AR003928A1 - Comprimido del liberacion controlada - Google Patents
Comprimido del liberacion controladaInfo
- Publication number
- AR003928A1 AR003928A1 ARP960101520A AR10152096A AR003928A1 AR 003928 A1 AR003928 A1 AR 003928A1 AR P960101520 A ARP960101520 A AR P960101520A AR 10152096 A AR10152096 A AR 10152096A AR 003928 A1 AR003928 A1 AR 003928A1
- Authority
- AR
- Argentina
- Prior art keywords
- polymer
- tablet
- pharmaceutical agent
- rate
- water
- Prior art date
Links
- 229920000642 polymer Polymers 0.000 abstract 5
- 239000008177 pharmaceutical agent Substances 0.000 abstract 3
- 239000011230 binding agent Substances 0.000 abstract 1
- 239000000969 carrier Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000013270 controlled release Methods 0.000 abstract 1
- 239000003085 diluting agent Substances 0.000 abstract 1
- 238000004090 dissolution Methods 0.000 abstract 1
- 239000004615 ingredient Substances 0.000 abstract 1
- 239000000314 lubricant Substances 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 230000008961 swelling Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
Abstract
Un comprimido de liberación controlada que incluye un agente farmacéutico y un excipiente. El excipiente incluye por lo menos 50% de polímero susceptiblede hincharse con agua y un lubricante. El polímero susceptible de hincharse con agua seselecci ona de manera que la velocidad de hinchado del polímero seaigual a la velocidad de disolución de polímero hinchado. Además, el excipiente puede incluir otros ingredientes tales como diluyentes, soportes, ligantes yotros compuestosfarmacológicamente inactivos. El polímero se selecciona teniendo en cuenta el agente farmacéutico, de manera que el comprimido sedisuelva completamente al mismo tiempo que se libera la última porción del agente farmacéutico.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39579295A | 1995-02-28 | 1995-02-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR003928A1 true AR003928A1 (es) | 1998-09-30 |
Family
ID=23564527
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP960101520A AR003928A1 (es) | 1995-02-28 | 1996-02-26 | Comprimido del liberacion controlada |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP0821582B1 (es) |
| JP (1) | JPH11509169A (es) |
| AR (1) | AR003928A1 (es) |
| AT (1) | ATE228829T1 (es) |
| AU (1) | AU722741B2 (es) |
| CA (1) | CA2213455A1 (es) |
| DE (1) | DE69625189D1 (es) |
| MY (1) | MY113429A (es) |
| PA (1) | PA8388101A1 (es) |
| TW (1) | TW431891B (es) |
| WO (1) | WO1996026718A2 (es) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5945125A (en) * | 1995-02-28 | 1999-08-31 | Temple University | Controlled release tablet |
| WO1998029095A2 (en) * | 1997-01-03 | 1998-07-09 | Elan Corporation, Plc | Sustained release cisapride mini-tablet formulation |
| US6090411A (en) * | 1998-03-09 | 2000-07-18 | Temple University | Monolithic tablet for controlled drug release |
| ES2270982T3 (es) | 2000-02-04 | 2007-04-16 | Depomed, Inc. | Forma de dosificacion de nucleo y carcasa que se aproxima a una liberacion del farmaco de orden cero. |
| TWI312285B (en) | 2001-10-25 | 2009-07-21 | Depomed Inc | Methods of treatment using a gastric retained gabapentin dosage |
| US6723340B2 (en) * | 2001-10-25 | 2004-04-20 | Depomed, Inc. | Optimal polymer mixtures for gastric retentive tablets |
| US7612112B2 (en) | 2001-10-25 | 2009-11-03 | Depomed, Inc. | Methods of treatment using a gastric retained gabapentin dosage |
| AU2004204825B2 (en) | 2003-01-13 | 2007-07-19 | Dynogen Pharmaceuticals, Inc. | Method of treating functional bowel disorders |
| US20050013863A1 (en) | 2003-07-18 | 2005-01-20 | Depomed, Inc., A Corporation Of The State Of California | Dual drug dosage forms with improved separation of drugs |
| WO2006009769A1 (en) | 2004-06-17 | 2006-01-26 | Forest Laboratories, Inc. | Modified release formulation of memantine |
| EP1954257A4 (en) | 2005-10-14 | 2009-05-20 | Lundbeck & Co As H | METHOD FOR TREATING DISORDERS OF THE CENTRAL NERVOUS SYSTEM WITH A LOW-DOSED COMBINATION OF ESCITALOPRAM AND BUPROPION |
| US20090176882A1 (en) | 2008-12-09 | 2009-07-09 | Depomed, Inc. | Gastric retentive gabapentin dosage forms and methods for using same |
| US20070202164A1 (en) * | 2006-02-28 | 2007-08-30 | Hutchison Medipharma Enterprises Limited | Andrographis Extract Formulations |
| WO2010026467A2 (en) | 2008-09-04 | 2010-03-11 | Torrent Pharmaceuticals Ltd. | Controlled release dosage form of high solubility active ingredient |
| US9901551B2 (en) | 2009-04-20 | 2018-02-27 | Ambra Bioscience Llc | Chemosensory receptor ligand-based therapies |
| CN102481276A (zh) | 2009-04-20 | 2012-05-30 | 埃尔舍利克斯治疗公司 | 基于化学感受受体配体的治疗法 |
| US8828953B2 (en) | 2009-04-20 | 2014-09-09 | NaZura BioHealth, Inc. | Chemosensory receptor ligand-based therapies |
| WO2012054523A2 (en) | 2010-10-19 | 2012-04-26 | Elcelyx Therapeutics, Inc. | Chemosensory receptor ligand-based therapies |
| CA2823397C (en) | 2011-01-07 | 2020-03-10 | Elcelyx Therapeutics, Inc. | Chemosensory receptor ligand-based therapies |
| US20130143867A1 (en) | 2011-12-02 | 2013-06-06 | Sychroneuron Inc. | Acamprosate formulations, methods of using the same, and combinations comprising the same |
| WO2013158928A2 (en) | 2012-04-18 | 2013-10-24 | Elcelyx Therapeutics, Inc. | Chemosensory receptor ligand-based therapies |
| EP3878445A3 (en) | 2013-06-05 | 2021-10-27 | Synchroneuron Inc. | Acamprosate formulations, methods of using the same, and combinations comprising the same |
| US9617230B2 (en) | 2014-12-22 | 2017-04-11 | Farmington Pharma Development | Creatine prodrugs, compositions and methods of use thereof |
| US11332438B2 (en) | 2017-12-01 | 2022-05-17 | Ultragenyx Pharmaceutical Inc. | Creatine prodrugs, compositions and methods of use thereof |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5252338A (en) * | 1991-06-27 | 1993-10-12 | Alza Corporation | Therapy delayed |
-
1996
- 1996-02-16 MY MYPI96000592A patent/MY113429A/en unknown
- 1996-02-26 AR ARP960101520A patent/AR003928A1/es unknown
- 1996-02-28 WO PCT/US1996/002290 patent/WO1996026718A2/en not_active Ceased
- 1996-02-28 CA CA002213455A patent/CA2213455A1/en not_active Abandoned
- 1996-02-28 DE DE69625189T patent/DE69625189D1/de not_active Expired - Lifetime
- 1996-02-28 JP JP8526317A patent/JPH11509169A/ja not_active Ceased
- 1996-02-28 AT AT96908487T patent/ATE228829T1/de not_active IP Right Cessation
- 1996-02-28 AU AU51711/96A patent/AU722741B2/en not_active Ceased
- 1996-02-28 EP EP96908487A patent/EP0821582B1/en not_active Expired - Lifetime
- 1996-02-29 TW TW085102434A patent/TW431891B/zh not_active IP Right Cessation
- 1996-11-08 PA PA19968388101A patent/PA8388101A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPH11509169A (ja) | 1999-08-17 |
| AU5171196A (en) | 1996-09-18 |
| EP0821582A2 (en) | 1998-02-04 |
| PA8388101A1 (es) | 1997-09-30 |
| AU722741B2 (en) | 2000-08-10 |
| MY113429A (en) | 2002-02-28 |
| CA2213455A1 (en) | 1996-09-06 |
| WO1996026718A3 (en) | 1996-10-10 |
| EP0821582B1 (en) | 2002-12-04 |
| WO1996026718A2 (en) | 1996-09-06 |
| DE69625189D1 (de) | 2003-01-16 |
| TW431891B (en) | 2001-05-01 |
| ATE228829T1 (de) | 2002-12-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |