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NO20013072L - Nitrogenholdige heterocykler som faktor Xa-inhibitorer - Google Patents

Nitrogenholdige heterocykler som faktor Xa-inhibitorer

Info

Publication number
NO20013072L
NO20013072L NO20013072A NO20013072A NO20013072L NO 20013072 L NO20013072 L NO 20013072L NO 20013072 A NO20013072 A NO 20013072A NO 20013072 A NO20013072 A NO 20013072A NO 20013072 L NO20013072 L NO 20013072L
Authority
NO
Norway
Prior art keywords
inhibitors
nitrogen
factor
containing heterocycles
heterocycles
Prior art date
Application number
NO20013072A
Other languages
English (en)
Other versions
NO319816B1 (no
NO20013072D0 (no
Inventor
John Matthew Fevig
Joseph Cacciola
Charles G Clark
Patrick Yuk-Sun Lam
Donald J P Pinto
James Russell Pruitt
Karen Anita Rossi
Qui Han
Mimi Lifen Quan
Original Assignee
Du Pont Pharm Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26811284&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20013072(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Du Pont Pharm Co filed Critical Du Pont Pharm Co
Publication of NO20013072D0 publication Critical patent/NO20013072D0/no
Publication of NO20013072L publication Critical patent/NO20013072L/no
Publication of NO319816B1 publication Critical patent/NO319816B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO20013072A 1998-12-23 2001-06-20 Nitrogenholdige heterocykler,anvendelse av disse for fremstilling av medikamenter samt farmasoytiske preparater. NO319816B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11362898P 1998-12-23 1998-12-23
US12763399P 1999-04-02 1999-04-02
PCT/US1999/030316 WO2000039131A1 (en) 1998-12-23 1999-12-17 Nitrogen containing heterobicycles as factor xa inhibitors

Publications (3)

Publication Number Publication Date
NO20013072D0 NO20013072D0 (no) 2001-06-20
NO20013072L true NO20013072L (no) 2001-06-20
NO319816B1 NO319816B1 (no) 2005-09-19

Family

ID=26811284

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20013072A NO319816B1 (no) 1998-12-23 2001-06-20 Nitrogenholdige heterocykler,anvendelse av disse for fremstilling av medikamenter samt farmasoytiske preparater.

Country Status (26)

Country Link
US (2) US6413980B1 (no)
EP (1) EP1140941B1 (no)
JP (1) JP2002533465A (no)
KR (1) KR100628407B1 (no)
CN (1) CN100340559C (no)
AR (1) AR024242A1 (no)
AT (1) ATE280171T1 (no)
AU (1) AU759711B2 (no)
BR (1) BR9917080A (no)
CA (1) CA2349330C (no)
DE (1) DE69921358T2 (no)
DK (1) DK1140941T3 (no)
EA (1) EA004515B1 (no)
ES (1) ES2232202T3 (no)
HK (1) HK1052508B (no)
HR (1) HRP990396A2 (no)
IL (2) IL142959A0 (no)
MX (1) MXPA01006502A (no)
MY (1) MY138239A (no)
NO (1) NO319816B1 (no)
NZ (1) NZ511674A (no)
PT (1) PT1140941E (no)
SI (1) SI1140941T1 (no)
TW (1) TWI225862B (no)
WO (1) WO2000039131A1 (no)
ZA (1) ZA200103795B (no)

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US20040077605A1 (en) * 2001-06-20 2004-04-22 Salvati Mark E. Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
EP1854798A3 (en) 2000-09-19 2007-11-28 Bristol-Myers Squibb Company Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
US20040087548A1 (en) 2001-02-27 2004-05-06 Salvati Mark E. Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
US6960595B2 (en) * 2001-03-23 2005-11-01 Bristol-Myers Squibb Pharma Company 5-6 to 5-7 Heterobicycles as factor Xa inhibitors
US6750225B2 (en) 2001-04-18 2004-06-15 Bristol-Myers Squibb Pharms Company 1,4,5,6-tetrahydropyrazolo-[3,4,-c]-pyridin-7-ones useful as factor Xa inhibitors
CA2441772A1 (en) * 2001-04-18 2002-10-31 Bristol-Myers Squibb Company 1,4,5,6-tetrahydropyrazolo-¬3,4-c|-pyridin-7-ones as factor xa inhibitors
WO2002094197A2 (en) * 2001-05-22 2002-11-28 Bristol-Myers Squibb Company Bicyclic inhibitors of factor xa
TWI320039B (en) 2001-09-21 2010-02-01 Lactam-containing compounds and derivatives thereof as factor xa inhibitors
IL160693A0 (en) * 2001-09-21 2004-08-31 Bristol Myers Squibb Co Lactam-containing compounds and derivatives thereof as factor xa inhibitors
WO2003048081A2 (en) * 2001-12-04 2003-06-12 Bristol-Myers Squibb Company Glycinamides as factor xa inhibitors
TW200302225A (en) 2001-12-04 2003-08-01 Bristol Myers Squibb Co Substituted amino methyl factor Xa inhibitors
TW200303201A (en) 2001-12-10 2003-09-01 Bristol Myers Squibb Co Synthesis of 4,5-dihydro-pyrazolo [3,4-c] pyrid-2-ones
AU2002364082A1 (en) * 2001-12-19 2003-07-09 Bristol-Myers Squibb Company Fused heterocyclic compounds and analogs thereof: modulators of nuclear hormone receptor function
WO2003075921A2 (en) * 2002-03-05 2003-09-18 Transtech Pharma, Inc. Mono- and bicyclic azole derivatives that inhibit the interaction of ligands with rage
EP1505966A4 (en) * 2002-05-10 2006-08-30 Bristol Myers Squibb Co 1,1-DISUBSTITUTED CYCLOALKYL DERIVATIVES AS FACTOR XA HEMMER
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CN104530029B (zh) * 2014-12-09 2017-04-12 广东东阳光药业有限公司 作为Xa因子抑制剂的杂环化合物及其使用方法和用途
CN104513239B (zh) * 2014-12-10 2017-08-22 沈阳药科大学 吡唑并[3,4‑c]吡啶‑7‑酮类化合物及其应用
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KR102128509B1 (ko) * 2018-12-19 2020-07-01 한국과학기술연구원 말단 아민기에 아릴 또는 헤테로아릴기가 치환된 신규한 히드라존 유도체 및 이의 용도
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Also Published As

Publication number Publication date
SI1140941T1 (en) 2005-04-30
CA2349330A1 (en) 2000-07-06
DK1140941T3 (da) 2005-02-14
MY138239A (en) 2009-05-29
EP1140941A1 (en) 2001-10-10
HK1052508A1 (zh) 2003-09-19
NO319816B1 (no) 2005-09-19
NZ511674A (en) 2003-11-28
NO20013072D0 (no) 2001-06-20
EA200100688A1 (ru) 2001-12-24
HK1052508B (zh) 2008-08-01
PT1140941E (pt) 2005-02-28
IL142959A (en) 2010-05-31
CN100340559C (zh) 2007-10-03
AR024242A1 (es) 2002-09-25
KR20010092754A (ko) 2001-10-26
ES2232202T3 (es) 2005-05-16
DE69921358D1 (de) 2004-11-25
IL142959A0 (en) 2002-04-21
US6673810B2 (en) 2004-01-06
HRP990396A2 (en) 2000-08-31
WO2000039131A1 (en) 2000-07-06
US20030004167A1 (en) 2003-01-02
CA2349330C (en) 2009-09-29
KR100628407B1 (ko) 2006-09-26
AU2371700A (en) 2000-07-31
CN1391575A (zh) 2003-01-15
TWI225862B (en) 2005-01-01
JP2002533465A (ja) 2002-10-08
ZA200103795B (en) 2002-08-12
DE69921358T2 (de) 2006-03-09
US6413980B1 (en) 2002-07-02
BR9917080A (pt) 2002-03-12
AU759711B2 (en) 2003-04-17
EA004515B1 (ru) 2004-04-29
MXPA01006502A (es) 2002-04-08
ATE280171T1 (de) 2004-11-15
EP1140941B1 (en) 2004-10-20

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