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NO874856D0 - Fremgangsmaate til fremstilling av nye substituerte alkandifosfonsyrer. - Google Patents

Fremgangsmaate til fremstilling av nye substituerte alkandifosfonsyrer.

Info

Publication number
NO874856D0
NO874856D0 NO874856A NO874856A NO874856D0 NO 874856 D0 NO874856 D0 NO 874856D0 NO 874856 A NO874856 A NO 874856A NO 874856 A NO874856 A NO 874856A NO 874856 D0 NO874856 D0 NO 874856D0
Authority
NO
Norway
Prior art keywords
halogen
acids
substituted
phosphono group
atoms
Prior art date
Application number
NO874856A
Other languages
English (en)
Other versions
NO173446B (no
NO874856L (no
NO173446C (no
Inventor
Knut A Jaeggi
Leo Widler
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4280350&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO874856(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of NO874856D0 publication Critical patent/NO874856D0/no
Publication of NO874856L publication Critical patent/NO874856L/no
Publication of NO173446B publication Critical patent/NO173446B/no
Publication of NO173446C publication Critical patent/NO173446C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6536Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and sulfur atoms with or without oxygen atoms, as the only ring hetero atoms
    • C07F9/6539Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/02Nutrients, e.g. vitamins, minerals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503Five-membered rings
    • C07F9/65031Five-membered rings having the nitrogen atoms in the positions 1 and 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503Five-membered rings
    • C07F9/6506Five-membered rings having the nitrogen atoms in positions 1 and 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6515Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having three nitrogen atoms as the only ring hetero atoms
    • C07F9/6518Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Nutrition Science (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Control Of El Displays (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
  • Glass Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
NO874856A 1986-11-21 1987-11-20 Analogifremgangsmaate til fremstilling av nye, terapeutisk aktive, substituerte alkandifosfonsyrer NO173446C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH466686 1986-11-21

Publications (4)

Publication Number Publication Date
NO874856D0 true NO874856D0 (no) 1987-11-20
NO874856L NO874856L (no) 1988-05-24
NO173446B NO173446B (no) 1993-09-06
NO173446C NO173446C (no) 1993-12-15

Family

ID=4280350

Family Applications (2)

Application Number Title Priority Date Filing Date
NO874856A NO173446C (no) 1986-11-21 1987-11-20 Analogifremgangsmaate til fremstilling av nye, terapeutisk aktive, substituerte alkandifosfonsyrer
NO2001015C NO2001015I2 (no) 1986-11-21 2001-09-04 Zoledronsyre

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO2001015C NO2001015I2 (no) 1986-11-21 2001-09-04 Zoledronsyre

Country Status (27)

Country Link
US (1) US4939130A (no)
EP (1) EP0275821B1 (no)
JP (1) JP2744238B2 (no)
KR (1) KR960010752B1 (no)
AT (1) ATE72816T1 (no)
AU (1) AU607722B2 (no)
CA (1) CA1338937C (no)
CY (1) CY1827A (no)
DD (1) DD270533A5 (no)
DE (2) DE3776880D1 (no)
DK (1) DK174098B1 (no)
ES (1) ES2038692T4 (no)
FI (1) FI87570C (no)
GR (1) GR3003895T3 (no)
HK (1) HK114894A (no)
HU (1) HU199150B (no)
IE (1) IE59816B1 (no)
IL (1) IL84497A (no)
LU (1) LU90838I2 (no)
MX (1) MX9427A (no)
NL (1) NL300058I2 (no)
NO (2) NO173446C (no)
NZ (1) NZ222610A (no)
PH (1) PH24345A (no)
PT (1) PT86167B (no)
SG (1) SG92194G (no)
ZA (1) ZA878698B (no)

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* Cited by examiner, † Cited by third party
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US5753634A (en) * 1992-05-29 1998-05-19 The Procter & Gamble Company Quaternary nitrogen containing phosphonate compounds, pharmaceutical compostions, and methods for treating abnormal calcium and phosphate metabolism
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US9943531B2 (en) 2014-08-08 2018-04-17 Antecip Bioventures Ii Llc Osteoclast inhibitors such as zoledronic acid for low back pain treatment
US9956234B2 (en) 2012-05-14 2018-05-01 Antecip Bioventures Ii Llc Osteoclast inhibitors for joint conditions
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JP2744238B2 (ja) 1998-04-28
US4939130A (en) 1990-07-03
KR880006204A (ko) 1988-07-22
IE873148L (en) 1988-05-21
DK609587D0 (da) 1987-11-20
ZA878698B (en) 1988-05-23
MX9427A (es) 1993-12-01
AU8145387A (en) 1988-05-26
EP0275821A1 (de) 1988-07-27
CY1827A (en) 1995-12-01
DD270533A5 (de) 1989-08-02
CA1338937C (en) 1997-02-25
SG92194G (en) 1995-04-28
PT86167A (en) 1987-12-01
EP0275821B1 (de) 1992-02-26
FI875096A0 (fi) 1987-11-18
JPS63150291A (ja) 1988-06-22
IL84497A (en) 1994-10-21
NO2001015I2 (no) 2004-10-11
HK114894A (en) 1994-10-27
NO874856L (no) 1988-05-24
HU199150B (en) 1990-01-29
GR3003895T3 (no) 1993-03-16
FI87570B (fi) 1992-10-15
DK609587A (da) 1988-05-22
NO173446C (no) 1993-12-15
NL300058I2 (nl) 2002-02-01
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DK174098B1 (da) 2002-06-17
NZ222610A (en) 1990-09-26
FI875096A7 (fi) 1988-05-22
DE3776880D1 (de) 1992-04-02
IL84497A0 (en) 1988-04-29
IE59816B1 (en) 1994-04-06
LU90838I2 (fr) 2001-11-19
AU607722B2 (en) 1991-03-14
HUT46330A (en) 1988-10-28
PT86167B (pt) 1990-08-31
ATE72816T1 (de) 1992-03-15
DE10199052I1 (de) 2002-01-10
FI87570C (fi) 1993-01-25

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