[go: up one dir, main page]

NO20005743L - Fremgangsmåte til fremstilling av 4,5-epoksymorfinan-6- glukuronider - Google Patents

Fremgangsmåte til fremstilling av 4,5-epoksymorfinan-6- glukuronider

Info

Publication number
NO20005743L
NO20005743L NO20005743A NO20005743A NO20005743L NO 20005743 L NO20005743 L NO 20005743L NO 20005743 A NO20005743 A NO 20005743A NO 20005743 A NO20005743 A NO 20005743A NO 20005743 L NO20005743 L NO 20005743L
Authority
NO
Norway
Prior art keywords
epoxymorphinan
glucuronides
preparation
Prior art date
Application number
NO20005743A
Other languages
English (en)
Other versions
NO20005743D0 (no
Inventor
Arie L Gutman
Genadi Nisnevitch
Lev Yudovitch
Igor Rokhman
Original Assignee
Cenes Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from IL12446098A external-priority patent/IL124460A0/xx
Application filed by Cenes Ltd filed Critical Cenes Ltd
Publication of NO20005743D0 publication Critical patent/NO20005743D0/no
Publication of NO20005743L publication Critical patent/NO20005743L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Neurosurgery (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
NO20005743A 1998-05-13 2000-11-13 Fremgangsmåte til fremstilling av 4,5-epoksymorfinan-6- glukuronider NO20005743L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IL12446098A IL124460A0 (en) 1998-05-13 1998-05-13 Preparation of per-o-acylated alkyl 4,5-epoxymorphinane-6-beta-D-glucuronides
GB9900832 1999-01-15
PCT/GB1999/001508 WO1999058545A1 (en) 1998-05-13 1999-05-12 Process for preparation of 4,5-epoxymorphinan-6-oxyglucuronides

Publications (2)

Publication Number Publication Date
NO20005743D0 NO20005743D0 (no) 2000-11-13
NO20005743L true NO20005743L (no) 2001-01-03

Family

ID=26314988

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20005743A NO20005743L (no) 1998-05-13 2000-11-13 Fremgangsmåte til fremstilling av 4,5-epoksymorfinan-6- glukuronider

Country Status (9)

Country Link
US (2) US6737518B1 (no)
EP (1) EP1077985A1 (no)
JP (1) JP2002514655A (no)
AU (1) AU761629B2 (no)
CA (1) CA2331866A1 (no)
HU (1) HUP0102297A3 (no)
NO (1) NO20005743L (no)
PL (1) PL344141A1 (no)
WO (1) WO1999058545A1 (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2568249C (en) * 2004-05-28 2014-12-09 Human Biomolecular Research Institute Synthesis of metabolically stable analgesics, pain medications and other agents
ITRM20130223A1 (it) * 2013-04-15 2014-10-16 Rosario Nicoletti Derivati della codeina come inibitori della glucuronazione della morfina
CN103864866B (zh) * 2014-03-26 2016-05-25 宜昌人福药业有限责任公司 一种吗啡-6-β-D-葡萄糖醛酸苷的合成方法及其中间体化合物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9116909D0 (en) * 1991-08-06 1991-09-18 Salford Ultrafine Chem & Res Morphine derivatives
FR2680786B1 (fr) 1991-09-04 1995-03-10 Irepa Procede de synthese de glucuronides d'epoxy-4,5 morphinanes.

Also Published As

Publication number Publication date
PL344141A1 (en) 2001-10-08
AU761629B2 (en) 2003-06-05
CA2331866A1 (en) 1999-11-18
HUP0102297A2 (hu) 2001-10-28
EP1077985A1 (en) 2001-02-28
HUP0102297A3 (en) 2003-07-28
JP2002514655A (ja) 2002-05-21
NO20005743D0 (no) 2000-11-13
US20040053854A1 (en) 2004-03-18
US6737518B1 (en) 2004-05-18
AU4050499A (en) 1999-11-29
WO1999058545A1 (en) 1999-11-18

Similar Documents

Publication Publication Date Title
NO20011936L (no) Fremgangsmate for fremstilling av citalopram
NO980707D0 (no) Fremgangsmåte til fremstilling av kopolymerer
NO20011214L (no) Fremgangsmåte for fremstilling av aromatiske aldehyder
NO981800D0 (no) FremgangsmÕte for fremstilling av 1,1,1,3,3-pentafluorpentan
IS5952A (is) Aðferð til framleiðslu á 5-sýanóþalíði
EP1023250A4 (en) METHOD FOR PRODUCING 2,6-DIALKYLNAPHTHALINE
NO993912L (no) FremgangsmÕte for fremstilling av eprosartan
NO20000933D0 (no) Fremgangsmåte for fremstilling av polymer
NO20005424L (no) Fremgangsmåte ved fremstilling av 1,3-disubstituert-4- oksocykliske ureaer
DK0815092T3 (da) Fremgangsmåde til fremstilling af 1,2-benzisothiazolin-3-oner
NO993913D0 (no) Fremgangsmåte for fremstilling av eprosartan
NO20000456D0 (no) Fremgangsmåte for fremstilling av 1,2-dikloretan
NO985535L (no) FremgangsmÕte for fremstilling av 1,3-alkandioler
NO996432L (no) Fremgangsmåte for fremstilling av 4-substituert-1H-indol-3- glykosamider
DK0735043T3 (da) Fremgangsmåde til fremstilling af 2-substitueret 3,3-difluorfuran
NO20005425L (no) Fremgangsmåte ved fremstilling av 1,3-disubstituert-4- oksocykliske ureaer
NO20005743L (no) Fremgangsmåte til fremstilling av 4,5-epoksymorfinan-6- glukuronider
NO20011652L (no) Fremgangsmåte for fremstilling av 1,5-diaryl-3-substituerte pyrazoler
FI964829A0 (fi) Menetelmä 2,2,4-trimetyyli-1,3-pentaanidioli-isobutyraatin valmistamiseksi
NO20012811D0 (no) Fremgangsmåte for fremstilling av p-klorfenyl-propanol- derivat
TR199900757A3 (tr) Fenoksifenilsülfonil halidlerin hazirlanmasi için islem.
NO20003077L (no) FremgangsmÕte for fremstilling av klorbenzooksazolen
NO994557D0 (no) Fremgangsmaate for fremstilling av arylaminotriazolopyridiner
NO20013044D0 (no) Fremgangsmåte for fremstilling av NG-substituerte deaza- adenosinderivater
ZA991215B (en) Process for the preparation of 1,3-disubstituted 2-nitroguanidines.