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NO176099C - Analogifremgangsmåte for fremstilling av terapeutisk aktive 4-(2-okso-3-pyridyl)-kromanderivater - Google Patents

Analogifremgangsmåte for fremstilling av terapeutisk aktive 4-(2-okso-3-pyridyl)-kromanderivater

Info

Publication number
NO176099C
NO176099C NO903043A NO903043A NO176099C NO 176099 C NO176099 C NO 176099C NO 903043 A NO903043 A NO 903043A NO 903043 A NO903043 A NO 903043A NO 176099 C NO176099 C NO 176099C
Authority
NO
Norway
Prior art keywords
pyridyl
oxo
preparation
therapeutically active
analogous process
Prior art date
Application number
NO903043A
Other languages
English (en)
Other versions
NO903043D0 (no
NO176099B (no
NO903043L (no
Inventor
Rolf Gericke
Manfred Baumgarth
Ingeborg Lues
Rolf Bergmann
Jacques De Peyer
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of NO903043D0 publication Critical patent/NO903043D0/no
Publication of NO903043L publication Critical patent/NO903043L/no
Publication of NO176099B publication Critical patent/NO176099B/no
Publication of NO176099C publication Critical patent/NO176099C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
NO903043A 1989-07-07 1990-07-06 Analogifremgangsmåte for fremstilling av terapeutisk aktive 4-(2-okso-3-pyridyl)-kromanderivater NO176099C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3922392A DE3922392A1 (de) 1989-07-07 1989-07-07 Chromanderivate

Publications (4)

Publication Number Publication Date
NO903043D0 NO903043D0 (no) 1990-07-06
NO903043L NO903043L (no) 1991-01-08
NO176099B NO176099B (no) 1994-10-24
NO176099C true NO176099C (no) 1995-02-01

Family

ID=6384507

Family Applications (1)

Application Number Title Priority Date Filing Date
NO903043A NO176099C (no) 1989-07-07 1990-07-06 Analogifremgangsmåte for fremstilling av terapeutisk aktive 4-(2-okso-3-pyridyl)-kromanderivater

Country Status (19)

Country Link
US (1) US5112839A (no)
EP (1) EP0406656B1 (no)
JP (1) JPH0344389A (no)
KR (1) KR910002842A (no)
AR (1) AR245940A1 (no)
AT (1) ATE116985T1 (no)
AU (1) AU622338B2 (no)
CA (1) CA2020553A1 (no)
DE (2) DE3922392A1 (no)
DK (1) DK0406656T3 (no)
ES (1) ES2066913T3 (no)
FI (1) FI95131C (no)
HU (1) HUT58726A (no)
IE (1) IE902477A1 (no)
IL (1) IL94987A (no)
NO (1) NO176099C (no)
NZ (1) NZ234395A (no)
PT (1) PT94629B (no)
ZA (1) ZA905325B (no)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5387587A (en) * 1986-12-23 1995-02-07 Merck Patent Gesellschaft Mit Beschrankter Haftung Chroman derivatives
US5284838A (en) * 1987-06-23 1994-02-08 Elf Sanofi Use of 2,2-dimethylchroman-3-ol derivatives in the treatment of asthma
KR950009863B1 (ko) * 1991-05-22 1995-08-29 재단법인한국화학연구소 벤조피란 유도체와 그의 제조방법
FR2698873B1 (fr) * 1992-12-07 1995-02-24 Lipha Benzocycloheptènes, benzoxépines et benzothiépines activateurs des canaux potassiques, procédé de préparation, composition pharmaceutique les contenant.
US5719155A (en) * 1993-11-10 1998-02-17 Japan Tobacco Inc. Chroman derivative and pharmaceutical use thereof
US5470861A (en) * 1994-08-04 1995-11-28 Hoffmann-La Roche Inc. Method of promoting hair growth
JP5082033B2 (ja) 2001-12-21 2012-11-28 エグゼリクシス パテント カンパニー エルエルシー Lxrのモジュレーター
US7482366B2 (en) 2001-12-21 2009-01-27 X-Ceptor Therapeutics, Inc. Modulators of LXR
AU2006284675A1 (en) 2005-09-01 2007-03-08 Janssen Pharmaceutica N.V. Novel benzopyran derivatives as potassium channel openers
EP1940516A2 (en) 2005-09-01 2008-07-09 Janssen Pharmaceutica, N.V. Benzopyran and pyranopyridine derivatives as potassium channel openers
KR100559450B1 (ko) * 2005-12-31 2006-03-10 이삼준 안전모 및 모자용 착탈그늘막
BR112023015584A2 (pt) 2021-02-02 2023-10-24 Liminal Biosciences Ltd Antagonistas de gpr84 e usos dos mesmos

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE23718T1 (de) 1981-09-25 1986-12-15 Beecham Group Plc Benzopyran-verbindungen mit pharmazeutischer wirkung.
GB8308062D0 (en) 1983-03-24 1983-05-05 Beecham Group Plc Active compounds
GB8419515D0 (en) 1984-07-31 1984-09-05 Beecham Group Plc Treatment
GB8419516D0 (en) 1984-07-31 1984-09-05 Beecham Group Plc Treatment
EP0218373B1 (en) * 1985-09-11 1990-03-07 Beecham Group Plc Chroman derivatives and analogues having antihypertensive activity
AU7875487A (en) 1986-08-08 1988-02-24 Upjohn Company, The Methods, compositions and solutions for treating alopecia
DE3726261A1 (de) * 1986-12-23 1988-07-07 Merck Patent Gmbh Chromanderivate
US4971982A (en) * 1987-07-06 1990-11-20 Hoffmann-La Roche Inc. Benzopyran derivatives
DE3924417A1 (de) * 1989-07-24 1991-01-31 Merck Patent Gmbh Chromanderivate

Also Published As

Publication number Publication date
FI95131B (fi) 1995-09-15
ATE116985T1 (de) 1995-01-15
EP0406656A1 (de) 1991-01-09
DE59008224D1 (de) 1995-02-23
AU622338B2 (en) 1992-04-02
HU904114D0 (en) 1990-12-28
EP0406656B1 (de) 1995-01-11
US5112839A (en) 1992-05-12
IL94987A (en) 1996-01-19
ES2066913T3 (es) 1995-03-16
NO903043D0 (no) 1990-07-06
FI95131C (fi) 1995-12-27
ZA905325B (en) 1991-04-24
IL94987A0 (en) 1991-06-10
JPH0344389A (ja) 1991-02-26
HUT58726A (en) 1992-03-30
IE902477A1 (en) 1991-02-13
DK0406656T3 (da) 1995-03-27
NO176099B (no) 1994-10-24
AR245940A1 (es) 1994-03-30
CA2020553A1 (en) 1991-01-08
PT94629A (pt) 1991-03-20
NZ234395A (en) 1991-08-27
NO903043L (no) 1991-01-08
AU5872590A (en) 1991-01-10
KR910002842A (ko) 1991-02-26
FI903431A0 (fi) 1990-07-06
DE3922392A1 (de) 1991-01-17
PT94629B (pt) 1997-06-30

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