NO981813L - Mellomprodukter til bruk ved fremstilling av taxanderivater - Google Patents
Mellomprodukter til bruk ved fremstilling av taxanderivaterInfo
- Publication number
- NO981813L NO981813L NO981813A NO981813A NO981813L NO 981813 L NO981813 L NO 981813L NO 981813 A NO981813 A NO 981813A NO 981813 A NO981813 A NO 981813A NO 981813 L NO981813 L NO 981813L
- Authority
- NO
- Norway
- Prior art keywords
- radical
- taxane derivatives
- phenyl
- intermediates
- preparation
- Prior art date
Links
- DKPFODGZWDEEBT-QFIAKTPHSA-N taxane Chemical class C([C@]1(C)CCC[C@@H](C)[C@H]1C1)C[C@H]2[C@H](C)CC[C@@H]1C2(C)C DKPFODGZWDEEBT-QFIAKTPHSA-N 0.000 title abstract 3
- 239000000543 intermediate Substances 0.000 title 1
- 150000003254 radicals Chemical group 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000006239 protecting group Chemical group 0.000 abstract 2
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical group [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
- TUCNEACPLKLKNU-UHFFFAOYSA-N acetyl Chemical compound C[C]=O TUCNEACPLKLKNU-UHFFFAOYSA-N 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000005036 alkoxyphenyl group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 150000005840 aryl radicals Chemical class 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
- 125000003884 phenylalkyl group Chemical group 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9213000A FR2697522B1 (fr) | 1992-10-30 | 1992-10-30 | Procédé de préparation de dérivés du taxane. |
| PCT/FR1993/001058 WO1994010169A1 (fr) | 1992-10-30 | 1993-10-28 | Procede de preparation de derives du taxane |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO981813L true NO981813L (no) | 1995-04-26 |
| NO981813D0 NO981813D0 (no) | 1998-04-22 |
| NO306062B1 NO306062B1 (no) | 1999-09-13 |
Family
ID=9435013
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO951587A NO304114B1 (no) | 1992-10-30 | 1995-04-26 | Taxanderivater og fremstilling derav |
| NO981813A NO306062B1 (no) | 1992-10-30 | 1998-04-22 | Syremellomprodukter til bruk ved fremstilling av taxanderivater |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO951587A NO304114B1 (no) | 1992-10-30 | 1995-04-26 | Taxanderivater og fremstilling derav |
Country Status (24)
| Country | Link |
|---|---|
| US (3) | US5686623A (no) |
| EP (1) | EP0666857B1 (no) |
| JP (1) | JP3030088B2 (no) |
| KR (1) | KR100255460B1 (no) |
| AT (1) | ATE180258T1 (no) |
| AU (1) | AU679947B2 (no) |
| CA (1) | CA2148103C (no) |
| CZ (1) | CZ287805B6 (no) |
| DE (1) | DE69325031T2 (no) |
| DK (1) | DK0666857T3 (no) |
| ES (1) | ES2133418T3 (no) |
| FI (1) | FI109798B (no) |
| FR (1) | FR2697522B1 (no) |
| GR (1) | GR3030268T3 (no) |
| HU (1) | HUT73780A (no) |
| MX (1) | MX9306606A (no) |
| NO (2) | NO304114B1 (no) |
| NZ (1) | NZ257578A (no) |
| PL (1) | PL177746B1 (no) |
| RU (2) | RU2188198C2 (no) |
| SK (1) | SK281045B6 (no) |
| TW (1) | TW427988B (no) |
| WO (1) | WO1994010169A1 (no) |
| ZA (1) | ZA938012B (no) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL107950A (en) | 1992-12-15 | 2001-04-30 | Upjohn Co | 7β, 8β - METHANO-TAXOLS, THEIR PREPARATION AND ANTINEOPLASTIC PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| AU7138894A (en) * | 1993-06-11 | 1995-01-03 | Pharmacia & Upjohn Company | Delta 6,7--taxols antineoplastic use and pharmaceutical compositions containing them |
| IL127597A (en) * | 1994-01-28 | 2003-07-31 | Upjohn Co | Iso-taxol analogs |
| CA2170661A1 (en) | 1995-03-22 | 1996-09-23 | John K. Thottathil | Novel methods for the preparation of taxanes using oaxzolidine intermediates |
| EP1099696A3 (en) * | 1995-06-06 | 2001-05-23 | Dr. Reddy's Research Foundation | Preparation of oxazolidine |
| AU4768797A (en) * | 1996-10-24 | 1998-05-15 | Institute Armand-Frappier | A family of canadensol taxanes, the semi-synthetic preparation and therapeutic use thereof |
| US6150537A (en) * | 1997-12-12 | 2000-11-21 | Emory University | Methods for the esterification of alcohols and compounds useful therefor as potential anticancer agents |
| EP0982028A1 (en) * | 1998-08-20 | 2000-03-01 | Aventis Pharma S.A. | New use of taxoid derivatives |
| EP1105119A2 (en) * | 1998-08-20 | 2001-06-13 | Aventis Pharma S.A. | New use of taxoid derivatives |
| JP4502338B2 (ja) * | 1999-09-17 | 2010-07-14 | 株式会社横浜国際バイオ研究所 | タキソイド化合物の製造法 |
| EP2289549A3 (en) | 1999-10-01 | 2011-06-15 | Immunogen, Inc. | Immunoconjugates for treating cancer |
| AU2000261768A1 (en) * | 2000-08-08 | 2002-02-18 | Dr. Reddy's Research Foundation | An improved process for the preparation of docetaxel |
| JP2002088935A (ja) | 2000-09-14 | 2002-03-27 | Nichiha Corp | 外装材の縦目地ジョイナー |
| US8338617B2 (en) | 2004-11-19 | 2012-12-25 | Dr. Reddy's Laboratories Limited | Process for preparing oxazolidine derivatives |
| CZ298332B6 (cs) * | 2005-09-26 | 2007-08-29 | Zentiva, A. S | Zpusob prípravy kyseliny (4S,5R)-2,4-difenyloxazolin-4,5-dihydro-5-karboxylové |
| CA2634746A1 (en) * | 2005-12-21 | 2007-07-05 | Tapestry Pharmaceuticals, Inc. | Processes for taxane derivatives and intermediates useful therein |
| WO2008074178A1 (fr) * | 2006-11-23 | 2008-06-26 | Shanghai Bailing Pharmaceutical Technology Co., Ltd | Nouveau procédé de préparation de paclitaxel semi-synthétique |
| CN101020672B (zh) * | 2006-12-28 | 2010-08-25 | 上海百灵医药科技有限公司 | 多烯紫杉醇的合成方法 |
| PL388144A1 (pl) | 2009-05-29 | 2010-12-06 | Przedsiębiorstwo Produkcyjno-Wdrożeniowe Ifotam Spółka Z Ograniczoną Odpowiedzialnością | Solwaty (2R,3S)-3-tert-butoksykarbonylamino-2-hydroksy-3-fenylopropionianu 4-acetoksy-2α-benzoiloksy -5β,20-epoksy-1,7β,10β-trihydroksy-9-okso-taks-11-en-13α-ylu, sposób ich otrzymywania i zastosowanie |
| KR101379694B1 (ko) * | 2011-09-30 | 2014-03-31 | 주식회사 삼양바이오팜 | 탁산유도체의 제조방법 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2629819B1 (fr) * | 1988-04-06 | 1990-11-16 | Rhone Poulenc Sante | Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii |
| MX9102128A (es) * | 1990-11-23 | 1992-07-08 | Rhone Poulenc Rorer Sa | Derivados de taxano,procedimiento para su preparacion y composicion farmaceutica que los contiene |
| FR2696464B1 (fr) * | 1992-10-05 | 1994-11-10 | Rhone Poulenc Rorer Sa | Nouveau procédé d'estérification de la baccatine III et de la désacétyl-10 baccatine III. |
| FR2696459B1 (fr) * | 1992-10-05 | 1994-11-25 | Rhone Poulenc Rorer Sa | Procédé de préparation de dérivés du taxane. |
| FR2696460B1 (fr) * | 1992-10-05 | 1994-11-25 | Rhone Poulenc Rorer Sa | Procédé de préparation de dérivés du taxane. |
| FR2696458B1 (fr) * | 1992-10-05 | 1994-11-10 | Rhone Poulenc Rorer Sa | Procédé de préparation de dérivés du taxane. |
| AU7138894A (en) * | 1993-06-11 | 1995-01-03 | Pharmacia & Upjohn Company | Delta 6,7--taxols antineoplastic use and pharmaceutical compositions containing them |
-
1992
- 1992-10-30 FR FR9213000A patent/FR2697522B1/fr not_active Expired - Fee Related
-
1993
- 1993-10-25 MX MX9306606A patent/MX9306606A/es not_active IP Right Cessation
- 1993-10-27 ZA ZA938012A patent/ZA938012B/xx unknown
- 1993-10-28 JP JP6510775A patent/JP3030088B2/ja not_active Expired - Lifetime
- 1993-10-28 WO PCT/FR1993/001058 patent/WO1994010169A1/fr not_active Ceased
- 1993-10-28 DK DK93924646T patent/DK0666857T3/da active
- 1993-10-28 US US08/424,386 patent/US5686623A/en not_active Expired - Fee Related
- 1993-10-28 AT AT93924646T patent/ATE180258T1/de not_active IP Right Cessation
- 1993-10-28 HU HU9501235A patent/HUT73780A/hu unknown
- 1993-10-28 CZ CZ19951092A patent/CZ287805B6/cs not_active IP Right Cessation
- 1993-10-28 CA CA002148103A patent/CA2148103C/fr not_active Expired - Fee Related
- 1993-10-28 SK SK557-95A patent/SK281045B6/sk unknown
- 1993-10-28 RU RU98103160/04A patent/RU2188198C2/ru not_active IP Right Cessation
- 1993-10-28 EP EP93924646A patent/EP0666857B1/fr not_active Expired - Lifetime
- 1993-10-28 ES ES93924646T patent/ES2133418T3/es not_active Expired - Lifetime
- 1993-10-28 RU RU95111381/04A patent/RU2118958C1/ru not_active IP Right Cessation
- 1993-10-28 KR KR1019950701766A patent/KR100255460B1/ko not_active Expired - Fee Related
- 1993-10-28 NZ NZ257578A patent/NZ257578A/en unknown
- 1993-10-28 AU AU54237/94A patent/AU679947B2/en not_active Ceased
- 1993-10-28 PL PL93308638A patent/PL177746B1/pl unknown
- 1993-10-28 TW TW082109008A patent/TW427988B/zh not_active IP Right Cessation
- 1993-10-28 DE DE69325031T patent/DE69325031T2/de not_active Expired - Fee Related
-
1995
- 1995-04-26 NO NO951587A patent/NO304114B1/no not_active IP Right Cessation
- 1995-04-28 FI FI952059A patent/FI109798B/fi active
-
1997
- 1997-08-08 US US08/908,807 patent/US6433180B1/en not_active Expired - Fee Related
-
1998
- 1998-04-22 NO NO981813A patent/NO306062B1/no not_active IP Right Cessation
-
1999
- 1999-05-20 GR GR990400398T patent/GR3030268T3/el unknown
-
2002
- 2002-06-26 US US10/179,027 patent/US20030013889A1/en not_active Abandoned
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |