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NO971946D0 - Fenyloksazolidinon-antimikrobielle midler - Google Patents

Fenyloksazolidinon-antimikrobielle midler

Info

Publication number
NO971946D0
NO971946D0 NO971946A NO971946A NO971946D0 NO 971946 D0 NO971946 D0 NO 971946D0 NO 971946 A NO971946 A NO 971946A NO 971946 A NO971946 A NO 971946A NO 971946 D0 NO971946 D0 NO 971946D0
Authority
NO
Norway
Prior art keywords
antimicrobial agents
phenyloxazolidinone
species
bacteroids
enterococci
Prior art date
Application number
NO971946A
Other languages
English (en)
Other versions
NO971946L (no
NO309478B1 (no
Inventor
Douglas K Hutchinson
Michael Robert Barbachyn
Mikio Taniguchi
Kiyotaka Munesada
Hiroyoshi Yamada
Steven J Brickner
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of NO971946D0 publication Critical patent/NO971946D0/no
Publication of NO971946L publication Critical patent/NO971946L/no
Publication of NO309478B1 publication Critical patent/NO309478B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO971946A 1994-10-26 1997-04-25 Fenyloksazolidinon-antimikrobielle midler NO309478B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32971794A 1994-10-26 1994-10-26
PCT/US1995/010992 WO1996013502A1 (en) 1994-10-26 1995-09-12 Phenyloxazolidinone antimicrobials

Publications (3)

Publication Number Publication Date
NO971946D0 true NO971946D0 (no) 1997-04-25
NO971946L NO971946L (no) 1997-06-25
NO309478B1 NO309478B1 (no) 2001-02-05

Family

ID=23286694

Family Applications (1)

Application Number Title Priority Date Filing Date
NO971946A NO309478B1 (no) 1994-10-26 1997-04-25 Fenyloksazolidinon-antimikrobielle midler

Country Status (22)

Country Link
EP (1) EP0788498B1 (no)
JP (1) JP3933198B2 (no)
KR (1) KR100383403B1 (no)
CN (1) CN1068325C (no)
AT (1) ATE204277T1 (no)
AU (1) AU694271B2 (no)
BR (1) BR9509136A (no)
CA (1) CA2200433C (no)
CZ (1) CZ291847B6 (no)
DE (1) DE69522234T2 (no)
DK (1) DK0788498T3 (no)
ES (1) ES2162941T3 (no)
FI (1) FI971774A0 (no)
HU (1) HU224044B1 (no)
NO (1) NO309478B1 (no)
NZ (1) NZ293741A (no)
PL (1) PL183512B1 (no)
PT (1) PT788498E (no)
RU (1) RU2134692C1 (no)
SI (1) SI0788498T1 (no)
SK (1) SK282869B6 (no)
WO (1) WO1996013502A1 (no)

Families Citing this family (45)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69631347T2 (de) * 1995-09-15 2004-10-07 Upjohn Co Aminoaryl oxazolidinone n-oxide
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
GB9702213D0 (en) 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
CZ298060B6 (cs) * 1996-04-11 2007-06-06 Pharmacia & Upjohn Company Zpusob prípravy oxazolidinonu
GB9609919D0 (en) 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
GB9717807D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9717804D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9725244D0 (en) 1997-11-29 1998-01-28 Zeneca Ltd Chemical compounds
US6562844B2 (en) 1998-01-23 2003-05-13 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
US7002020B1 (en) 1998-01-23 2006-02-21 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
CN1288462A (zh) 1998-01-23 2001-03-21 法玛西雅厄普约翰美国公司 噁唑烷酮组合库、组合物和制备方法
ES2182485T3 (es) * 1998-02-13 2003-03-01 Upjohn Co Derivados de aminofenil isosazolina sustituidos utiles como agentes antimicrobianos.
KR20010052615A (ko) 1998-06-05 2001-06-25 다비드 에 질레스 옥사졸리디논 유도체, 이것의 제조 방법 및 이것을함유하는 약학 조성물
WO2000051998A1 (en) 1999-03-02 2000-09-08 Boehringer Ingelheim Pharmaceuticals, Inc. Compounds useful as reversible inhibitors of cathepsin s
DE19919708A1 (de) * 1999-04-30 2001-03-01 Univ Stuttgart Stufenweise Alkylierung von polymeren Aminen
US6608081B2 (en) 1999-08-12 2003-08-19 Ortho-Mcneil Pharmaceutical, Inc. Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods
US6420364B1 (en) 1999-09-13 2002-07-16 Boehringer Ingelheim Pharmaceuticals, Inc. Compound useful as reversible inhibitors of cysteine proteases
FR2802091A1 (fr) * 1999-12-08 2001-06-15 Oreal Compositions pour la teinture des fibres keratiniques contenant des derives de paraphenylenediamine a groupement azetidinyle
ATE321024T1 (de) 2000-10-17 2006-04-15 Pharmacia & Upjohn Co Llc Verfahren zur herstellung von oxazolidinonverbindungen
YU52403A (sh) * 2000-12-26 2006-03-03 Dr.Reddy's Research Foundation Heterociklična jedinjenja koja imaju antibakterijsko dejstvo, postupak za njihovo dobijanje i farmaceutske smeše koje ih sadrže
US7160912B2 (en) 2000-12-26 2007-01-09 Dr.Reddy's Laboratories Ltd. Heterocyclic compounds having antibacterial activity: process for their preparation and pharmaceutical compositions containing them
EP1358185A2 (en) 2001-02-07 2003-11-05 Ortho-Mcneil Pharmaceutical, Inc. Pyridoarylphenyl oxazolidinone antibacterials, and related compositions and methods
ES2186550B2 (es) * 2001-06-27 2003-11-16 Vita Lab Nuevos derivados de oxazolidinonas como antibacterianos.
US6914058B2 (en) * 2002-01-18 2005-07-05 Dr. Reddy's Laboratories, Limited Antibacterial compounds: process for their preparation and pharmaceutical compositions containing them
AR038536A1 (es) 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
US7141588B2 (en) 2002-02-25 2006-11-28 Pfizer, Inc. N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
CA2492194A1 (en) * 2002-07-11 2004-01-22 Wockhardt Limited Antibacterial cyano-(substituted)-methylenepiperidinophenyl oxazolidinones targeting multiple ribonucleoproteins sites
EP1546140A2 (en) * 2002-07-11 2005-06-29 Wockhardt Limited Antimicrobial oxazolidinones, process of their preparation, and pharmaceutical compositions containing them
DE60304360T2 (de) 2002-08-12 2006-11-16 Pharmacia & Upjohn Co. Llc, Kalamazoo N-aryl-2-oxazolidinone und deren derivate
AR042086A1 (es) 2002-11-21 2005-06-08 Upjohn Co N-aril-2- oxazolidinon -5- carboxamidas y sus derivados, usados como agentes antibacterianos
US7223788B2 (en) 2003-02-14 2007-05-29 Sanofi-Aventis Deutschland Gmbh Substituted N-aryl heterocycles, process for their preparation and their use as medicaments
DE10306250A1 (de) * 2003-02-14 2004-09-09 Aventis Pharma Deutschland Gmbh Substituierte N-Arylheterozyklen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
US7687627B2 (en) * 2003-09-08 2010-03-30 Wockhardt Limited Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy
US7304050B2 (en) 2003-09-16 2007-12-04 Pfizer Inc. Antibacterial agents
FR2862969A1 (fr) * 2003-11-28 2005-06-03 Oreal Procede de preparation de derives paraphenylenediamine a groupement pyrrolidinyle, substitue par un radical azote, et composes intermediaires
WO2007004049A1 (en) * 2005-07-06 2007-01-11 Pharmacia & Upjohn Company Llc Oxazolidinones containing azetidine as antibacterial agents
WO2007004037A1 (en) * 2005-07-06 2007-01-11 Pharmacia & Upjohn Company Llc Oxazolidinone carboxamides containing azetidine and cyclobutane as antibacterial agents
US8952199B2 (en) 2007-07-24 2015-02-10 Dow Global Technologies Llc Methods of and formulations for reducing and inhibiting the growth of the concentration of microbes in water-based fluids and systems used with them
JP5368443B2 (ja) 2007-07-24 2013-12-18 ダウ グローバル テクノロジーズ エルエルシー 水系流体及び水系流体と共に用いられるシステム中の微生物濃度の増大を低減及び抑制するための方法及び配合物
EP2141162A1 (en) * 2008-07-01 2010-01-06 Ferrer Internacional, S.A. 3-(n-heterocyclyl)-pyrrolidinyl-phenyl-oxazolidinones as antibacterial agents
EP2141161A1 (en) * 2008-07-01 2010-01-06 Ferrer Internacional, S.A. 3-cyanopyrrolidinyl-phenyl-oxazolidinones as antibacterial agents
CN101798302B (zh) * 2009-02-06 2014-11-05 上海盟科药业有限公司 抗生素类药物1-(邻-氟苯基)二氢吡啶酮的合成及生产的方法和工艺
EP2635589A1 (en) 2010-11-03 2013-09-11 Wockhardt Limited Process for the preparation of phosphoric acid mono- (l-{4- [(s) -5- (acetylaminomethyl) - 2 - oxo - oxazolidin- 3 - yl]- 2, 6 - difluorophenyl} - 4 -methoxymethylpiperidin- 4 - yl) ester
WO2015173664A1 (en) 2014-05-14 2015-11-19 Wockhardt Limited Process for the preparation of (5s)-n-{3-[3,5-difluoro-4-(4-hydroxy-4-methoxymethyl-piperidin-1-yl)-phenyl]-2-oxo-oxazolidin-5-ylmethyl}-acetamide
WO2020234636A1 (en) 2019-05-17 2020-11-26 Cadila Healthcare Limited Novel compounds for the treatment of mammalian infections

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES8506659A1 (es) * 1983-06-07 1985-08-01 Du Pont Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno.
CA1317594C (en) * 1987-10-21 1993-05-11 Chung-Ho Park Aminomethyloxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents
US4948801A (en) * 1988-07-29 1990-08-14 E. I. Du Pont De Nemours And Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
EP0609905B1 (en) * 1988-09-15 2001-06-06 PHARMACIA & UPJOHN COMPANY 3-(Nitrogen substituted)phenyl-5beta-amidomethyloxazolidin-2-ones
KR100257418B1 (ko) * 1991-11-01 2000-05-15 로렌스 티. 마이젠헬더 치환된 아릴-및 헤테로아릴-페닐옥사졸리디논

Also Published As

Publication number Publication date
KR970707123A (ko) 1997-12-01
SI0788498T1 (en) 2001-12-31
ATE204277T1 (de) 2001-09-15
CA2200433A1 (en) 1996-05-09
DE69522234D1 (de) 2001-09-20
DE69522234T2 (de) 2002-05-16
NZ293741A (en) 1998-06-26
CN1162312A (zh) 1997-10-15
SK49497A3 (en) 1998-01-14
NO971946L (no) 1997-06-25
JP3933198B2 (ja) 2007-06-20
PL183512B1 (pl) 2002-06-28
AU3625495A (en) 1996-05-23
NO309478B1 (no) 2001-02-05
AU694271B2 (en) 1998-07-16
WO1996013502A1 (en) 1996-05-09
FI971774A7 (fi) 1997-04-25
CZ121797A3 (en) 1997-07-16
CZ291847B6 (cs) 2003-06-18
SK282869B6 (sk) 2003-01-09
FI971774A0 (fi) 1997-04-25
CN1068325C (zh) 2001-07-11
EP0788498B1 (en) 2001-08-16
ES2162941T3 (es) 2002-01-16
PT788498E (pt) 2002-02-28
DK0788498T3 (da) 2001-11-05
PL319873A1 (en) 1997-09-01
KR100383403B1 (ko) 2004-05-31
EP0788498A1 (en) 1997-08-13
CA2200433C (en) 2006-02-07
HU224044B1 (hu) 2005-05-30
BR9509136A (pt) 1998-07-21
RU2134692C1 (ru) 1999-08-20
JPH10508017A (ja) 1998-08-04
HUT77602A (hu) 1998-06-29

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