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NO974956L - Therapeutic composition for arthritis - Google Patents

Therapeutic composition for arthritis

Info

Publication number
NO974956L
NO974956L NO974956A NO974956A NO974956L NO 974956 L NO974956 L NO 974956L NO 974956 A NO974956 A NO 974956A NO 974956 A NO974956 A NO 974956A NO 974956 L NO974956 L NO 974956L
Authority
NO
Norway
Prior art keywords
arthritis
agent
administration
inflammatory
acting
Prior art date
Application number
NO974956A
Other languages
Norwegian (no)
Other versions
NO974956D0 (en
Inventor
Haruhiko Makino
Takashi Sohda
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of NO974956L publication Critical patent/NO974956L/en
Publication of NO974956D0 publication Critical patent/NO974956D0/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Det blir fremskaffet et farmasøytisk middel som viser hurtigvirkende og vedvarende anti-inflammatorisk analgesisk virkning mot kronisk artritis med lav fremtreden av bieffekter. En farmasøytisk sammensetning omfattende en kombinasjon av et quinolin-/quina- zolinserier profylaktisk/terapeutisk middel for artritis og hurtigvirkende anti-inflam- matorisk analgesisk middel omfattende (1) en cyklooksygenaseinhibitor, (2) et sentralt analgesika, (3) et steroid eller (4) et anti-inflammatorisk enzym-middel. Foreliggende preparat viser utmerkede effekter mot artritis fra administrasjon for å sikre stabil anti-inflammatorisk analgesisk virkning med lav fremtreden av bieffekter selv ved kronisk administrasjon, forutsatt at medikamentsammensetning, administrasjonsmetode og dose er passende valgt ifølge symptomene.A pharmaceutical agent is provided which shows fast-acting and sustained anti-inflammatory analgesic action against chronic arthritis with a low onset of side effects. A pharmaceutical composition comprising a combination of a quinoline / quinazoline series prophylactic / therapeutic agent for arthritis and fast-acting anti-inflammatory analgesic agent comprising (1) a cyclooxygenase inhibitor, (2) a central analgesic, (3) a steroid or ( 4) an anti-inflammatory enzyme agent. The present preparation shows excellent effects against arthritis from administration to ensure stable anti-inflammatory analgesic effect with low appearance of side effects even in chronic administration, provided that drug composition, administration method and dose are appropriately selected according to the symptoms.

NO974956A 1995-04-28 1997-10-27 Therapeutic composition for arthritis NO974956D0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP10631695 1995-04-28
JP27085695 1995-10-19
PCT/JP1996/001102 WO1996033717A1 (en) 1995-04-28 1996-04-24 Therapeutic composition for arthritis

Publications (2)

Publication Number Publication Date
NO974956L true NO974956L (en) 1997-10-27
NO974956D0 NO974956D0 (en) 1997-10-27

Family

ID=26446436

Family Applications (1)

Application Number Title Priority Date Filing Date
NO974956A NO974956D0 (en) 1995-04-28 1997-10-27 Therapeutic composition for arthritis

Country Status (7)

Country Link
EP (1) EP0830133A1 (en)
KR (1) KR19990008148A (en)
AU (1) AU715358B2 (en)
CA (1) CA2216138A1 (en)
HU (1) HUP9801628A2 (en)
NO (1) NO974956D0 (en)
WO (1) WO1996033717A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6262269B1 (en) 1997-02-04 2001-07-17 Trega Biosciences, Inc. 4-Substituted-quinoline derivatives and 4-substituted-quinoline combinatorial libraries
CA2279977A1 (en) * 1997-02-04 1998-08-06 John S. Kiely 4-substituted-quinoline derivatives and 4-substituted-quinoline combinatorial libraries
DE60129445T2 (en) 2000-08-09 2008-04-24 F. Hoffmann-La Roche Ag QUINOLINE DERIVATIVES AS AN ANTI-INFLAMMATORY AGENT
EP1354603A1 (en) * 2000-12-26 2003-10-22 Takeda Chemical Industries, Ltd. Concomitant drugs

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4968701A (en) * 1988-04-26 1990-11-06 E. I. Du Pont De Nemours And Company 4-Quinoline carboxylic acid derivatives useful as immunosuppressive agents
DE68908459T2 (en) * 1988-04-26 1994-04-07 Asahi Glass Co Ltd Prepolymer composition, process for its preparation and its use.
US5187180A (en) * 1990-07-26 1993-02-16 Merck Frosst Canada, Inc. (quinolin-2-ylmethoxy)heterotetrahydrocarbazoles as inhibitors of the biosynthesis of leukotrienes
IE920499A1 (en) * 1991-02-21 1992-08-26 Merck Frosst Canada Inc Quinoline-containing ketoacids as leukotriene antagonists
TW232013B (en) * 1992-04-24 1994-10-11 Takeda Pharm Industry Co Ltd
KR100224135B1 (en) * 1993-01-28 1999-10-15 다께다 구니오 Quinoline or quinazoline derivatives, preparations and uses thereof
US5641788A (en) * 1994-06-07 1997-06-24 Takeda Chemical Industries, Ltd. Quinoline derivatives and pharmaceutical composition containing them

Also Published As

Publication number Publication date
CA2216138A1 (en) 1996-10-31
AU715358B2 (en) 2000-01-20
WO1996033717A1 (en) 1996-10-31
KR19990008148A (en) 1999-01-25
AU5513696A (en) 1996-11-18
HUP9801628A2 (en) 1999-01-28
EP0830133A1 (en) 1998-03-25
NO974956D0 (en) 1997-10-27

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