NO326831B1 - Pyrimidinderivater samt anvendelse og fremgangsmate for fremstilling derav, og farmasoytisk preparat - Google Patents

Pyrimidinderivater samt anvendelse og fremgangsmate for fremstilling derav, og farmasoytisk preparat Download PDF

Info

Publication number: NO326831B1
Authority: NO; Norway
Prior art keywords: sulfamoyl; formula; compound; pharmaceutically acceptable; acceptable salt
Prior art date: 2001-02-17

Application number

NO20033635A

Other languages

English (en)

Norwegian (no)

Other versions

NO20033635L (no

NO20033635D0 (no

Inventor

Andrew Peter Thomas

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-02-17

Filing date

2003-08-15

Publication date

2009-02-23

2003-08-15 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2003-08-15 Publication of NO20033635L publication Critical patent/NO20033635L/no

2003-08-15 Publication of NO20033635D0 publication Critical patent/NO20033635D0/no

2009-02-23 Publication of NO326831B1 publication Critical patent/NO326831B1/no

Links

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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/04—Drugs for skeletal disorders for non-specific disorders of the connective tissue
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Medicinal Chemistry (AREA)
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NO20033635A 2001-02-17 2003-08-15 Pyrimidinderivater samt anvendelse og fremgangsmate for fremstilling derav, og farmasoytisk preparat NO326831B1 (no)

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CA2438646A1 (en)	2002-08-29
ES2236494T3 (es)	2005-07-16
KR20030077021A (ko)	2003-09-29
ATE288436T1 (de)	2005-02-15
AU2002231960B2 (en)	2007-10-11
EP1362050B1 (en)	2005-02-02
CA2438646C (en)	2010-03-16
IL157282A0 (en)	2004-02-19
JP2004521916A (ja)	2004-07-22
DE60202844T2 (de)	2006-01-12
CN1307179C (zh)	2007-03-28
EP1362050A1 (en)	2003-11-19
WO2002066481A1 (en)	2002-08-29
KR100829035B1 (ko)	2008-05-16
US6844341B2 (en)	2005-01-18
MY136643A (en)	2008-11-28
IL157282A (en)	2008-04-13
AR037487A1 (es)	2004-11-17
CN1524081A (zh)	2004-08-25
ZA200306081B (en)	2004-11-17
PT1362050E (pt)	2005-05-31
DK1362050T3 (da)	2005-05-09
BR0207294A (pt)	2004-03-02
NO20033635L (no)	2003-08-15
GB0103926D0 (en)	2001-04-04
DE60202844D1 (de)	2005-03-10
US20040097506A1 (en)	2004-05-20
MXPA03007351A (es)	2003-12-04
JP4421189B2 (ja)	2010-02-24
NO20033635D0 (no)	2003-08-15
NZ527367A (en)	2005-04-29

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EP2044058A1 (en)	2009-04-08	Chemical compounds
MX2008004175A (es)	2008-09-02	Imidazo[1,2-a]piridina que tiene actividad de antiproliferacion celular

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