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AR004703A1 - Hidrazidil, bis-hidrazil y bis-aminometil-carbonil, inhibidores de proteasas, una composicin farmaceutica, metodo para inhibir proteasas, y uso en la preparacion de medicamentos. - Google Patents

Hidrazidil, bis-hidrazil y bis-aminometil-carbonil, inhibidores de proteasas, una composicin farmaceutica, metodo para inhibir proteasas, y uso en la preparacion de medicamentos.

Info

Publication number
AR004703A1
AR004703A1 ARP960104972A ARP960104972A AR004703A1 AR 004703 A1 AR004703 A1 AR 004703A1 AR P960104972 A ARP960104972 A AR P960104972A AR P960104972 A ARP960104972 A AR P960104972A AR 004703 A1 AR004703 A1 AR 004703A1
Authority
AR
Argentina
Prior art keywords
bis
preparation
hydrazidil
hydrazil
aminometil
Prior art date
Application number
ARP960104972A
Other languages
English (en)
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of AR004703A1 publication Critical patent/AR004703A1/es

Links

Classifications

    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Compuestos de fórmula (I) que inhiben proteasas, con inclusión de catepsina K, composiciones farmacéuticas que dichos compuestos y uso de dichos compuestosen la preparación de medicamentos para el tratamiento de enfermedades de pérdida ósea odegradación de cartílago o matriz excesivas, con inclusión deosteoporosis; enfermedad gingival con inclusión de gingivitis y periodontitis; artritis, más específicamente, osteoartritis y artritis reumatoide; enfermedadde Paget, hipercalcemia decará cter maligno; y enfermedad metabólica ósea, donde la definición de los sustituyentes son tal como figuran en la memoria.
ARP960104972A 1995-10-30 1996-10-30 Hidrazidil, bis-hidrazil y bis-aminometil-carbonil, inhibidores de proteasas, una composicin farmaceutica, metodo para inhibir proteasas, y uso en la preparacion de medicamentos. AR004703A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US810895P 1995-10-30 1995-10-30
US747395P 1995-11-22 1995-11-22
US899295P 1995-12-21 1995-12-21
US1374896P 1996-03-20 1996-03-20

Publications (1)

Publication Number Publication Date
AR004703A1 true AR004703A1 (es) 1999-03-10

Family

ID=27485695

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP960104972A AR004703A1 (es) 1995-10-30 1996-10-30 Hidrazidil, bis-hidrazil y bis-aminometil-carbonil, inhibidores de proteasas, una composicin farmaceutica, metodo para inhibir proteasas, y uso en la preparacion de medicamentos.

Country Status (2)

Country Link
AR (1) AR004703A1 (es)
BR (1) BR9612344A (es)

Also Published As

Publication number Publication date
BR9612344A (pt) 1999-07-13

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal
FB Suspension of granting procedure