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NO900790L - Melatoninanaloger. - Google Patents

Melatoninanaloger.

Info

Publication number
NO900790L
NO900790L NO90900790A NO900790A NO900790L NO 900790 L NO900790 L NO 900790L NO 90900790 A NO90900790 A NO 90900790A NO 900790 A NO900790 A NO 900790A NO 900790 L NO900790 L NO 900790L
Authority
NO
Norway
Prior art keywords
melatonin analogues
melatonin
analogues
Prior art date
Application number
NO90900790A
Other languages
English (en)
Other versions
NO173732B (no
NO173732C (no
NO900790D0 (no
Inventor
Margarita L Dubocovich
James V Peck
Atef A Helmy
Vithal J Rajadhyaksha
Original Assignee
Nelson Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nelson Res & Dev filed Critical Nelson Res & Dev
Publication of NO900790D0 publication Critical patent/NO900790D0/no
Publication of NO900790L publication Critical patent/NO900790L/no
Publication of NO173732B publication Critical patent/NO173732B/no
Publication of NO173732C publication Critical patent/NO173732C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Saccharide Compounds (AREA)
NO900790A 1987-08-17 1990-02-19 Analogifremgangsmaate for fremstilling av 2-arylsubstituerte N- acetyltryptaminer NO173732C (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8629087A 1987-08-17 1987-08-17
US8606287A 1987-08-17 1987-08-17
PCT/US1988/001859 WO1989001472A1 (en) 1987-08-17 1988-05-20 Melatonin analogues

Publications (4)

Publication Number Publication Date
NO900790D0 NO900790D0 (no) 1990-02-19
NO900790L true NO900790L (no) 1990-03-26
NO173732B NO173732B (no) 1993-10-18
NO173732C NO173732C (no) 1994-01-26

Family

ID=26774333

Family Applications (1)

Application Number Title Priority Date Filing Date
NO900790A NO173732C (no) 1987-08-17 1990-02-19 Analogifremgangsmaate for fremstilling av 2-arylsubstituerte N- acetyltryptaminer

Country Status (7)

Country Link
EP (1) EP0375726A4 (no)
KR (1) KR910006124B1 (no)
AU (1) AU616907B2 (no)
DK (1) DK42490A (no)
FI (1) FI900801A7 (no)
NO (1) NO173732C (no)
WO (1) WO1989001472A1 (no)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK108022C (da) * 1964-10-15 1967-07-31 Svend Anton Hansen Wexel Fremgangsmåde til hel eller delvis udskæring af rygbenet af opskårne slagtekroppe, navnlig grisekroppe, og anlæg til udførelse af denne fremgangsmåde.
AU644367B2 (en) * 1989-05-17 1993-12-09 Applied Medical Research Ltd Use of melatonin derivatives for effecting contraception
US5071875A (en) * 1989-09-25 1991-12-10 Northwestern University Substituted 2-amidotetralins as melatonin agonists and antagonists
IT1251544B (it) * 1991-05-13 1995-05-17 Gabriele Biella Composizioni farmaceutiche attive nella terapia dei disturbi del sonno comprendenti melatonina o un suo derivato in associazione con un derivato benzodiazepinico
FR2680366B1 (fr) * 1991-08-13 1995-01-20 Adir Nouveaux derives d'arylethylamines, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
AU660336B2 (en) * 1991-10-18 1995-06-22 Alza Corporation Device for the transdermal administration of melatonin
US5206377A (en) * 1991-12-05 1993-04-27 Whitby Research, Inc. Compounds useful as antiproliferative agents
IT1255199B (it) * 1992-07-01 1995-10-20 Franco Fraschini Farmaco sintetizzato analogo della melatonina particolarmente efficacenelle patologie che interferiscono con i ritmi circadiani
US5300481A (en) * 1993-05-05 1994-04-05 The Regents Of The University Of California Methods for controlling flowering in plants
US5654325A (en) * 1993-11-18 1997-08-05 Eli Lilly And Company Melatonin derivatives for use in treating sleep disorders
US6180657B1 (en) 1993-11-18 2001-01-30 Eli Lilly And Company Melatonin derivatives for use in treating desynchronization disorders
FR2713636B1 (fr) * 1993-12-07 1996-01-05 Adir Nouveaux dérivés naphtaléniques, leur procédé de préparation, et les compositions pharmaceutiques qui les contiennent.
US5403851A (en) * 1994-04-05 1995-04-04 Interneuron Pharmaceuticals, Inc. Substituted tryptamines, phenalkylamines and related compounds
FR2718445B1 (fr) * 1994-04-07 1996-06-28 Cemaf Nouveaux dérivés de spiro [indole-pyrrolidine] agonistes de la mélatonine, leur procédé de préparation et leur utilisation à titre de médicament.
FR2724170B1 (fr) * 1994-09-02 1997-05-30 Cemaf Nouveaux derives de spiro(indole-pyrrolidine) agonistes de la melatonine, leur procede de preparation et leur utilisation a titre de medicament
EP0754183A1 (fr) * 1994-04-07 1997-01-22 Cemaf Nouveaux derives de spiro[indole-pyrrolidine] agonistes melatoninergiques, leur procede de preparation et leur utilisation a titre de medicament
AU2001280984A1 (en) * 2000-07-28 2002-02-13 Inspire Pharmaceuticals, Inc. Use of indole derivatives for the manufacture of a medicament for reducing intracular pressure
ES2172415B2 (es) * 2000-07-28 2003-11-16 Univ Madrid Complutense Tratamiento del glaucoma y la hipertension ocular por medio de un analogo de la melatonina.
US7335776B2 (en) 2001-03-14 2008-02-26 Ono Pharmaceutical Co., Ltd. Remedies for depression containing EP1 antagonist as the active ingredient
FR2874611B1 (fr) * 2004-08-31 2006-11-17 Servier Lab Nouveaux derives d'imidazopyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
WO2010012789A1 (en) 2008-07-30 2010-02-04 Ferrer Internacional S. A. 1,6-dihydro-2h-3-oxa-6-aza-as-indacene compounds
KR101534523B1 (ko) * 2013-04-30 2015-07-09 경희대학교 산학협력단 1,2,3,4-테트라히드로-6-메톡시-1-옥소-베타-카르볼린을 포함하는 피부 미백용 화장료 조성물
FR3065225B1 (fr) 2017-04-12 2024-04-05 Patrick Choay Sas Adjuvants depourvus de cytokines pour milieux de culture cellulaire, notamment pour fecondation in vitro, ou pour la culture de follicules, cellules germinales males ou embryons

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3370063A (en) * 1964-10-05 1968-02-20 Mcneilab Inc Substituted dimethoxy indoles and method of making the same
US3915990A (en) * 1973-03-13 1975-10-28 Nelson Res & Dev Tryptamines
US4087444A (en) * 1976-09-08 1978-05-02 Eli Lilly And Company Amides as ovulation inhibitors

Also Published As

Publication number Publication date
NO173732B (no) 1993-10-18
KR910006124B1 (ko) 1991-08-13
NO173732C (no) 1994-01-26
WO1989001472A1 (en) 1989-02-23
NO900790D0 (no) 1990-02-19
DK42490A (da) 1990-04-17
FI900801A0 (fi) 1990-02-16
KR890701558A (ko) 1989-12-20
DK42490D0 (da) 1990-02-16
AU2309788A (en) 1989-03-09
FI900801A7 (fi) 1990-02-16
EP0375726A1 (en) 1990-07-04
EP0375726A4 (en) 1991-01-30
AU616907B2 (en) 1991-11-14

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