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NO20034836D0 - Sammensmeltede pyrimidiner som antagonister av kortikotropinfrigivelsesfaktoren (CRF) - Google Patents

Sammensmeltede pyrimidiner som antagonister av kortikotropinfrigivelsesfaktoren (CRF)

Info

Publication number
NO20034836D0
NO20034836D0 NO20034836A NO20034836A NO20034836D0 NO 20034836 D0 NO20034836 D0 NO 20034836D0 NO 20034836 A NO20034836 A NO 20034836A NO 20034836 A NO20034836 A NO 20034836A NO 20034836 D0 NO20034836 D0 NO 20034836D0
Authority
NO
Norway
Prior art keywords
crf
pyrimidines
antagonists
concentrated
release factor
Prior art date
Application number
NO20034836A
Other languages
English (en)
Other versions
NO20034836L (no
Inventor
Anna Maria Capelli
Benedetta Perini
Chiara Marchionni
Yves St-Denis
Fabrizio Micheli
Romano Di Fabio
Alessandra Pasquarello
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0110570A external-priority patent/GB0110570D0/en
Priority claimed from GB0110569A external-priority patent/GB0110569D0/en
Priority claimed from GB0110567A external-priority patent/GB0110567D0/en
Priority claimed from GB0117401A external-priority patent/GB0117401D0/en
Priority claimed from GB0117399A external-priority patent/GB0117399D0/en
Priority claimed from GB0117420A external-priority patent/GB0117420D0/en
Priority claimed from GB0203201A external-priority patent/GB0203201D0/en
Priority claimed from GB0206834A external-priority patent/GB0206834D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20034836L publication Critical patent/NO20034836L/no
Publication of NO20034836D0 publication Critical patent/NO20034836D0/no

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
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    • A61K51/04Organic compounds
    • A61K51/041Heterocyclic compounds
    • A61K51/044Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0459Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
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    • A61K51/041Heterocyclic compounds
    • A61K51/044Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0463Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • A61K51/04Organic compounds
    • A61K51/041Heterocyclic compounds
    • A61K51/044Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0465Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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    • CCHEMISTRY; METALLURGY
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    • C07D239/72Quinazolines; Hydrogenated quinazolines
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    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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NO20034836A 2001-04-30 2003-10-29 Sammensmeltede pyrimidiner som antagonister av kortikotropinfrigivelsesfaktoren (CRF) NO20034836D0 (no)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
GB0110570A GB0110570D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110569A GB0110569D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110567A GB0110567D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0117401A GB0117401D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117399A GB0117399D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117420A GB0117420D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0203201A GB0203201D0 (en) 2002-02-11 2002-02-11 Chemical compounds
GB0206834A GB0206834D0 (en) 2002-03-22 2002-03-22 Chemical compounds
PCT/GB2002/002029 WO2002088095A1 (en) 2001-04-30 2002-04-30 Fused pyrimidines as antagonists of the corticotropin releasing factor (crf)

Publications (2)

Publication Number Publication Date
NO20034836L NO20034836L (no) 2003-10-29
NO20034836D0 true NO20034836D0 (no) 2003-10-29

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Application Number Title Priority Date Filing Date
NO20034836A NO20034836D0 (no) 2001-04-30 2003-10-29 Sammensmeltede pyrimidiner som antagonister av kortikotropinfrigivelsesfaktoren (CRF)

Country Status (19)

Country Link
US (1) US7279474B2 (no)
EP (1) EP1383747B1 (no)
JP (1) JP2004528349A (no)
KR (1) KR20040015206A (no)
CN (1) CN1649848A (no)
AR (1) AR033295A1 (no)
AT (1) ATE386727T1 (no)
AU (1) AU2002253357B2 (no)
BR (1) BR0209267A (no)
CA (1) CA2446514A1 (no)
CZ (1) CZ20032946A3 (no)
DE (1) DE60225127T2 (no)
ES (1) ES2301633T3 (no)
HU (1) HUP0304054A2 (no)
IL (1) IL158062A0 (no)
MX (1) MXPA03009938A (no)
NO (1) NO20034836D0 (no)
PL (1) PL366934A1 (no)
WO (1) WO2002088095A1 (no)

Families Citing this family (66)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1395591B1 (en) * 2001-06-12 2008-06-04 Glaxo Group Limited Corticotropin releasing factor antagonists
GB0117396D0 (en) * 2001-07-17 2001-09-05 Glaxo Group Ltd Chemical compounds
US20070066640A1 (en) * 2003-01-16 2007-03-22 Emiliano Castiglioni Heteroaryl-substituted pyrrolo'2,3-b1 pyridine derivatives as crf receptor antagonists
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
GB0308208D0 (en) 2003-04-09 2003-05-14 Glaxo Group Ltd Chemical compounds
AU2004235907B2 (en) * 2003-05-05 2007-08-30 F. Hoffmann La-Roche Ag Fused pyrimidine derivatives with CRF activity
EP1656145A1 (en) 2003-08-12 2006-05-17 F. Hoffmann-La Roche Ag Spiro-substituted tetrahydroquinazolines as corticotropin releasing factor (cfr) antagonists
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US20040176400A1 (en) 2004-09-09
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MXPA03009938A (es) 2005-09-07
US7279474B2 (en) 2007-10-09
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WO2002088095A1 (en) 2002-11-07
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IL158062A0 (en) 2004-03-28
AR033295A1 (es) 2003-12-10
EP1383747B1 (en) 2008-02-20
BR0209267A (pt) 2004-06-15
CZ20032946A3 (en) 2004-05-12
PL366934A1 (en) 2005-02-07
ATE386727T1 (de) 2008-03-15
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