NO954767D0 - 4-amino-17 delser som C17-20-lyase- og 5 - Google Patents

4-amino-17 delser som C17-20-lyase- og 5

Info

Publication number: NO954767D0
Authority: NO; Norway
Prior art keywords: lyase; amino; compounds
Prior art date: 1993-05-25

Application number

NO954767A

Other languages

English (en)

Other versions

NO954767L (no

Inventor

Philip Marvin Weintraub

Cynthia Gates

Michael Angelastro

J O'neal Johnston

Timothy T Curran

Original Assignee

Merrell Pharma Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-05-25

Filing date

1995-11-24

Publication date

1995-11-24

1995-11-24 Application filed by Merrell Pharma Inc filed Critical Merrell Pharma Inc

1995-11-24 Publication of NO954767D0 publication Critical patent/NO954767D0/no

1996-01-25 Publication of NO954767L publication Critical patent/NO954767L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0011—Unsubstituted amino radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0027—Azides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

NO954767A 1993-05-25 1995-11-24 4-amino-17 delser som C17-20-lyase- og 5 NO954767L (no)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US6674493A	1993-05-25	1993-05-25
US20950194A	1994-03-16	1994-03-16
US08/231,434 US5486511A (en)	1993-05-25	1994-05-02	4-amino-17β-(cyclopropyloxy)androst-4-en-3-one, 4-amino-17β-(cyclopropylamino)androst-4-en-3-one and related compounds as C17-20 lyase and 5α-reductase
PCT/US1994/005075 WO1994028010A1 (en)	1993-05-25	1994-05-06	4-AMINO-17β-(CYCLOPROPYLOXY)ANDROST-4-EN-3-ONE, 4-AMINO-17β-(CYCLOPROPYLAMINO)ANDROST-4-EN-3-ONE AND RELATED COMPOUNDS AS C17-20 LYASE AND 5α-REDUCTASE INHIBITORS

Publications (2)

Publication Number	Publication Date
NO954767D0 true NO954767D0 (no)	1995-11-24
NO954767L NO954767L (no)	1996-01-25

Family

ID=27371031

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO954767A NO954767L (no)	1993-05-25	1995-11-24	4-amino-17 delser som C17-20-lyase- og 5

Country Status (11)

Country	Link
US (1)	US5486511A (no)
EP (1)	EP0700400A1 (no)
JP (1)	JPH08510733A (no)
CN (1)	CN1124490A (no)
AU (1)	AU674971B2 (no)
CA (1)	CA2161649A1 (no)
FI (1)	FI955642A7 (no)
HU (1)	HUT73239A (no)
NO (1)	NO954767L (no)
NZ (1)	NZ267231A (no)
WO (1)	WO1994028010A1 (no)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6407082B1 (en) *	1996-09-13	2002-06-18	New Life Pharmaceuticals Inc.	Prevention of ovarian cancer by administration of a vitamin D compound
US6365597B1 (en)	1996-02-14	2002-04-02	Aventis Pharmaceuticals Inc.	4-aza steroids
DE69713285T2 (de) *	1996-02-14	2003-01-02	Aventis Pharmaceuticals Inc., Bridgewater	17-beta-cyclopropyl(amino/oxy)4-aza steroide als testosterone 5-alpha-rectase und c17-20-lyase hemmende verbindungen
US6028064A (en)	1996-09-13	2000-02-22	New Life Pharmaceuticals Inc.	Prevention of ovarian cancer by administration of progestin products
US6034074A (en)	1996-09-13	2000-03-07	New Life Pharmaceuticals Inc.	Prevention of ovarian cancer by administration of a Vitamin D compound
US6511970B1 (en)	1996-09-13	2003-01-28	New Life Pharmaceuticals Inc.	Prevention of ovarian cancer by administration of products that induce transforming growth factor-beta and/or apoptosis in the ovarian epithelium
US6765002B2 (en)	2000-03-21	2004-07-20	Gustavo Rodriguez	Prevention of ovarian cancer by administration of products that induce transforming growth factor-β and/or apoptosis in the ovarian epithelium
BR9811293A (pt) *	1997-07-29	2000-08-29	Sankyo Co	Composições para o tratamento da alopecia, do hirsutismo feminino ou da seborréia, ou uma composição para a prevenção da metástase óssea causada por câncer prostático, e, usos de um composto e de n-{1-metil-1-(4-metoxifenil)etil}-3-oxo-4-aza-5-alfa-and rost-1-eno-17-beta-c arboxamida
US7291626B1 (en) *	1998-04-09	2007-11-06	John Hopkins University School Of Medicine	Inhibitors of hedgehog signaling pathways, compositions and uses related thereto
NZ515134A (en)	1999-05-04	2004-01-30	Strakan Ltd	Androgen glycosides and androgenic activity thereof
AU781524B2 (en) *	1999-10-13	2005-05-26	Johns Hopkins University School Of Medicine, The	Regulators of the hedgehog pathway, compositions and uses related thereto
US20010044431A1 (en) *	2000-03-21	2001-11-22	Rodriguez Gustavo C.	Prevention of ovarian cancer by administration of products that induce biologic effects in the ovarian epithelium
WO2005116047A2 (en) *	2004-05-27	2005-12-08	Migenix Corp.	2-substituted 17-imino estrogen compounds for cytoprotection
CN100355772C (zh) *	2005-12-28	2007-12-19	天津大学	具有5α－还原酶抑制活性的甾体化合物及其制备方法
EP2060261B1 (en)	2007-11-13	2016-03-09	Athenion AG	C-19 steroids for cosmetic uses

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB204888A (en) *	1922-09-26	1923-10-11	William Gibson	Flap support for clubs in golf bags
DK120154B (da) *	1968-02-29	1971-04-19	Schering Ag	Fremgangsmåde til fremstilling af N-substituerede 4-amino-3-oxosteroid-4,6-diener af androstan- eller pregnanrækken eller deres ammoniumsalte.
US3732209A (en) *	1971-03-15	1973-05-08	Hoffmann La Roche	Novel 17beta-oxygenated cyclopropa(16alpha,17alpha)steroids
GB8503940D0 (en) *	1985-02-15	1985-03-20	Erba Farmitalia	4-substituted androstendione derivatives
DE3711772A1 (de) *	1987-04-08	1988-10-27	Schering Ag	4- und 15-disubstituierte 4-androsten-3,17-dione und verfahren zu deren herstellung
US4891367A (en) *	1987-04-22	1990-01-02	Merrell Dow Pharmaceuticals Inc.	17β-(cyclopropyloxy)androst-5-en-3β-ol and related compounds useful as C17-20 lyase inhibitors
AU606677B2 (en) *	1987-04-22	1991-02-14	Merrell Dow Pharmaceuticals Inc.	17 beta -(cyclopropylimino) androst-5-EN-3 beta- Ol and related compounds useful as C17-20 lyase inhibitors
GB8711579D0 (en) *	1987-05-15	1987-06-17	Erba Farmitalia	4-amino-androstenedione derivatives
US4966897A (en) *	1989-08-15	1990-10-30	Merrell Dow Pharmaceuticals Inc.	4-substituted 17β-(cyclopropyloxy)androst-5-en-3β-ol and related compounds useful as C17-20 lyase inhibitors
US5318961A (en) *	1990-08-01	1994-06-07	Merrell Dow Pharmaceuticals Inc.	4-amino-Δ4-steroids and their use as 5α-reductase inhibitors
US5143909A (en) *	1991-03-19	1992-09-01	Merrell Dow Pharmaceuticals Inc.	Aminosteroids in a method for inhibiting c17-20 lyase
US5218110A (en) *	1990-08-01	1993-06-08	Merrell Dow Pharmaceuticals	4-amino-Δ4 -steroids and their use as 5α-reductase inhibitors
NZ239142A (en) *	1990-08-01	1994-05-26	Merrell Dow Pharma	4-amino-delta-4-steroids; preparatory processes and pharmaceutical compositions
US5130424A (en) *	1990-08-01	1992-07-14	Merrell Dow Pharmaceuticals Inc.	4-amino-delta-4,6-steroids and their use as 5 alpha-reductase inhibitors
NZ239141A (en) *	1990-08-01	1994-04-27	Merrell Dow Pharma	4-amino-delta-4,6-steroids; preparatory processes and pharmaceutical compositions
US5120840A (en) *	1990-08-01	1992-06-09	Merrell Dow Pharmaceuticals Inc.	4-amino-4-ene-steroids and their use as 5α-reductase inhibitors
JPH06510982A (ja) *	1991-02-27	1994-12-08	ニューヨークユニバーシティ	抗テストステロン化合物およびその使用方法
US5189032A (en) *	1991-03-19	1993-02-23	Merrell Dow Pharmaceuticals Inc.	4-amino-Δ4,6 -steroids and their use as 5α-reductase inhibitors
US5218810A (en) *	1992-02-25	1993-06-15	Hexcel Corporation	Fabric reinforced concrete columns

1994
- 1994-05-02 US US08/231,434 patent/US5486511A/en not_active Expired - Fee Related
- 1994-05-06 AU AU69455/94A patent/AU674971B2/en not_active Ceased
- 1994-05-06 WO PCT/US1994/005075 patent/WO1994028010A1/en not_active Ceased
- 1994-05-06 HU HU9503369A patent/HUT73239A/hu unknown
- 1994-05-06 EP EP94917930A patent/EP0700400A1/en not_active Withdrawn
- 1994-05-06 NZ NZ267231A patent/NZ267231A/en unknown
- 1994-05-06 JP JP7500673A patent/JPH08510733A/ja active Pending
- 1994-05-06 CA CA002161649A patent/CA2161649A1/en not_active Abandoned
- 1994-05-06 CN CN94192228A patent/CN1124490A/zh active Pending
1995
- 1995-11-23 FI FI955642A patent/FI955642A7/fi not_active Application Discontinuation
- 1995-11-24 NO NO954767A patent/NO954767L/no unknown

Also Published As

Publication number	Publication date
FI955642A0 (fi)	1995-11-23
HUT73239A (en)	1996-07-29
NZ267231A (en)	1997-05-26
AU674971B2 (en)	1997-01-16
AU6945594A (en)	1994-12-20
HU9503369D0 (en)	1996-01-29
US5486511A (en)	1996-01-23
WO1994028010A1 (en)	1994-12-08
NO954767L (no)	1996-01-25
JPH08510733A (ja)	1996-11-12
FI955642A7 (fi)	1995-11-23
EP0700400A1 (en)	1996-03-13
CN1124490A (zh)	1996-06-12
CA2161649A1 (en)	1994-12-08

Publication	Publication Date	Title
NO943999D0 (no)	1994-10-21	1-aminoetylindolderivater
DE69423670D1 (de)	2000-05-04	Siloxy-aluminoxan-Zusammensetzungen
FI961720A0 (fi)	1996-04-19	Uusi koostumus
FI944624A0 (fi)	1994-10-04	4-aryyliaminobentsopyraani- ja niiden kaltaisia yhdisteitä
NO954767D0 (no)	1995-11-24	4-amino-17 delser som C17-20-lyase- og 5
DE69419101D1 (de)	1999-07-22	Hochreine thiol-en-zusammensetzung
FI932094A0 (fi)	1993-05-07	Kylningsapparat i kranens vaexel
FI932732A0 (fi)	1993-06-15	Rotorkonstruktion i en tvaolindningselektricitetsmaskin
DE69430362D1 (de)	2002-05-16	Ektoparasitizide formulierung
FI932264A0 (fi)	1993-05-18	Gapformare i en pappersmaskin
KR950703340A (ko)	1995-09-20	항엠알에스에이 조성물
FI930927A0 (fi)	1993-03-02	Banformningsparti i en pappersmaskin
FIU950356U0 (fi)	1995-08-15	Anordning foer oekning av oeppningstrycket i oevertrycksventilrna i en defekt aonggenerator
SE9302054D0 (sv)	1993-06-14	Tas - mob 2
ITBO930051A0 (it)	1993-02-17	Avismag 2000
ITBO930050A0 (it)	1993-02-17	Magstop 2000
ITPV930002A0 (it)	1993-02-15	Iolanda 92
SE9301471D0 (sv)	1993-04-29	New formulation
SE9303993D0 (sv)	1993-12-01	Ny tandborste -art 2000
DK0707579T3 (da)	1999-09-13	Piperidinylsubstituerede methanoanthracener som D1/D2-antagonister og 5 HT2-serotanin-antagonister
DK40893A (da)	1993-04-06	Mikrobicid sammensaetning
UA27833C2 (uk)	2000-10-16	Деревинно-клейова композиція
ITIS930001A0 (it)	1993-02-09	U l 9 3
FI932312A0 (fi)	1993-05-21	Anordning som underlaettar borstning av taender
FI933315A0 (fi)	1993-07-23	Anordning som underlaettar plockning av jordgubbar