NO932685L - Aminoalkyl-pyrrolidinyl-tiokarbapenem-derivater - Google Patents
Aminoalkyl-pyrrolidinyl-tiokarbapenem-derivaterInfo
- Publication number
- NO932685L NO932685L NO93932685A NO932685A NO932685L NO 932685 L NO932685 L NO 932685L NO 93932685 A NO93932685 A NO 93932685A NO 932685 A NO932685 A NO 932685A NO 932685 L NO932685 L NO 932685L
- Authority
- NO
- Norway
- Prior art keywords
- hydrogen
- group
- different
- lower alkyl
- same
- Prior art date
Links
- 229910052739 hydrogen Inorganic materials 0.000 abstract 7
- 239000001257 hydrogen Substances 0.000 abstract 7
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 5
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 125000003282 alkyl amino group Chemical group 0.000 abstract 2
- 125000002947 alkylene group Chemical group 0.000 abstract 2
- 125000004423 acyloxy group Chemical group 0.000 abstract 1
- 125000005236 alkanoylamino group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
- -1 amino, sulfamoylamino Chemical group 0.000 abstract 1
- 125000005239 aroylamino group Chemical group 0.000 abstract 1
- 125000002393 azetidinyl group Chemical group 0.000 abstract 1
- 125000004069 aziridinyl group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 125000004573 morpholin-4-yl group Chemical group N1(CCOCC1)* 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
- 125000004193 piperazinyl group Chemical group 0.000 abstract 1
- 125000005936 piperidyl group Chemical group 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 125000000719 pyrrolidinyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Forbindelse med formelen (I) hvor R1 er hydrogen eller metyl, R2 er hydrogen eller en negativ ladning, R3 er hydrogen, halogen, hydroksyl, lavere alkoksy, lavere alkanoyloksy, amino, N-lavere alkylamino, N,N- di-lavere alkylamino, lavere alkanoylamino, aroylamino, (lave- re alkylsulfonyl)amino, sulfamoylamino, cyano, nitro, en gruppe -COOR' (hvor R' er hydrogen eller lavere alkyl) eller en gruppe -CON(R1) R6 (hvor hver av R5 og R6 som kan være like eller forskjellige, er hydrogen eller lavere alkyl, eller R5 og R" danner sammen med det tilstøtende nitrogen, en heterocyklisk gruppe valgt fra gruppen bestående av aziridinyl, azetidinyl, pyrrolidinyl, piperidyl, piperazinyl, 4-lavere alkyl- piperazinyl og morfolino), A er lineær eller forgrenet lavere alkylen, X er en gruppe -N(R7) R8 (hvor hver av R7 og R6, som kan være like eller forskjellige, er hydrogen eller lavere alkyl) eller en gruppe -N" (R9) (R10) R11 (hvor hver av R9, R10 og R11, som kan være like eller forskjellige, er lavere alkyl), forutsatt at når A er lineær, lavere alkylen, er R3 forskjellig fra hydrogen; eller et farmasøytisk godtagbart salt eller ester derav.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP33588891 | 1991-11-27 | ||
| JP21561392 | 1992-07-21 | ||
| PCT/JP1992/001544 WO1993011128A1 (en) | 1991-11-27 | 1992-11-26 | Aminoalkylpyrrolidinylthiocarbapenem derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO932685D0 NO932685D0 (no) | 1993-07-26 |
| NO932685L true NO932685L (no) | 1993-07-27 |
Family
ID=27306909
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO93932685A NO932685L (no) | 1991-11-27 | 1993-07-26 | Aminoalkyl-pyrrolidinyl-tiokarbapenem-derivater |
Country Status (1)
| Country | Link |
|---|---|
| NO (1) | NO932685L (no) |
-
1993
- 1993-07-26 NO NO93932685A patent/NO932685L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO932685D0 (no) | 1993-07-26 |
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