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NO996108L - 9-oksinerytromycinderivater - Google Patents

9-oksinerytromycinderivater

Info

Publication number
NO996108L
NO996108L NO996108A NO996108A NO996108L NO 996108 L NO996108 L NO 996108L NO 996108 A NO996108 A NO 996108A NO 996108 A NO996108 A NO 996108A NO 996108 L NO996108 L NO 996108L
Authority
NO
Norway
Prior art keywords
compounds
formula
disclosed
methods
oksinerytromycinderivater
Prior art date
Application number
NO996108A
Other languages
English (en)
Norwegian (no)
Other versions
NO996108D0 (no
Inventor
Yong-Jin Wu
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO996108D0 publication Critical patent/NO996108D0/no
Publication of NO996108L publication Critical patent/NO996108L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
NO996108A 1997-06-11 1999-12-10 9-oksinerytromycinderivater NO996108L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4934997P 1997-06-11 1997-06-11
PCT/IB1998/000741 WO1998056800A1 (en) 1997-06-11 1998-05-15 9-oxime erythromycin derivatives

Publications (2)

Publication Number Publication Date
NO996108D0 NO996108D0 (no) 1999-12-10
NO996108L true NO996108L (no) 2000-02-10

Family

ID=21959341

Family Applications (1)

Application Number Title Priority Date Filing Date
NO996108A NO996108L (no) 1997-06-11 1999-12-10 9-oksinerytromycinderivater

Country Status (31)

Country Link
EP (1) EP0988308A1 (pt)
JP (1) JP2000513026A (pt)
KR (1) KR20010013660A (pt)
CN (1) CN1259135A (pt)
AP (1) AP9801253A0 (pt)
AR (1) AR012244A1 (pt)
AU (1) AU7226798A (pt)
BG (1) BG103947A (pt)
BR (1) BR9810021A (pt)
CA (1) CA2293335A1 (pt)
CO (1) CO4940506A1 (pt)
CZ (1) CZ9904388A3 (pt)
EA (1) EA199901016A1 (pt)
GT (1) GT199800074A (pt)
HN (1) HN1998000073A (pt)
HR (1) HRP980316A2 (pt)
HU (1) HUP0002252A3 (pt)
ID (1) ID24529A (pt)
IL (1) IL132767A0 (pt)
IS (1) IS5251A (pt)
MA (1) MA26505A1 (pt)
NO (1) NO996108L (pt)
OA (1) OA11225A (pt)
PA (1) PA8451801A1 (pt)
PE (1) PE79899A1 (pt)
PL (1) PL337606A1 (pt)
TN (1) TNSN98083A1 (pt)
TR (1) TR199902995T2 (pt)
TW (1) TW448174B (pt)
WO (1) WO1998056800A1 (pt)
ZA (1) ZA985018B (pt)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000159A (es) * 1997-10-29 1999-02-09 Monsanto Co Derivados de 9- amino - 3 ceto eritromicina
ATE298761T1 (de) * 1998-09-22 2005-07-15 Pfizer Prod Inc Carbamat- und carbazatketolidantibiotika
FR2786188B1 (fr) * 1998-11-24 2002-10-31 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments
US6258785B1 (en) 1998-12-02 2001-07-10 Pfizer Inc. Crystalline 9-E-(O-methyl)oxime of 11, 12-dideoxy-3-de(2,6-dideoxy-3-C-methyl-3-O-methyl-α-L-ribohexopyranosyloxy)-6-O-methyl-12,11-(iminocarbonyl-(2-(3-(4-(3-pyridinyl)1H-imadazol-1-yl)propyl)hydrazono))-3-oxoerythromycin
EP1298138B1 (en) * 1998-12-10 2006-11-02 Pfizer Products Inc. Carbamate and Carbazate Ketolide Antibiotics
US6284732B1 (en) * 1998-12-18 2001-09-04 Bio-Rad Laboratories, Inc. Peptides and peptide analogues designed from HFE protein and their uses in the treatment of iron overload diseases
NZ515027A (en) * 1999-04-16 2004-01-30 Kosan Biosciences Inc Erythromycin derivatives as antibiotics
CN1351608A (zh) 1999-05-24 2002-05-29 辉瑞产品公司 13－甲基红霉素衍生物
EP1181300B1 (en) * 1999-06-07 2003-09-17 Abbott Laboratories 6-o-carbamate ketolide derivatives
ID27331A (id) * 1999-09-29 2001-03-29 Pfizer Prod Inc Pembuatan antibiotik-antibiotik ketolida karbamat
EP1439186A3 (en) * 1999-12-29 2004-11-03 Pfizer Products Inc. Intermediates for novel antibacterial and prokinetic macrolides
EP1114826A3 (en) * 1999-12-29 2001-10-31 Pfizer Products Inc. Novel antibacterial and prokinetic macrolides
US6946446B2 (en) 2000-02-24 2005-09-20 Abbott Laboratories Anti-infective agents useful against multidrug-resistant strains of bacteria
US6403776B1 (en) 2000-07-05 2002-06-11 Pfizer Inc. Synthesis of carbamate ketolide antibiotics
WO2003090761A1 (en) * 2002-04-25 2003-11-06 Abbott Laboratories 9-oxime macrolide antibacterials
US7091196B2 (en) 2002-09-26 2006-08-15 Rib-X Pharmaceuticals, Inc. Bifunctional heterocyclic compounds and methods of making and using same
EP3738591A3 (en) * 2003-03-10 2021-03-24 Merck Sharp & Dohme Corp. Novel antibacterial agents
US8202843B2 (en) 2004-02-27 2012-06-19 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same
WO2009055557A1 (en) 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
DK2358379T3 (en) 2008-10-24 2016-03-07 Cempra Pharmaceuticals Inc BIOFORSVAR USING TRIAZOLHOLDIGE macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
EP2475253B1 (en) 2009-09-10 2016-10-26 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and mac diseases
CN102146085B (zh) * 2010-02-09 2014-03-26 北京理工大学 一种9-肟醚酮内酯衍生物、制备方法及其药物组合物
JP5711352B2 (ja) 2010-03-22 2015-04-30 センプラ ファーマシューティカルズ，インコーポレイテッド マクロライドの結晶形、およびその使用
WO2011146829A1 (en) 2010-05-20 2011-11-24 Cempra Pharmaceuticals, Inc. Processes for preparing macrolides and ketolides and intermediates therefor
US9815863B2 (en) 2010-09-10 2017-11-14 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
US10188674B2 (en) 2012-03-27 2019-01-29 Cempra Pharmaceuticals, Inc. Parenteral formulations for administering macrolide antibiotics
EP2968801B1 (en) 2013-03-14 2018-09-26 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
CN105188712A (zh) 2013-03-15 2015-12-23 森普拉制药公司 用于制备大环内酯抗菌剂的收敛方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of erythromycin derivatives
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2718450B1 (fr) * 1994-04-08 1997-01-10 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
BR9810021A (pt) 2000-09-19
IS5251A (is) 1999-11-16
IL132767A0 (en) 2001-03-19
JP2000513026A (ja) 2000-10-03
ZA985018B (en) 1999-12-10
NO996108D0 (no) 1999-12-10
TNSN98083A1 (fr) 2005-03-15
PL337606A1 (en) 2000-08-28
CN1259135A (zh) 2000-07-05
AR012244A1 (es) 2000-09-27
PE79899A1 (es) 1999-08-25
OA11225A (en) 2003-07-17
GT199800074A (es) 1999-11-27
HUP0002252A3 (en) 2002-01-28
HRP980316A2 (en) 1999-04-30
PA8451801A1 (es) 2000-05-24
BG103947A (en) 2000-07-31
HUP0002252A2 (hu) 2000-12-28
EP0988308A1 (en) 2000-03-29
AP9801253A0 (en) 1999-12-04
TR199902995T2 (xx) 2000-02-21
MA26505A1 (fr) 2004-12-20
TW448174B (en) 2001-08-01
CO4940506A1 (es) 2000-07-24
CA2293335A1 (en) 1998-12-17
EA199901016A1 (ru) 2000-06-26
AU7226798A (en) 1998-12-30
CZ9904388A3 (cs) 2002-10-16
WO1998056800A1 (en) 1998-12-17
KR20010013660A (ko) 2001-02-26
ID24529A (id) 2000-07-20
HN1998000073A (es) 1999-01-08

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application