NO20013809L - Indolderivater og anvendelse derav som MCP-1 antagonister - Google Patents
Indolderivater og anvendelse derav som MCP-1 antagonisterInfo
- Publication number
- NO20013809L NO20013809L NO20013809A NO20013809A NO20013809L NO 20013809 L NO20013809 L NO 20013809L NO 20013809 A NO20013809 A NO 20013809A NO 20013809 A NO20013809 A NO 20013809A NO 20013809 L NO20013809 L NO 20013809L
- Authority
- NO
- Norway
- Prior art keywords
- mcp
- antagonists
- indole derivatives
- indole
- derivatives
- Prior art date
Links
- 229940123313 MCP-1 antagonist Drugs 0.000 title 1
- 229940054051 antipsychotic indole derivative Drugs 0.000 title 1
- 150000002475 indoles Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9902461.4A GB9902461D0 (en) | 1999-02-05 | 1999-02-05 | Chemical compounds |
| PCT/GB2000/000265 WO2000046196A1 (en) | 1999-02-05 | 2000-01-31 | Indole derivatives and their use as mcp-1 antagonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20013809D0 NO20013809D0 (no) | 2001-08-03 |
| NO20013809L true NO20013809L (no) | 2001-10-02 |
Family
ID=10847084
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20013809A NO20013809L (no) | 1999-02-05 | 2001-08-03 | Indolderivater og anvendelse derav som MCP-1 antagonister |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US6737435B1 (id) |
| EP (1) | EP1150952B1 (id) |
| JP (1) | JP2002536359A (id) |
| KR (1) | KR20010094755A (id) |
| CN (1) | CN1339025A (id) |
| AR (1) | AR022461A1 (id) |
| AT (1) | ATE280757T1 (id) |
| AU (1) | AU770856B2 (id) |
| BR (1) | BR0007984A (id) |
| CA (1) | CA2356898A1 (id) |
| CZ (1) | CZ20012807A3 (id) |
| DE (1) | DE60015296T2 (id) |
| EE (1) | EE200100403A (id) |
| GB (1) | GB9902461D0 (id) |
| HU (1) | HUP0105079A3 (id) |
| ID (1) | ID30401A (id) |
| IL (1) | IL144611A0 (id) |
| IS (1) | IS5980A (id) |
| MY (1) | MY133209A (id) |
| NO (1) | NO20013809L (id) |
| NZ (1) | NZ512680A (id) |
| PL (1) | PL350184A1 (id) |
| RU (1) | RU2235090C2 (id) |
| SK (1) | SK11152001A3 (id) |
| TR (1) | TR200102233T2 (id) |
| WO (1) | WO2000046196A1 (id) |
| ZA (1) | ZA200105311B (id) |
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| GB9902461D0 (en) | 1999-02-05 | 1999-03-24 | Zeneca Ltd | Chemical compounds |
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-
1999
- 1999-02-05 GB GBGB9902461.4A patent/GB9902461D0/en not_active Ceased
-
2000
- 2000-01-31 AR ARP000100407A patent/AR022461A1/es not_active Application Discontinuation
- 2000-01-31 CN CN00803463A patent/CN1339025A/zh active Pending
- 2000-01-31 PL PL00350184A patent/PL350184A1/xx not_active Application Discontinuation
- 2000-01-31 SK SK1115-2001A patent/SK11152001A3/sk unknown
- 2000-01-31 IL IL14461100A patent/IL144611A0/xx unknown
- 2000-01-31 ID IDW00200101667A patent/ID30401A/id unknown
- 2000-01-31 US US09/889,599 patent/US6737435B1/en not_active Expired - Fee Related
- 2000-01-31 DE DE60015296T patent/DE60015296T2/de not_active Expired - Lifetime
- 2000-01-31 RU RU2001124567/04A patent/RU2235090C2/ru not_active IP Right Cessation
- 2000-01-31 EP EP20000901259 patent/EP1150952B1/en not_active Expired - Lifetime
- 2000-01-31 AU AU21213/00A patent/AU770856B2/en not_active Ceased
- 2000-01-31 BR BR0007984-7A patent/BR0007984A/pt not_active IP Right Cessation
- 2000-01-31 WO PCT/GB2000/000265 patent/WO2000046196A1/en not_active Ceased
- 2000-01-31 NZ NZ512680A patent/NZ512680A/en unknown
- 2000-01-31 HU HU0105079A patent/HUP0105079A3/hu unknown
- 2000-01-31 EE EEP200100403A patent/EE200100403A/xx unknown
- 2000-01-31 TR TR2001/02233T patent/TR200102233T2/xx unknown
- 2000-01-31 JP JP2000597267A patent/JP2002536359A/ja active Pending
- 2000-01-31 KR KR1020017009862A patent/KR20010094755A/ko not_active Withdrawn
- 2000-01-31 CZ CZ20012807A patent/CZ20012807A3/cs unknown
- 2000-01-31 CA CA002356898A patent/CA2356898A1/en not_active Abandoned
- 2000-01-31 AT AT00901259T patent/ATE280757T1/de not_active IP Right Cessation
- 2000-02-04 MY MYPI20000404A patent/MY133209A/en unknown
-
2001
- 2001-06-26 IS IS5980A patent/IS5980A/is unknown
- 2001-06-27 ZA ZA200105311A patent/ZA200105311B/en unknown
- 2001-08-03 NO NO20013809A patent/NO20013809L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| RU2001124567A (ru) | 2004-01-10 |
| DE60015296T2 (de) | 2006-02-02 |
| EE200100403A (et) | 2002-10-15 |
| NZ512680A (en) | 2003-11-28 |
| NO20013809D0 (no) | 2001-08-03 |
| TR200102233T2 (tr) | 2001-12-21 |
| SK11152001A3 (sk) | 2001-12-03 |
| ATE280757T1 (de) | 2004-11-15 |
| AR022461A1 (es) | 2002-09-04 |
| EP1150952A1 (en) | 2001-11-07 |
| CZ20012807A3 (cs) | 2001-10-17 |
| JP2002536359A (ja) | 2002-10-29 |
| KR20010094755A (ko) | 2001-11-01 |
| ID30401A (id) | 2001-11-29 |
| PL350184A1 (en) | 2002-11-18 |
| MY133209A (en) | 2007-10-31 |
| IS5980A (is) | 2001-06-26 |
| RU2235090C2 (ru) | 2004-08-27 |
| GB9902461D0 (en) | 1999-03-24 |
| CA2356898A1 (en) | 2000-08-10 |
| CN1339025A (zh) | 2002-03-06 |
| WO2000046196A1 (en) | 2000-08-10 |
| US6737435B1 (en) | 2004-05-18 |
| DE60015296D1 (de) | 2004-12-02 |
| HUP0105079A2 (hu) | 2002-04-29 |
| BR0007984A (pt) | 2001-11-06 |
| ZA200105311B (en) | 2002-09-27 |
| AU2121300A (en) | 2000-08-25 |
| HUP0105079A3 (en) | 2002-11-28 |
| EP1150952B1 (en) | 2004-10-27 |
| AU770856B2 (en) | 2004-03-04 |
| IL144611A0 (en) | 2002-05-23 |
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| FC2A | Withdrawal, rejection or dismissal of laid open patent application |