AR004113A1 - Inhibidores de actividad de enzima rotamasa. - Google Patents
Inhibidores de actividad de enzima rotamasa.Info
- Publication number
- AR004113A1 AR004113A1 ARP960104917A ARP960104917A AR004113A1 AR 004113 A1 AR004113 A1 AR 004113A1 AR P960104917 A ARP960104917 A AR P960104917A AR P960104917 A ARP960104917 A AR P960104917A AR 004113 A1 AR004113 A1 AR 004113A1
- Authority
- AR
- Argentina
- Prior art keywords
- enzyme activity
- rotamasa
- activity inhibitors
- inhibitors
- immunophilins
- Prior art date
Links
- 102000004190 Enzymes Human genes 0.000 title abstract 3
- 108090000790 Enzymes Proteins 0.000 title abstract 3
- 230000000694 effects Effects 0.000 title abstract 3
- 239000003112 inhibitor Substances 0.000 title abstract 3
- 102000000521 Immunophilins Human genes 0.000 abstract 2
- 108010016648 Immunophilins Proteins 0.000 abstract 2
- 101710103508 FK506-binding protein Proteins 0.000 abstract 1
- 101710104425 FK506-binding protein 2 Proteins 0.000 abstract 1
- 101710104423 FK506-binding protein 3 Proteins 0.000 abstract 1
- 101710104333 FK506-binding protein 4 Proteins 0.000 abstract 1
- 101710104342 FK506-binding protein 5 Proteins 0.000 abstract 1
- 101710149710 FKBP-type 16 kDa peptidyl-prolyl cis-trans isomerase Proteins 0.000 abstract 1
- 101710121306 FKBP-type 22 kDa peptidyl-prolyl cis-trans isomerase Proteins 0.000 abstract 1
- 101710180800 FKBP-type peptidyl-prolyl cis-trans isomerase FkpA Proteins 0.000 abstract 1
- HXEACLLIILLPRG-YFKPBYRVSA-N L-pipecolic acid Chemical compound [O-]C(=O)[C@@H]1CCCC[NH2+]1 HXEACLLIILLPRG-YFKPBYRVSA-N 0.000 abstract 1
- 101710104030 Long-type peptidyl-prolyl cis-trans isomerase Proteins 0.000 abstract 1
- 101710114693 Outer membrane protein MIP Proteins 0.000 abstract 1
- 101710116692 Peptidyl-prolyl cis-trans isomerase Proteins 0.000 abstract 1
- 101710111764 Peptidyl-prolyl cis-trans isomerase FKBP10 Proteins 0.000 abstract 1
- 101710111749 Peptidyl-prolyl cis-trans isomerase FKBP11 Proteins 0.000 abstract 1
- 101710111747 Peptidyl-prolyl cis-trans isomerase FKBP12 Proteins 0.000 abstract 1
- 101710111757 Peptidyl-prolyl cis-trans isomerase FKBP14 Proteins 0.000 abstract 1
- 101710111682 Peptidyl-prolyl cis-trans isomerase FKBP1A Proteins 0.000 abstract 1
- 101710111689 Peptidyl-prolyl cis-trans isomerase FKBP1B Proteins 0.000 abstract 1
- 101710147154 Peptidyl-prolyl cis-trans isomerase FKBP2 Proteins 0.000 abstract 1
- 101710147149 Peptidyl-prolyl cis-trans isomerase FKBP3 Proteins 0.000 abstract 1
- 101710147152 Peptidyl-prolyl cis-trans isomerase FKBP4 Proteins 0.000 abstract 1
- 101710147150 Peptidyl-prolyl cis-trans isomerase FKBP5 Proteins 0.000 abstract 1
- 101710147138 Peptidyl-prolyl cis-trans isomerase FKBP7 Proteins 0.000 abstract 1
- 101710147137 Peptidyl-prolyl cis-trans isomerase FKBP8 Proteins 0.000 abstract 1
- 101710147136 Peptidyl-prolyl cis-trans isomerase FKBP9 Proteins 0.000 abstract 1
- 102100038809 Peptidyl-prolyl cis-trans isomerase FKBP9 Human genes 0.000 abstract 1
- 101710174853 Peptidyl-prolyl cis-trans isomerase Mip Proteins 0.000 abstract 1
- 101710200991 Peptidyl-prolyl cis-trans isomerase, rhodopsin-specific isozyme Proteins 0.000 abstract 1
- 101710092145 Peptidyl-prolyl cis-trans isomerase-like 1 Proteins 0.000 abstract 1
- 101710092146 Peptidyl-prolyl cis-trans isomerase-like 2 Proteins 0.000 abstract 1
- 101710092148 Peptidyl-prolyl cis-trans isomerase-like 3 Proteins 0.000 abstract 1
- 101710092149 Peptidyl-prolyl cis-trans isomerase-like 4 Proteins 0.000 abstract 1
- 102000009658 Peptidylprolyl Isomerase Human genes 0.000 abstract 1
- 108010020062 Peptidylprolyl Isomerase Proteins 0.000 abstract 1
- 101710113444 Probable parvulin-type peptidyl-prolyl cis-trans isomerase Proteins 0.000 abstract 1
- 101710090737 Probable peptidyl-prolyl cis-trans isomerase Proteins 0.000 abstract 1
- 101710133309 Putative peptidyl-prolyl cis-trans isomerase Proteins 0.000 abstract 1
- 101710124237 Short-type peptidyl-prolyl cis-trans isomerase Proteins 0.000 abstract 1
- 102000018679 Tacrolimus Binding Proteins Human genes 0.000 abstract 1
- 108010027179 Tacrolimus Binding Proteins Proteins 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- HXEACLLIILLPRG-RXMQYKEDSA-N l-pipecolic acid Natural products OC(=O)[C@H]1CCCCN1 HXEACLLIILLPRG-RXMQYKEDSA-N 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000007514 neuronal growth Effects 0.000 abstract 1
- 230000009689 neuronal regeneration Effects 0.000 abstract 1
- 230000000508 neurotrophic effect Effects 0.000 abstract 1
- 238000011069 regeneration method Methods 0.000 abstract 1
Landscapes
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere al método de usar compuestos neurotróficos derivados del ácido pipecólico que tienen afinidad con inmunofilinas del tipoFKBP como inhibidores de actividad de enzima relacionada con proteínas inmunifilinas, yparticularmente inhibidores de actividad de enzima peptidil-prolil isomerasa o rotamasa para estimular o promover el crecimiento o regeneración neuronal.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/653,905 US5696135A (en) | 1995-06-07 | 1996-05-28 | Inhibitors of rotamase enzyme activity effective at stimulating neuronal growth |
| PCT/US1996/009561 WO1996040140A1 (en) | 1995-06-07 | 1996-06-05 | Inhibitors of rotamase enzyme activity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR004113A1 true AR004113A1 (es) | 1998-09-30 |
Family
ID=24622745
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP960104917A AR004113A1 (es) | 1996-05-28 | 1996-10-25 | Inhibidores de actividad de enzima rotamasa. |
Country Status (3)
| Country | Link |
|---|---|
| AR (1) | AR004113A1 (es) |
| ID (1) | ID16708A (es) |
| ZA (1) | ZA968981B (es) |
-
1996
- 1996-10-25 ZA ZA9608981A patent/ZA968981B/xx unknown
- 1996-10-25 ID IDP963063A patent/ID16708A/id unknown
- 1996-10-25 AR ARP960104917A patent/AR004113A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA968981B (en) | 1998-05-25 |
| ID16708A (id) | 1997-11-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |