TIAZOLIDINDIONA COMPOUNDS, A PROCESS FOR PREPARATION, PHARMACEUTICAL COMPOSITION THAT INCLUDES THEM AND THE USE OF THEM FOR THE MANUFACTURE OF A MEDICINAL PRODUCTInfo
- Publication number
- AR018994A1 AR018994A1 ARP990105329A AR018994A1 AR 018994 A1 AR018994 A1 AR 018994A1 AR P990105329 A ARP990105329 A AR P990105329A AR 018994 A1 AR018994 A1 AR 018994A1
- Authority
- AR
- Argentina
- Prior art keywords
- manufacture
- preparation
- pharmaceutical composition
- tiazolidindiona
- compounds
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title 1
- 229940126601 medicinal product Drugs 0.000 title 1
- 239000012453 solvate Substances 0.000 abstract 2
- -1 thiazolidinedione compound Chemical class 0.000 abstract 2
- ZOBPZXTWZATXDG-UHFFFAOYSA-N 1,3-thiazolidine-2,4-dione Chemical compound O=C1CSC(=O)N1 ZOBPZXTWZATXDG-UHFFFAOYSA-N 0.000 abstract 1
- 208000024172 Cardiovascular disease Diseases 0.000 abstract 1
- 208000031226 Hyperlipidaemia Diseases 0.000 abstract 1
- 206010020772 Hypertension Diseases 0.000 abstract 1
- 229940123464 Thiazolidinedione Drugs 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 125000001301 ethoxy group Chemical group [H]C([H])([H])C([H])([H])O* 0.000 abstract 1
- 201000001421 hyperglycemia Diseases 0.000 abstract 1
- 150000002688 maleic acid derivatives Chemical class 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- SUFUKZSWUHZXAV-BTJKTKAUSA-N rosiglitazone maleate Chemical compound [H+].[H+].[O-]C(=O)\C=C/C([O-])=O.C=1C=CC=NC=1N(C)CCOC(C=C1)=CC=C1CC1SC(=O)NC1=O SUFUKZSWUHZXAV-BTJKTKAUSA-N 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Un compuesto tiazolidindiona que comprende la sal del ácido maleico 5-[4-[2-(N-metil-N-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4-diona o un isomeroo forma tautomérica del mismo y/o un solvato farmacéuticamente aceptable del mismo, un proceso parasu preparacion, composicion farmacéutica quelos comprende y el uso de la sal del ácido maleico 5-[4-[2-(N-metil-N-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4-diona o un isomero o formatautomérica del mismo y/o un solvato farmacéuticamente aceptabledel mismo para la fabricacion de un medicamento para el tratamiento y/o profilaxis de lahiperglicemia, hiperlipidemia, la hipertension y la enfermedad cardiovascular.A thiazolidinedione compound comprising the maleic acid salt 5- [4- [2- (N-methyl-N- (2-pyridyl) amino) ethoxy] benzyl] thiazolidin-2,4-dione or an isomeric tautomeric form thereof and / or a pharmaceutically acceptable solvate thereof, a process for its preparation, pharmaceutical composition which comprises and the use of the maleic acid salt 5- [4- [2- (N-methyl-N- (2-pyridyl) amino)) ethoxy] benzyl] thiazolidin-2,4-dione or an isomer or formatautomer thereof and / or a pharmaceutically acceptable solvate thereof for the manufacture of a medicament for the treatment and / or prophylaxis of hyperglycemia, hyperlipidemia, hypertension and cardiovascular disease .
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ARP990105329 AR018994A1 (en) | 1999-10-21 | 1999-10-21 | TIAZOLIDINDIONA COMPOUNDS, A PROCESS FOR PREPARATION, PHARMACEUTICAL COMPOSITION THAT INCLUDES THEM AND THE USE OF THEM FOR THE MANUFACTURE OF A MEDICINAL PRODUCT |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ARP990105329 AR018994A1 (en) | 1999-10-21 | 1999-10-21 | TIAZOLIDINDIONA COMPOUNDS, A PROCESS FOR PREPARATION, PHARMACEUTICAL COMPOSITION THAT INCLUDES THEM AND THE USE OF THEM FOR THE MANUFACTURE OF A MEDICINAL PRODUCT |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR018994A1 true AR018994A1 (en) | 2001-12-26 |
Family
ID=45606574
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP990105329 AR018994A1 (en) | 1999-10-21 | 1999-10-21 | TIAZOLIDINDIONA COMPOUNDS, A PROCESS FOR PREPARATION, PHARMACEUTICAL COMPOSITION THAT INCLUDES THEM AND THE USE OF THEM FOR THE MANUFACTURE OF A MEDICINAL PRODUCT |
Country Status (1)
| Country | Link |
|---|---|
| AR (1) | AR018994A1 (en) |
-
1999
- 1999-10-21 AR ARP990105329 patent/AR018994A1/en unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |