NO890155L - Fremgangsmaate for fremstilling av terapeutisk aktive indolpiperidin-forbindelser. - Google Patents

Fremgangsmaate for fremstilling av terapeutisk aktive indolpiperidin-forbindelser.

Info

Publication number: NO890155L
Authority: NO; Norway
Prior art keywords: indolpiperidin; compounds; procedure; preparation; therapeutic active
Prior art date: 1988-01-14

Application number

NO89890155A

Other languages

English (en)

Other versions

NO890155D0 (no

NO172539B (no

NO172539C (no

Inventor

Masaaki Matsuo

Takashi Manabe

Shinji Shigenaga

Hiroshi Matsuda

Original Assignee

Fujisawa Pharmaceutical Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-01-14

Filing date

1989-01-13

Publication date

1989-07-17

1988-01-14 Priority claimed from GB888800795A external-priority patent/GB8800795D0/en

1988-08-01 Priority claimed from GB888818260A external-priority patent/GB8818260D0/en

1989-01-13 Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co

1989-01-13 Publication of NO890155D0 publication Critical patent/NO890155D0/no

1989-07-17 Publication of NO890155L publication Critical patent/NO890155L/no

1993-04-26 Publication of NO172539B publication Critical patent/NO172539B/no

1993-08-04 Publication of NO172539C publication Critical patent/NO172539C/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pulmonology (AREA)
Immunology (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

NO890155A 1988-01-14 1989-01-13 Analogifremgangsmaate for fremstilling av terapeutisk aktive indolpiperidin-forbindelser NO172539C (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB888800795A GB8800795D0 (en)	1988-01-14	1988-01-14	New indolylpiperidine compounds processes for preparations thereof & pharmaceutical composition comprising same
GB888818260A GB8818260D0 (en)	1988-08-01	1988-08-01	New indolylpiperidine compounds processes for preparation thereof & pharmaceutical composition comprising same

Publications (4)

Publication Number	Publication Date
NO890155D0 NO890155D0 (no)	1989-01-13
NO890155L true NO890155L (no)	1989-07-17
NO172539B NO172539B (no)	1993-04-26
NO172539C NO172539C (no)	1993-08-04

Family

ID=26293316

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO890155A NO172539C (no)	1988-01-14	1989-01-13	Analogifremgangsmaate for fremstilling av terapeutisk aktive indolpiperidin-forbindelser

Country Status (16)

Country	Link
US (2)	US4935432A (no)
EP (1)	EP0324431B1 (no)
JP (1)	JPH0759577B2 (no)
KR (1)	KR0130899B1 (no)
CN (1)	CN1021733C (no)
AU (1)	AU620583B2 (no)
CA (1)	CA1336605C (no)
DE (1)	DE68901039D1 (no)
DK (1)	DK733788A (no)
ES (1)	ES2032339T3 (no)
FI (1)	FI91863C (no)
GR (1)	GR3004987T3 (no)
HU (2)	HU202224B (no)
IE (1)	IE63476B1 (no)
IL (1)	IL88903A (no)
NO (1)	NO172539C (no)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK733788A (da) *	1988-01-14	1989-07-15	Fujisawa Pharmaceutical Co	Indolylpiperidinderivater og fremgangsmaade til fremstilling deraf
US5521196A (en) *	1994-10-05	1996-05-28	Eli Lilly And Company	5-HT1F agonists for the treatment of migraine
US5521197A (en) *	1994-12-01	1996-05-28	Eli Lilly And Company	3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT1F agonists
DE19500689A1 (de) *	1995-01-12	1996-07-18	Merck Patent Gmbh	Indolpiperidin-Derivate
WO1996029075A1 (en) *	1995-03-20	1996-09-26	Eli Lilly And Company	5-substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)- and 3-(piperidin-4-yl)-1h-indoles: new 5-ht1f agonists
US6458806B1 (en) *	1996-08-15	2002-10-01	Millennium Pharmaceuticals, Inc.	Aryl alkenamides derivatives as MCP-1 antagonists
ES2165274B1 (es)	1999-06-04	2003-04-01	Almirall Prodesfarma Sa	Nuevos derivados de indolilpiperidina como agentes antihistaminicos y antialergicos.
KR20010085555A (ko) *	1999-06-24	2001-09-07	히라이 가쯔히꼬	아드레날린 알파1비 수용체 길항약
US6693099B2 (en) *	2000-10-17	2004-02-17	The Procter & Gamble Company	Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance
US6376514B1 (en) *	2000-10-17	2002-04-23	The Procter & Gamble Co.	Substituted six-membered heterocyclic compounds useful for treating multidrug resistance and compositions and methods thereof
ES2172436B1 (es)	2000-10-31	2004-01-16	Almirall Prodesfarma Sa	Derivados de indolilpiperidina como agentes antihistaminicos y antialergicos.
US6803362B2 (en)	2001-03-09	2004-10-12	Ortho-Mcneil Pharmaceutical Inc.	Heterocyclic compounds
ES2201907B1 (es)	2002-05-29	2005-06-01	Almirall Prodesfarma, S.A.	Nuevos derivados de indolilpiperidina como potentes agentes antihistaminicos y antialergicos.
AU2003274956A1 (en) *	2002-09-06	2004-03-29	Janssen Pharmaceutica, N.V.	Use of indolyl derivatives for the manufacture of a medicament for the treatment allergic rhinitis
PL377087A1 (pl)	2002-09-06	2006-01-23	Janssen Pharmaceutica, N.V.	Związki heterocykliczne

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2193584B1 (no) *	1972-07-28	1975-08-08	Roussel Uclaf
GB1425354A (en) *	1973-10-10	1976-02-18	Wyeth John & Brother Ltd	Indole derivatives
FR2258843B1 (no) *	1974-01-30	1977-09-09	Roussel Uclaf
IL48508A (en) *	1974-12-09	1979-10-31	Roussel Uclaf	Pharmaceutical compositions comprising piperidylindole derivatives
FR2349331A1 (fr) *	1976-04-30	1977-11-25	Roussel Uclaf	Nouveaux derives de 2,3 dihydro a/4-(3-indolyl) 1-piperidinyl/methyl 1,4-benzodioxin-2-methanol, un procede pour leur preparation et leur application comme medicaments
US4359468A (en) *	1981-02-25	1982-11-16	Boehringer Ingelheim Ltd.	Antiallergic N-[4-(indolyl)-piperidino-alkyl]-benzimidazolones
JPS57188567A (en) *	1981-05-13	1982-11-19	Fujimoto Seiyaku Kk	Novel preparation of etomidoline
US4443461A (en) *	1981-09-10	1984-04-17	John Wyeth & Brother Limited	N-[2-[[1-[1H-Indolylalkyl- or oxoalkyl]-4-piperidinyl]-amino]-2-oxoethyl]-arylcarboxamide derivatives
FR2533924A1 (fr) *	1982-10-05	1984-04-06	Roussel Uclaf	Nouveaux derives du 4-(1h-indol-3-yl)a-methyl piperidine-1-ethanol, leurs sels, le procede de preparation, l'application a titre de medicaments et les compositions les renfermant
JPS60142981A (ja) *	1983-12-28	1985-07-29	Yoshitomi Pharmaceut Ind Ltd	３−インド−ルカルボキサミド誘導体
US4673684A (en) *	1984-04-04	1987-06-16	Terumo Corporation	Amide derivatives and 5-lipoxygenase inhibitors containing the same as an active ingredient
US4548939A (en) *	1984-10-01	1985-10-22	Janssen Pharmaceutica N. V.	1H-Indol-3-yl containing 1,3-dimethyl-1H-purine-2,6-diones
IE58370B1 (en) *	1985-04-10	1993-09-08	Lundbeck & Co As H	Indole derivatives
US4742057A (en) *	1985-12-05	1988-05-03	Fujisawa Pharmaceutical Co., Ltd.	Antiallergic thiazole compounds
DK733788A (da) *	1988-01-14	1989-07-15	Fujisawa Pharmaceutical Co	Indolylpiperidinderivater og fremgangsmaade til fremstilling deraf
GB8819024D0 (en) *	1988-08-10	1988-09-14	Glaxo Group Ltd	Chemical compounds
GB8903036D0 (en) *	1989-02-10	1989-03-30	Glaxo Group Ltd	Chemical compounds

1988
- 1988-12-30 DK DK733788A patent/DK733788A/da not_active Application Discontinuation
1989
- 1989-01-06 IL IL88903A patent/IL88903A/xx not_active IP Right Cessation
- 1989-01-09 IE IE4889A patent/IE63476B1/en not_active IP Right Cessation
- 1989-01-10 ES ES198989100332T patent/ES2032339T3/es not_active Expired - Lifetime
- 1989-01-10 DE DE8989100332T patent/DE68901039D1/de not_active Expired - Fee Related
- 1989-01-10 EP EP89100332A patent/EP0324431B1/en not_active Expired - Lifetime
- 1989-01-11 FI FI890123A patent/FI91863C/fi not_active IP Right Cessation
- 1989-01-11 AU AU28370/89A patent/AU620583B2/en not_active Ceased
- 1989-01-11 US US07/295,569 patent/US4935432A/en not_active Expired - Fee Related
- 1989-01-13 KR KR1019890000297A patent/KR0130899B1/ko not_active Expired - Fee Related
- 1989-01-13 CA CA000588224A patent/CA1336605C/en not_active Expired - Fee Related
- 1989-01-13 HU HU89132A patent/HU202224B/hu not_active IP Right Cessation
- 1989-01-13 CN CN89100182A patent/CN1021733C/zh not_active Expired - Fee Related
- 1989-01-13 NO NO890155A patent/NO172539C/no unknown
- 1989-01-13 JP JP1007272A patent/JPH0759577B2/ja not_active Expired - Lifetime
- 1989-09-28 US US07/414,022 patent/US5017703A/en not_active Expired - Fee Related
1992
- 1992-06-19 GR GR910402226T patent/GR3004987T3/el unknown
1995
- 1995-06-22 HU HU95P/P00342P patent/HU211485A9/hu unknown

Also Published As

Publication number	Publication date
HU211485A9 (en)	1995-11-28
JPH0759577B2 (ja)	1995-06-28
DK733788A (da)	1989-07-15
DK733788D0 (da)	1988-12-30
IE890048L (en)	1989-07-14
KR0130899B1 (ko)	1998-04-23
CN1021733C (zh)	1993-08-04
NO890155D0 (no)	1989-01-13
EP0324431A1 (en)	1989-07-19
NO172539B (no)	1993-04-26
NO172539C (no)	1993-08-04
GR3004987T3 (no)	1993-04-28
JPH01221377A (ja)	1989-09-04
IL88903A0 (en)	1989-08-15
FI91863B (fi)	1994-05-13
AU2837089A (en)	1989-07-20
CA1336605C (en)	1995-08-08
FI890123L (fi)	1989-07-15
FI890123A0 (fi)	1989-01-11
IE63476B1 (en)	1995-04-19
ES2032339T3 (es)	1993-02-01
HU202224B (en)	1991-02-28
HUT49871A (en)	1989-11-28
CN1035112A (zh)	1989-08-30
DE68901039D1 (de)	1992-04-30
IL88903A (en)	1993-03-15
US5017703A (en)	1991-05-21
AU620583B2 (en)	1992-02-20
EP0324431B1 (en)	1992-03-25
FI91863C (fi)	1994-08-25
KR890011872A (ko)	1989-08-23
US4935432A (en)	1990-06-19

Publication	Publication Date	Title
NO871267L (no)	1987-09-28	Fremgangsmaate for fremstilling av terapeutisk aktive tiazepinforbindelser.
NO895086D0 (no)	1989-12-18	Fremgangsmaate for fremstilling av terapeutisk aktive heterocykliske forbindelser.
NO894630L (no)	1990-05-23	Fremgangsmaate for fremstilling av terapeutisk aktive kinuklidin-derivater.
NO904694L (no)	1991-05-02	Fremgangsmaate for fremstilling av terapeutisk aktive imidazolderivater.
NO901684D0 (no)	1990-04-17	Fremgangsmaate for fremstilling av terapeutisk aktive 3-substituerte-2-oksindol-derivater.
NO883974L (no)	1989-03-09	Fremgangsmaate for fremstilling av terapeutiske aktive tetrahydro-hydroksypyranon-derivater.
NO871266L (no)	1987-09-28	Fremgangsmaate for fremstilling av terapeutisk aktive kinazolin-derivater.
NO870526D0 (no)	1987-02-11	Fremgangsmaate for fremstilling av terapeutisk aktive dikloranilin-derivater.
NO893616D0 (no)	1989-09-08	Fremgangsmaate for fremstilling av terapeutisk aktive tricykliske forbindelser.
NO902411D0 (no)	1990-05-31	Analogifremgangsmaate for fremstilling av terapeutisk aktive 2-hydroksy-n-propylaminer.
NO874032D0 (no)	1987-09-25	Fremgangsmaate for fremstilling av terapeutisk aktive catecholderivater.
NO864879L (no)	1987-06-09	Fremgangsmaate for fremstilling av terapeutisk aktive tiazolforbindelser.
NO883485D0 (no)	1988-08-05	Fremgangsmaate for fremstilling av terapeutisk aktive piperidinyl-isokinolinforbindelser.
NO890155L (no)	1989-07-17	Fremgangsmaate for fremstilling av terapeutisk aktive indolpiperidin-forbindelser.
NO880667L (no)	1988-08-18	Fremgangsmaate for fremstilling av terapeutisk aktive arylpiperazinyl-alkylen-fenyl-heterocykliske forbindelser.
NO891723D0 (no)	1989-04-26	Fremgangsmaate for fremstilling av terapeutisk aktive kinazolin-derivater.
NO900972D0 (no)	1990-03-01	Fremgangsmaate for fremstilling av terapeutisk aktive naftalen-derivater.
NO168247C (no)	1992-01-29	Analogifremgangsmaate for fremstilling av terapeutisk aktive 5-metoksy-alkyl-ammonium-tetrahydrofuraner.
NO892871D0 (no)	1989-07-11	Fremgangsmaate for fremstilling av terapeutisk aktive forbindelser.
NO882281D0 (no)	1988-05-25	Fremgangsmaate for fremstilling av terapeutisk aktive pyrazinamider.
NO871907D0 (no)	1987-05-07	Fremgangsmaate for fremstilling av terapeutisk aktive alkenamid-derivater.
NO900942D0 (no)	1990-02-28	Fremgangsmaate for fremstilling av terapeutisk aktive azacyklooktadien-derivater.
NO890724D0 (no)	1989-02-21	Fremgangsmaate for fremstilling av terapeutisk aktive tetraazaacenaftylen-derivater.
NO883959D0 (no)	1988-09-06	Fremgangsmaate for fremstilling av terapeutisk aktive fenolestere.
NO882282L (no)	1988-11-28	Fremgangsmaate for fremstilling av terapeutisk aktive pyrazinamider.