AR015976A1 - Composiciones que contienen agonistas de h2 de histamina para el tratamiento del ojo seco y el uso de las mismas en la manufactura de un medicamento - Google Patents
Composiciones que contienen agonistas de h2 de histamina para el tratamiento del ojo seco y el uso de las mismas en la manufactura de un medicamentoInfo
- Publication number
- AR015976A1 AR015976A1 ARP980105251A ARP980105251A AR015976A1 AR 015976 A1 AR015976 A1 AR 015976A1 AR P980105251 A ARP980105251 A AR P980105251A AR P980105251 A ARP980105251 A AR P980105251A AR 015976 A1 AR015976 A1 AR 015976A1
- Authority
- AR
- Argentina
- Prior art keywords
- manufacture
- dry eye
- agonists
- same
- compositions containing
- Prior art date
Links
- 208000003556 Dry Eye Syndromes Diseases 0.000 title abstract 2
- 206010013774 Dry eye Diseases 0.000 title abstract 2
- 239000000556 agonist Substances 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title abstract 2
- NTYJJOPFIAHURM-UHFFFAOYSA-N Histamine Chemical compound NCCC1=CN=CN1 NTYJJOPFIAHURM-UHFFFAOYSA-N 0.000 title 2
- 229960001340 histamine Drugs 0.000 title 1
- 229940126601 medicinal product Drugs 0.000 title 1
- OLHQOJYVQUNWPL-UHFFFAOYSA-N dimaprit Chemical compound CN(C)CCCSC(N)=N OLHQOJYVQUNWPL-UHFFFAOYSA-N 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003937 drug carrier Substances 0.000 abstract 1
- MURRAGMMNAYLNA-UHFFFAOYSA-N impromidine Chemical compound N1C=NC(CSCCNC(N)=NCCCC=2NC=NC=2)=C1C MURRAGMMNAYLNA-UHFFFAOYSA-N 0.000 abstract 1
- 229950005073 impromidine Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Una composicion para el tratamiento del ojo seco en humanos, que comprende una cantidad farmacéuticamente efectiva de uno o más agonista(s) de H2 dehistamina tales como dimaprit, anthamine e impromidine, en un portador farmacéuticamente aceptable; yel uso de la misma para la manufactura de unmedicamento.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6290697P | 1997-10-21 | 1997-10-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR015976A1 true AR015976A1 (es) | 2001-05-30 |
Family
ID=22045617
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP980105251A AR015976A1 (es) | 1997-10-21 | 1998-10-21 | Composiciones que contienen agonistas de h2 de histamina para el tratamiento del ojo seco y el uso de las mismas en la manufactura de un medicamento |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US6274160B1 (es) |
| AR (1) | AR015976A1 (es) |
| AU (1) | AU1104799A (es) |
| WO (1) | WO1999020265A1 (es) |
| ZA (1) | ZA989513B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011034551A2 (en) | 2009-09-15 | 2011-03-24 | Qlt Inc. | Pharmaceutical formulations comprising 9-cis-retinyl esters in a lipid vehicle |
| KR20180043846A (ko) | 2010-04-19 | 2018-04-30 | 노벨리언 테라퓨틱스 인코포레이티드 | 내인성 레티노이드 결핍과 연관된 시각 장애의 치료 또는 완화를 위한 치료 요법 및 방법 |
| CA2865935C (en) | 2012-03-01 | 2021-12-14 | Qlt Inc. | Therapeutic regimens and methods for improving visual function in visual disorders associated with an endogenous retinoid deficiency |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3991759A (en) | 1975-10-28 | 1976-11-16 | Alza Corporation | Method and therapeutic system for treating aqueous deficient dry eye |
| US4131651A (en) | 1977-10-25 | 1978-12-26 | Barnes-Hind Pharmaceuticals, Inc. | Treatment of dry eye |
| US4409205A (en) | 1979-03-05 | 1983-10-11 | Cooper Laboratories, Inc. | Ophthalmic solution |
| US4370325A (en) | 1979-03-30 | 1983-01-25 | Dermik Laboratories | Pharmaceutical compositions and method of treatment |
| US4315024A (en) * | 1980-08-08 | 1982-02-09 | Cooper Laboratories, Inc. | Compositions and method for treating red eye |
| US4744980A (en) | 1986-04-28 | 1988-05-17 | Holly Frank J | Ophthalmic solution for treatment of dry eye syndrome |
| US4883658A (en) | 1986-04-28 | 1989-11-28 | Holly Frank J | Ophthalmic solution for treatment of dry-eye syndrome |
| US4818537A (en) | 1986-10-21 | 1989-04-04 | Liposome Technology, Inc. | Liposome composition for treating dry eye |
| US4966773A (en) | 1986-11-25 | 1990-10-30 | Alcon Laboratories, Inc. | Topical ophthalmic compositions containing microfine retinoid particles |
| US4914088A (en) | 1987-04-02 | 1990-04-03 | Thomas Glonek | Dry eye treatment solution and method |
| US5075104A (en) | 1989-03-31 | 1991-12-24 | Alcon Laboratories, Inc. | Ophthalmic carboxy vinyl polymer gel for dry eye syndrome |
| US5041434A (en) | 1991-08-17 | 1991-08-20 | Virginia Lubkin | Drugs for topical application of sex steroids in the treatment of dry eye syndrome, and methods of preparation and application |
| ES2084722T3 (es) | 1990-05-29 | 1996-05-16 | Boston Ocular Res | Composicion para tratamiento del ojo seco. |
| JP2594486B2 (ja) | 1991-01-15 | 1997-03-26 | アルコン ラボラトリーズ インコーポレイテッド | 局所的眼薬組成物 |
| US5294433A (en) | 1992-04-15 | 1994-03-15 | The Procter & Gamble Company | Use of H-2 antagonists for treatment of gingivitis |
| US5290572A (en) | 1992-08-06 | 1994-03-01 | Deo Corporation | Opthalmic composition for treating dry eye |
| BR9203277A (pt) | 1992-08-21 | 1994-03-01 | Cesar Roberto Dias Nahoum | Utilizaccao de drogas eretogenicas e respectivas metodologias de aplicacao |
| US5869479A (en) * | 1997-08-14 | 1999-02-09 | Schering Corporation | Treatment of upper airway allergic responses |
-
1998
- 1998-10-19 ZA ZA989513A patent/ZA989513B/xx unknown
- 1998-10-20 WO PCT/US1998/022144 patent/WO1999020265A1/en not_active Ceased
- 1998-10-20 AU AU11047/99A patent/AU1104799A/en not_active Abandoned
- 1998-10-20 US US09/529,837 patent/US6274160B1/en not_active Expired - Fee Related
- 1998-10-21 AR ARP980105251A patent/AR015976A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA989513B (en) | 1999-04-21 |
| WO1999020265A1 (en) | 1999-04-29 |
| US6274160B1 (en) | 2001-08-14 |
| AU1104799A (en) | 1999-05-10 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CL2008001920A1 (es) | Composicion farmaceutica que comprende un inhibidor de la pde 2, un agonista del receptor selectivo e2 y un portador; y uso en el tratamiento de fractura y/o defecto oseo (div. sol. 3179-04). | |
| YU38802A (sh) | Nova kompozicija i njena upotreba | |
| MD960330A (ro) | Compuşi nepeptidilici, compoziţie farmaceutică pe baza acestora, metodă de tratament | |
| AU2855399A (en) | Vascularization inhibitors | |
| ES2081531T3 (es) | Composiciones farmaceuticas que contienen rifaximina para el tratamiento de infecciones vaginales. | |
| MY129356A (en) | Electrospun pharmaceutical compositions | |
| ES2167377T3 (es) | Derivados de piridina farmacologicamente activos y procedimientos para la preparacion de los mismos. | |
| CR6592A (es) | Compuestos para el tratamiento de la isquemia | |
| AR066982A2 (es) | Compuestos heteroaromaticos sustituidos como inhibidoress tirosin quinasa, composiciones farmaceuticas que los contiene y su uso en la preparacion de medicamentos | |
| HUP0103567A3 (en) | 2-substituted-1-piperidyl benzimidazole compounds as orl1-receptor agonists, process for their preparation and pharmaceutical compositions containing the same | |
| ES2190205T3 (es) | Combinacion para el tratamiento de la dependencia del alcohol que contiene un antagonista opioide y un modulador del complejo receptor de nmda. | |
| AR017222A1 (es) | Procedimiento de utilizacion de un agente que inhibe el desarrollo de p.ovale, en la preparacion de medicamentos | |
| YU13301A (sh) | Muskarinski agonisti i antagonisti | |
| SV2008002856A (es) | 2-amino-7, 8-dihidro-6h-pirido [4,3-d] pirimidina-5-onas | |
| SE9802937D0 (sv) | Novel compounds | |
| IL139318A (en) | Sugar alcohol mixtures as therapeutic agents and pharmaceutical compositions containing the same | |
| CL2002001701A1 (es) | Uso de al menos un compuesto seleccionado entre melatonina, agentes melatoninergicos, agonistas y antagonistas de melatonina, en una cantidad de 0,0025-50 mg, para preparar un medicamento util para el tratamiento y mejora de la calidad repadora del sueno. | |
| AR024232A1 (es) | Bromhidrato de eletriptan monohidratado, composicion farmaceutica, su uso en la preparacion de medicamentos y procedimiento para su preparacion | |
| AR015976A1 (es) | Composiciones que contienen agonistas de h2 de histamina para el tratamiento del ojo seco y el uso de las mismas en la manufactura de un medicamento | |
| HRP20000781B1 (hr) | Šumeći pripravci | |
| ES2193007T1 (es) | Formulacion farmaceutica estable que comprende la modificacion ii de torsemida. | |
| ES2191908T3 (es) | 4-aminopirrol(3,2-d)pirimidinas como antagonistas del receptor del neuropeptido. | |
| ES2185698T3 (es) | Composicion de tratamiento anti-acne de la piel. | |
| BR9508021A (pt) | Composição farmacêutica para o tratamento de distúrbios esquizofrênicos, uso de um agente imunossupressor, e, processo de tratamento de um paciente esquizofrênico | |
| BR9802803A (pt) | ação e composições farmacêuticas contendo os mesmos. |