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NO903941D0 - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE DIAZEPINON DERIVATIVES. - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE DIAZEPINON DERIVATIVES.

Info

Publication number
NO903941D0
NO903941D0 NO903941A NO903941A NO903941D0 NO 903941 D0 NO903941 D0 NO 903941D0 NO 903941 A NO903941 A NO 903941A NO 903941 A NO903941 A NO 903941A NO 903941 D0 NO903941 D0 NO 903941D0
Authority
NO
Norway
Prior art keywords
diazepinon
derivatives
preparation
therapeutically active
analogue procedure
Prior art date
Application number
NO903941A
Other languages
Norwegian (no)
Other versions
NO903941L (en
Inventor
Wolfhard Engel
Wolfgang Eberlein
Guenter Trummlitz
Gerhard Mihm
Henri Doods
Norbert Mayer
Adriaan De Jonge
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of NO903941D0 publication Critical patent/NO903941D0/en
Publication of NO903941L publication Critical patent/NO903941L/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO90903941A 1989-09-11 1990-09-10 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE DIAZEPINON DERIVATIVES. NO903941L (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3930262A DE3930262A1 (en) 1989-09-11 1989-09-11 CONDENSED DIAZEPINONE, METHOD FOR THE PRODUCTION THEREOF AND MEDICAMENT CONTAINING THESE COMPOUNDS

Publications (2)

Publication Number Publication Date
NO903941D0 true NO903941D0 (en) 1990-09-10
NO903941L NO903941L (en) 1991-03-12

Family

ID=6389152

Family Applications (1)

Application Number Title Priority Date Filing Date
NO90903941A NO903941L (en) 1989-09-11 1990-09-10 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE DIAZEPINON DERIVATIVES.

Country Status (17)

Country Link
EP (1) EP0417631A3 (en)
JP (1) JPH03209382A (en)
KR (1) KR910006286A (en)
AU (1) AU626452B2 (en)
CA (1) CA2025005A1 (en)
DD (1) DD299308A5 (en)
DE (1) DE3930262A1 (en)
FI (1) FI904469A7 (en)
HU (1) HU206882B (en)
IL (1) IL95622A (en)
NO (1) NO903941L (en)
NZ (1) NZ235270A (en)
PL (1) PL165197B1 (en)
PT (1) PT95259A (en)
RU (1) RU2017740C1 (en)
YU (1) YU47372B (en)
ZA (1) ZA907199B (en)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3930266A1 (en) * 1989-09-11 1991-03-14 Thomae Gmbh Dr K CONDENSED DIAZEPINONE, METHOD FOR THE PRODUCTION THEREOF AND MEDICAMENT CONTAINING THESE COMPOUNDS
CA2491506C (en) 2002-07-05 2011-04-26 Targacept, Inc. N-aryl diazaspiracyclic compounds and methods of preparation and use thereof
SE0202133D0 (en) 2002-07-08 2002-07-08 Astrazeneca Ab Novel compounds
SE0303090D0 (en) 2003-11-20 2003-11-20 Astrazeneca Ab Novel compounds
SE0303541D0 (en) 2003-12-22 2003-12-22 Astrazeneca Ab New compounds
US8809552B2 (en) 2011-11-01 2014-08-19 Hoffmann-La Roche Inc. Azetidine compounds, compositions and methods of use
ES2618703T3 (en) 2012-06-13 2017-06-22 F. Hoffmann-La Roche Ag New diazaspyrocycloalkane and azaspyrocycloalkane compounds
CN104684915B (en) 2012-09-25 2017-10-31 霍夫曼-拉罗奇有限公司 Novel Bicyclic Derivatives
AR095079A1 (en) 2013-03-12 2015-09-16 Hoffmann La Roche DERIVATIVES OF OCTAHIDRO-PIRROLO [3,4-C] -PIRROL AND PIRIDINA-FENILO
KR20160087900A (en) 2013-11-26 2016-07-22 에프. 호프만-라 로슈 아게 The novel octahydro-cyclobuta [1,2-c: 3,4-c "] dipyrrol-2-yl
CN106029667B (en) 2014-03-26 2019-08-23 豪夫迈·罗氏有限公司 Fused [1,4]diaza* compounds as inhibitors of autotaxin (ATX) and lysophosphatidic acid (LPA) production
AU2015238537B2 (en) 2014-03-26 2019-08-01 F. Hoffmann-La Roche Ag Bicyclic compounds as autotaxin (ATX) and lysophosphatidic acid (LPA) production inhibitors
MA41898A (en) 2015-04-10 2018-02-13 Hoffmann La Roche BICYCLIC QUINAZOLINONE DERIVATIVES
EP3344619B1 (en) 2015-09-04 2020-10-28 H. Hoffnabb-La Roche Ag Phenoxymethyl derivatives
CN115124538A (en) 2015-09-24 2022-09-30 豪夫迈·罗氏有限公司 Bicyclic compounds as ATX inhibitors
RU2725138C2 (en) 2015-09-24 2020-06-30 Ф. Хоффманн-Ля Рош Аг New bicyclic compounds as double inhibitors of autotaxin (atx)/carbonic anhydrase (ca)
KR20180054634A (en) 2015-09-24 2018-05-24 에프. 호프만-라 로슈 아게 As a dual auto-thixin (ATX) / carbonic anhydrase (CA) inhibitor,
KR20180054635A (en) 2015-09-24 2018-05-24 에프. 호프만-라 로슈 아게 As an autotaxin (ATX) inhibitor,
JP7157755B2 (en) 2017-03-16 2022-10-20 エフ.ホフマン-ラ ロシュ アーゲー Heterocyclic compounds useful as dual ATX/CA inhibitors
JP7090099B2 (en) 2017-03-16 2022-06-23 エフ.ホフマン-ラ ロシュ アーゲー A novel bicyclic compound as an ATX inhibitor
JP7368357B2 (en) * 2017-09-05 2023-10-24 ブラックソーン セラピューティクス インコーポレイテッド Vasopressin receptor antagonists and related products and methods

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4210648A (en) * 1977-05-31 1980-07-01 Boehringer Ingelheim Gmbh II-Aminoacyl-5,11-dihydro-6H-pyrido(2,3-B) (1,4)benzodiazepin-6-ones and salts thereof
DE3204153A1 (en) * 1982-02-06 1983-08-11 Dr. Karl Thomae Gmbh, 7950 Biberach SUBSTITUTED THIENOBENZODIAZEPINONE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING IT
DE3204403A1 (en) * 1982-02-09 1983-08-11 Dr. Karl Thomae Gmbh, 7950 Biberach NEW PYRIDOBENZODIAZEPINONE, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
DE3726908A1 (en) * 1987-08-13 1989-02-23 Thomae Gmbh Dr K NEW CONDENSED DIAZEPINONE, PROCESS FOR THEIR MANUFACTURE AND MEDICAMENTS CONTAINING THESE COMPOUNDS
DE3930266A1 (en) * 1989-09-11 1991-03-14 Thomae Gmbh Dr K CONDENSED DIAZEPINONE, METHOD FOR THE PRODUCTION THEREOF AND MEDICAMENT CONTAINING THESE COMPOUNDS

Also Published As

Publication number Publication date
PL286835A1 (en) 1991-08-26
YU47372B (en) 1995-01-31
KR910006286A (en) 1991-04-29
HUT55393A (en) 1991-05-28
IL95622A0 (en) 1991-06-30
JPH03209382A (en) 1991-09-12
AU6235290A (en) 1991-03-14
NO903941L (en) 1991-03-12
EP0417631A3 (en) 1991-12-11
FI904469A7 (en) 1991-03-12
HU206882B (en) 1993-01-28
EP0417631A2 (en) 1991-03-20
RU2017740C1 (en) 1994-08-15
FI904469A0 (en) 1990-09-11
PL165197B1 (en) 1994-11-30
PT95259A (en) 1991-05-22
DE3930262A1 (en) 1991-03-21
AU626452B2 (en) 1992-07-30
YU171590A (en) 1993-05-28
IL95622A (en) 1994-04-12
ZA907199B (en) 1992-05-27
CA2025005A1 (en) 1991-03-12
NZ235270A (en) 1991-11-26
DD299308A5 (en) 1992-04-09
HU905852D0 (en) 1991-03-28

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