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NO20051689L - Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonister - Google Patents

Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonister

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Publication number
NO20051689L
NO20051689L NO20051689A NO20051689A NO20051689L NO 20051689 L NO20051689 L NO 20051689L NO 20051689 A NO20051689 A NO 20051689A NO 20051689 A NO20051689 A NO 20051689A NO 20051689 L NO20051689 L NO 20051689L
Authority
NO
Norway
Prior art keywords
histamine
antagonists
diaszepines
heptanes
diazabicyclo
Prior art date
Application number
NO20051689A
Other languages
English (en)
Norwegian (no)
Other versions
NO20051689D0 (no
Inventor
Heather Hobbs
David Matthew Wilson
Rachael Anne Ancliff
Colin David Eldred
Simon Tennby Hodgson
Thomas Daniel Heightman
Yvonne C Fogden
Ashley Paul Hancock
Matthew J Lindon
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20051689D0 publication Critical patent/NO20051689D0/no
Publication of NO20051689L publication Critical patent/NO20051689L/no

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P11/00—Drugs for disorders of the respiratory system
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NO20051689A 2002-10-16 2005-04-05 Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonister NO20051689L (no)

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NO20051689D0 (no) 2005-04-05
CN101070309A (zh) 2007-11-14
CN100400523C (zh) 2008-07-09
US20100075953A1 (en) 2010-03-25
MA27482A1 (fr) 2005-08-01
NZ549963A (en) 2008-03-28
JP2006508935A (ja) 2006-03-16
WO2004035556A1 (fr) 2004-04-29
ZA200603604B (en) 2007-04-25
BR0315283A (pt) 2005-08-30
RU2005110061A (ru) 2006-01-20
US20060025404A1 (en) 2006-02-02
KR20050049553A (ko) 2005-05-25
CN1726201A (zh) 2006-01-25
EP1567511A1 (fr) 2005-08-31
NZ539446A (en) 2006-11-30
PL376477A1 (en) 2005-12-27
GB0224084D0 (en) 2002-11-27
IS7782A (is) 2005-03-31
CA2502249A1 (fr) 2004-04-29
RU2328494C2 (ru) 2008-07-10
US7615550B2 (en) 2009-11-10
AU2003280380A1 (en) 2004-05-04
ZA200502873B (en) 2006-07-26
MXPA05004078A (es) 2005-06-08

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