[go: up one dir, main page]

NO904470D0 - PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZODIAZEPINE DERIVATIVES. - Google Patents

PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZODIAZEPINE DERIVATIVES.

Info

Publication number
NO904470D0
NO904470D0 NO904470A NO904470A NO904470D0 NO 904470 D0 NO904470 D0 NO 904470D0 NO 904470 A NO904470 A NO 904470A NO 904470 A NO904470 A NO 904470A NO 904470 D0 NO904470 D0 NO 904470D0
Authority
NO
Norway
Prior art keywords
procedure
preparation
therapeutic active
benzodiazepine derivatives
active benzodiazepine
Prior art date
Application number
NO904470A
Other languages
Norwegian (no)
Other versions
NO904470L (en
Inventor
Jean-Claude Muller
Gilbert Lassalle
Colombe Denys
Alistair Lochead
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of NO904470D0 publication Critical patent/NO904470D0/en
Publication of NO904470L publication Critical patent/NO904470L/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO90904470A 1989-10-17 1990-10-16 PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZOTIAZEPINE DERIVATIVES. NO904470L (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8913540A FR2653122B1 (en) 1989-10-17 1989-10-17 DERIVATIVES OF 5- [2 - [[2-AMINO-2-OXOETHYL] METHYLAMINO] ETHYL] -2,3-DIHYDRO-3-HYDROXY-2- (4-METHOXYPHENYL) -1.5 (5H) -BENZOTHIAZEPINE-4 -ONE, THEIR PREPARATION AND THEIR APPLICATION IN THERAPEUTICS.

Publications (2)

Publication Number Publication Date
NO904470D0 true NO904470D0 (en) 1990-10-16
NO904470L NO904470L (en) 1991-04-18

Family

ID=9386468

Family Applications (1)

Application Number Title Priority Date Filing Date
NO90904470A NO904470L (en) 1989-10-17 1990-10-16 PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZOTIAZEPINE DERIVATIVES.

Country Status (14)

Country Link
EP (1) EP0424214A1 (en)
JP (1) JPH03133970A (en)
KR (1) KR910007901A (en)
AU (1) AU6479690A (en)
CA (1) CA2027738A1 (en)
FI (1) FI905089A7 (en)
FR (1) FR2653122B1 (en)
HU (1) HUT57754A (en)
IE (1) IE903720A1 (en)
IL (1) IL95931A0 (en)
NO (1) NO904470L (en)
NZ (1) NZ235717A (en)
PT (1) PT95606A (en)
ZA (1) ZA908267B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69411387T2 (en) * 1994-09-16 1999-02-25 Orion Corp. FERMION, Espoo Process for the preparation of pharmaceutically active benzothiazepine derivatives.
FI97725C (en) * 1995-02-17 1997-02-10 Orion Yhtymae Oy Process for the preparation of diltiazem
WO2005035505A2 (en) * 2003-09-30 2005-04-21 Artesian Therapeutics, Inc. Compounds with phosphodiesterase inhibiting and calcium channel blocking activities

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH538492A (en) * 1970-10-07 1973-06-30 Hoffmann La Roche Process for the preparation of benzodiazepine derivatives
FR2624117B1 (en) * 1987-12-08 1991-02-22 Synthelabo HYDROXY-3 (METHOXY-4 PHENYL) -2 (METHYLAMINO-2 ETHYL) -5 DIHYDRO-2,3 5H-BENZOTHIAZEPINE-1,5 ONE-4 DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2630109B1 (en) * 1988-04-19 1991-11-29 Synthelabo DERIVATIVES OF ((N- (2-AMINO-2 OXO-2 ETHYL) METHYLAMINO) -2 ETHYL) -5 HYDROXY-3 (METHOXY-4 PHENYL) -2 DIHYDRO-2,3 5H-BENZOTHIAZEPINE-1,5 ONE-4, THEIR PREPARATION AND THEIR APPLICATION IN THERAPEUTICS

Also Published As

Publication number Publication date
CA2027738A1 (en) 1991-04-18
JPH03133970A (en) 1991-06-07
AU6479690A (en) 1991-07-11
PT95606A (en) 1991-09-13
FR2653122B1 (en) 1994-04-15
HUT57754A (en) 1991-12-30
FI905089A7 (en) 1991-04-18
NZ235717A (en) 1991-12-23
ZA908267B (en) 1991-08-28
HU906466D0 (en) 1991-04-29
NO904470L (en) 1991-04-18
IL95931A0 (en) 1991-07-18
IE903720A1 (en) 1991-04-24
EP0424214A1 (en) 1991-04-24
FR2653122A1 (en) 1991-04-19
KR910007901A (en) 1991-05-30
FI905089A0 (en) 1990-10-16

Similar Documents

Publication Publication Date Title
NO904694L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE IMIDAZOLD DERIVATIVES.
NO903088D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE DIAZEPINE DERIVATIVES.
NO901684D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 3-SUBSTITUTED-2-OXINDOL DERIVATIVES.
NO894630L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE KINUCLIDINE DERIVATIVES.
NO883974L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TETRAHYDRO-HYDROXYPYRANON DERIVATIVES.
NO904986L (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE DIAZEPINE DERIVATIVES.
NO893616D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TRICYCLIC COMPOUNDS.
NO902411D0 (en) ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 2-HYDROXY-N-PROPYLAMINES.
NO883122D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ARYLAMIDE DERIVATIVES.
NO890155L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE INDOLPIPERIDIN COMPOUNDS.
NO881762D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZAZEPINE DERIVATIVES.
NO900697D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ACETAMIDE DERIVATIVES.
NO891723L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE CHINAZOLINE DERIVATIVES.
NO905327D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE CARBAMOIL OIL DERIVATIVES.
NO865012L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZAZEPINE DERIVATIVES.
NO900972L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE NAFTALEN DERIVATIVES.
NO913187L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TRICYCLIC DERIVATIVES.
NO900942D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE AZACYCLOOKTADIEN DERIVATIVES.
NO904470D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZODIAZEPINE DERIVATIVES.
NO890724D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TETRAAZAACENAPYLENE DERIVATIVES.
NO890519D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PROPANON DERIVATIVES.
NO880492D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE TRICYCLIC TRIAZOLPYRIMIDINE DERIVATIVES.
NO890506D0 (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE CHLORANILIN DERIVATIVES.
NO891677L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PHENETANOLAMINE DERIVATIVES.
NO891678L (en) PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ETHANOLAMINE DERIVATIVES.