NO20010559D0 - Fremgangsmåte for syntese av (1H)-benzo[c]kinolizin-3-ones derivater - Google Patents

Fremgangsmåte for syntese av (1H)-benzo[c]kinolizin-3-ones derivater

Info

Publication number: NO20010559D0
Authority: NO; Norway
Prior art keywords: quinolizin; benzo; synthesis; ones derivatives; compounds
Prior art date: 1998-08-03

Application number

NO20010559A

Other languages

English (en)

Norwegian (no)

Other versions

NO20010559L (no

Inventor

Antonio Guarna

Mario Serio

Ernesto Giovanni Occhiato

Original Assignee

Serono Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-08-03

Filing date

2001-02-01

Publication date

2001-02-01

2001-02-01 Application filed by Serono Lab filed Critical Serono Lab

2001-02-01 Publication of NO20010559D0 publication Critical patent/NO20010559D0/no

2001-02-01 Publication of NO20010559L publication Critical patent/NO20010559L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/03—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/04—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Dermatology (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Inorganic Compounds Of Heavy Metals (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Carbon And Carbon Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

NO20010559A 1998-08-03 2001-02-01 Fremgangsmate for syntese av (1H)-benzo[c]kinolizin-3-ones derivater NO20010559L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP98114524		1998-08-03
PCT/EP1999/005277 WO2000008019A1 (en)	1998-08-03	1999-07-23	Process for the synthesis of (1h)-benzo[c]quinolizin-3-ones derivatives

Publications (2)

Publication Number	Publication Date
NO20010559D0 true NO20010559D0 (no)	2001-02-01
NO20010559L NO20010559L (no)	2001-02-01

Family

ID=8232396

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20010559A NO20010559L (no)	1998-08-03	2001-02-01	Fremgangsmate for syntese av (1H)-benzo[c]kinolizin-3-ones derivater

Country Status (28)

Country	Link
US (1)	US6723850B1 (pt)
EP (1)	EP1102765B1 (pt)
JP (1)	JP2002522435A (pt)
KR (1)	KR100624239B1 (pt)
CN (1)	CN1128148C (pt)
AT (1)	ATE250057T1 (pt)
AU (1)	AU751873B2 (pt)
BG (1)	BG65062B1 (pt)
BR (1)	BR9912870A (pt)
CA (1)	CA2338498C (pt)
CZ (1)	CZ291648B6 (pt)
DE (1)	DE69911430T2 (pt)
DK (1)	DK1102765T3 (pt)
EA (1)	EA003997B1 (pt)
EE (1)	EE04642B1 (pt)
ES (1)	ES2203169T3 (pt)
HU (1)	HUP0103241A3 (pt)
IL (2)	IL141212A0 (pt)
NO (1)	NO20010559L (pt)
NZ (1)	NZ509243A (pt)
PL (1)	PL198963B1 (pt)
PT (1)	PT1102765E (pt)
SI (1)	SI1102765T1 (pt)
SK (1)	SK285438B6 (pt)
TR (1)	TR200100286T2 (pt)
UA (1)	UA67787C2 (pt)
WO (1)	WO2000008019A1 (pt)
ZA (1)	ZA200100365B (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7495103B2 (en)	2004-06-24	2009-02-24	Vertex Pharmaceuticals Incorporated	Modulators of ATP-binding cassette transporters
US8354427B2 (en) *	2004-06-24	2013-01-15	Vertex Pharmaceutical Incorporated	Modulators of ATP-binding cassette transporters
EP1979367A2 (en) *	2005-12-24	2008-10-15	Vertex Pharmaceuticals Incorporated	Quinolin-4-one derivatives as modulators of abc transporters
CA2635581C (en)	2005-12-28	2017-02-28	Vertex Pharmaceuticals Incorporated	Solid forms of n-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide
US20100074949A1 (en)	2008-08-13	2010-03-25	William Rowe	Pharmaceutical composition and administration thereof
US12458635B2 (en)	2008-08-13	2025-11-04	Vertex Pharmaceuticals Incorporated	Pharmaceutical composition and administrations thereof
SMT201700593T1 (it)	2009-03-20	2018-03-08	Vertex Pharma	Procedimento per preparare modulatori di regolatore di conduttanza transmembrana di fibrosi cistica
US8802700B2 (en)	2010-12-10	2014-08-12	Vertex Pharmaceuticals Incorporated	Modulators of ATP-Binding Cassette transporters
ES2524422T3 (es) *	2010-12-14	2014-12-09	Syngenta Participations Ag	Derivados de estrigolactamas y su uso como reguladores del crecimiento vegetal
JP2015511583A (ja)	2012-02-27	2015-04-20	バーテックスファーマシューティカルズインコーポレイテッドＶｅｒｔｅｘＰｈａｒｍａｃｅｕｔｉｃａｌｓＩｎｃｏｒｐｏｒａｔｅｄ	薬学的組成物およびその投与
CA2963945C (en)	2014-10-07	2023-01-10	Vertex Pharmaceuticals Incorporated	Co-crystals of modulators of cystic fibrosis transmembrane conductance regulator
CN105001216B (zh) *	2015-07-08	2017-03-01	中国科学院兰州化学物理研究所	一种喹嗪酮的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5064961A (en) *	1989-12-18	1991-11-12	E. R. Squibb & Sons, Inc.	Process for preparing an optically active cyclobutane nucleoside
FR2696465B1 (fr) *	1992-10-02	1994-12-23	Adir	Nouveaux dérivés d'ellipticine, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
IT1286545B1 (it) *	1996-02-09	1998-07-15	Antonio Guarna	Derivati benzo(c) chinolizinici,loro preparazione ed uso come inibitori delle 5-alfa-riduttasi
JPH09316076A (ja) *	1996-05-24	1997-12-09	Nippon Paper Ind Co Ltd	９−置換プリン誘導体及びその抗ウイルス剤としての用途

1999
- 1999-07-23 HU HU0103241A patent/HUP0103241A3/hu unknown
- 1999-07-23 KR KR1020017000325A patent/KR100624239B1/ko not_active Expired - Fee Related
- 1999-07-23 EE EEP200100060A patent/EE04642B1/xx not_active IP Right Cessation
- 1999-07-23 PL PL345802A patent/PL198963B1/pl not_active IP Right Cessation
- 1999-07-23 EA EA200100213A patent/EA003997B1/ru not_active IP Right Cessation
- 1999-07-23 IL IL14121299A patent/IL141212A0/xx active IP Right Grant
- 1999-07-23 TR TR2001/00286T patent/TR200100286T2/xx unknown
- 1999-07-23 CZ CZ2001434A patent/CZ291648B6/cs not_active IP Right Cessation
- 1999-07-23 EP EP99941269A patent/EP1102765B1/en not_active Expired - Lifetime
- 1999-07-23 ES ES99941269T patent/ES2203169T3/es not_active Expired - Lifetime
- 1999-07-23 AU AU63123/99A patent/AU751873B2/en not_active Ceased
- 1999-07-23 DK DK99941269T patent/DK1102765T3/da active
- 1999-07-23 UA UA2001020777A patent/UA67787C2/uk unknown
- 1999-07-23 PT PT99941269T patent/PT1102765E/pt unknown
- 1999-07-23 NZ NZ509243A patent/NZ509243A/xx not_active IP Right Cessation
- 1999-07-23 JP JP2000563652A patent/JP2002522435A/ja active Pending
- 1999-07-23 SK SK167-2001A patent/SK285438B6/sk not_active IP Right Cessation
- 1999-07-23 AT AT99941269T patent/ATE250057T1/de not_active IP Right Cessation
- 1999-07-23 DE DE69911430T patent/DE69911430T2/de not_active Expired - Fee Related
- 1999-07-23 CA CA002338498A patent/CA2338498C/en not_active Expired - Fee Related
- 1999-07-23 BR BR9912870-5A patent/BR9912870A/pt not_active Application Discontinuation
- 1999-07-23 WO PCT/EP1999/005277 patent/WO2000008019A1/en not_active Ceased
- 1999-07-23 US US09/743,373 patent/US6723850B1/en not_active Expired - Fee Related
- 1999-07-23 SI SI9930419T patent/SI1102765T1/xx unknown
- 1999-07-23 CN CN99809204A patent/CN1128148C/zh not_active Expired - Fee Related
2001
- 2001-01-12 ZA ZA200100365A patent/ZA200100365B/en unknown
- 2001-01-30 BG BG105198A patent/BG65062B1/bg unknown
- 2001-02-01 IL IL141212A patent/IL141212A/en not_active IP Right Cessation
- 2001-02-01 NO NO20010559A patent/NO20010559L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
CN1311788A (zh)	2001-09-05
BR9912870A (pt)	2001-10-16
DE69911430T2 (de)	2004-07-22
CZ2001434A3 (cs)	2001-08-15
ZA200100365B (en)	2001-07-26
KR100624239B1 (ko)	2006-09-13
AU751873B2 (en)	2002-08-29
PL345802A1 (en)	2002-01-02
ES2203169T3 (es)	2004-04-01
EE04642B1 (et)	2006-06-15
HUP0103241A3 (en)	2002-10-28
BG105198A (en)	2001-12-29
BG65062B1 (bg)	2007-01-31
KR20010074684A (ko)	2001-08-09
NZ509243A (en)	2002-11-26
EP1102765B1 (en)	2003-09-17
DE69911430D1 (de)	2003-10-23
WO2000008019A1 (en)	2000-02-17
HUP0103241A2 (hu)	2002-01-28
IL141212A (en)	2006-12-31
IL141212A0 (en)	2002-03-10
DK1102765T3 (da)	2004-02-02
EA003997B1 (ru)	2003-12-25
CA2338498C (en)	2009-05-19
CN1128148C (zh)	2003-11-19
HK1037368A1 (en)	2002-02-08
SK285438B6 (sk)	2007-01-04
UA67787C2 (uk)	2004-07-15
TR200100286T2 (tr)	2001-07-23
EA200100213A1 (ru)	2001-08-27
SK1672001A3 (en)	2001-08-06
JP2002522435A (ja)	2002-07-23
US6723850B1 (en)	2004-04-20
ATE250057T1 (de)	2003-10-15
PT1102765E (pt)	2003-12-31
SI1102765T1 (en)	2003-12-31
EP1102765A1 (en)	2001-05-30
AU6312399A (en)	2000-02-28
CA2338498A1 (en)	2000-02-17
NO20010559L (no)	2001-02-01
PL198963B1 (pl)	2008-08-29
CZ291648B6 (cs)	2003-04-16
EE200100060A (et)	2002-06-17

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DE60204452D1 (de)	2005-07-07	Pyrazolo[1,5]pyridinderivate
IL135536A0 (en)	2001-05-20	Ortho-anthranilamide derivatives and pharmaceutical compositions containing the same
BG106340A (en)	2002-10-31	Substituted oxoazaheterocyclyl compounds
DE69831868D1 (en)	2006-02-23	Antithrombosemittel
ATE253545T1 (de)	2003-11-15	Biarylessigsäure-derivate und ihre verwendung als cox-2 inhibitoren
EA199700124A1 (ru)	1997-12-30	Производные гуанина
DE69709938D1 (de)	2002-02-28	N-benzylpiperidin- und tetrahydropyridin-derivate
WO2005005389A3 (en)	2005-03-24	Malonamide derivatives
NO20010559L (no)	2001-02-01	Fremgangsmate for syntese av (1H)-benzo[c]kinolizin-3-ones derivater
ZA200404752B (en)	2005-04-26	6-aminomorphinane derivatives method for the production and use thereof
WO2004050663A3 (en)	2004-10-28	An improved process for the preparation of cefuroxime sodium
DE60114640D1 (en)	2005-12-08	Antithrombosemittel
UA66866C2 (uk)	2004-06-15	Синтез морфолінових похідних
DE60235365D1 (de)	2010-04-01	Verfahren zur herstellung von 7-amino-syn-3,5-dihydroxyheptansäurederivaten und zwischenverbindungen diesesverfahrens und deren herestellung
AU2002357740A1 (en)	2003-06-23	Pyrazolo-pyridine derivatives as antiherpes agents
TR200003065T2 (tr)	2001-02-21	Nöraminidazların inhibitörleri olarak pirolidinler.
HUP0104213A2 (hu)	2002-03-28	Vankoreszmicin, eljárás előállítására és gyógyszerként történő alkalmazása
NO20052197L (no)	2005-05-04	Fremgangsmate for fremstilling av pyrazol
MX2022002533A (es)	2022-06-02	Ácidos nucleicos modificados con ligandos 2', síntesis de estos y compuestos intermedios de estos.
DE60006125D1 (de)	2003-11-27	Herstellung von 2-(2-arylmorpholin-2-yl)ethanolderivaten und zwischenprodukte
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BG104964A (bg)	2001-07-31	Подобрен метод за получаване на фармацевтично ценни норбензоморфанови производни
NO20020561L (no)	2002-02-05	Fremgangsmåte for fremstilling av syrer via alfa-klorepoksi- estere
MXPA03003466A (es)	2004-09-10	Derivados de piranosido.

Legal Events

Date	Code	Title	Description
2008-01-14	CREP	Change of representative	Representative=s name: ONSAGERS AS, POSTBOKS 6963 ST OLAVS PLASS, 0130 OS
2010-06-07	FC2A	Withdrawal, rejection or dismissal of laid open patent application