NO151824C - INTERMEDIATES FOR THE MANUFACTURE OF GUANIDINE DERIVATIVES - Google Patents
INTERMEDIATES FOR THE MANUFACTURE OF GUANIDINE DERIVATIVESInfo
- Publication number
- NO151824C NO151824C NO833255A NO833255A NO151824C NO 151824 C NO151824 C NO 151824C NO 833255 A NO833255 A NO 833255A NO 833255 A NO833255 A NO 833255A NO 151824 C NO151824 C NO 151824C
- Authority
- NO
- Norway
- Prior art keywords
- intermediates
- manufacture
- guanidine derivatives
- guanidine
- derivatives
- Prior art date
Links
- ZRALSGWEFCBTJO-UHFFFAOYSA-N Guanidine Chemical class NC(N)=N ZRALSGWEFCBTJO-UHFFFAOYSA-N 0.000 title 1
- 229940083094 guanine derivative acting on arteriolar smooth muscle Drugs 0.000 title 1
- 239000000543 intermediate Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C323/39—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
- C07C323/43—Y being a hetero atom
- C07C323/44—X or Y being nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US80300977A | 1977-06-03 | 1977-06-03 | |
| US82679677A | 1977-08-22 | 1977-08-22 | |
| US05/848,959 US4112234A (en) | 1977-08-22 | 1977-11-07 | Imidazolylmethylthioethyl alkynyl guanidines |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO833255L NO833255L (en) | 1978-12-05 |
| NO151824B NO151824B (en) | 1985-03-04 |
| NO151824C true NO151824C (en) | 1985-06-12 |
Family
ID=27419995
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO781928A NO152214C (en) | 1977-06-03 | 1978-06-02 | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE N-CYANO-N`- (2 - ((4-METHYL-5-IMIDAZOLYL) -METHYLTIO) ETHYL-N "-ALKNYLGUANIDINES |
| NO791637A NO791637L (en) | 1977-06-03 | 1979-05-16 | INTERMEDIATE PRODUCTS FOR THE MANUFACTURE OF GUANIDINE DERIVATIVES |
| NO833255A NO151824C (en) | 1977-06-03 | 1983-09-12 | INTERMEDIATES FOR THE MANUFACTURE OF GUANIDINE DERIVATIVES |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO781928A NO152214C (en) | 1977-06-03 | 1978-06-02 | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE N-CYANO-N`- (2 - ((4-METHYL-5-IMIDAZOLYL) -METHYLTIO) ETHYL-N "-ALKNYLGUANIDINES |
| NO791637A NO791637L (en) | 1977-06-03 | 1979-05-16 | INTERMEDIATE PRODUCTS FOR THE MANUFACTURE OF GUANIDINE DERIVATIVES |
Country Status (26)
| Country | Link |
|---|---|
| JP (1) | JPS543067A (en) |
| AR (2) | AR222797A1 (en) |
| CA (1) | CA1110251A (en) |
| CH (2) | CH641167A5 (en) |
| CY (3) | CY1231A (en) |
| DD (1) | DD140038A5 (en) |
| DE (1) | DE2824066A1 (en) |
| DK (1) | DK243178A (en) |
| ES (3) | ES470474A1 (en) |
| FI (1) | FI69069C (en) |
| FR (2) | FR2401143A1 (en) |
| GB (3) | GB1598630A (en) |
| GR (1) | GR73860B (en) |
| HK (3) | HK38084A (en) |
| HU (1) | HU186766B (en) |
| IE (1) | IE47543B1 (en) |
| IL (1) | IL54819A (en) |
| KE (1) | KE3373A (en) |
| LU (1) | LU79725A1 (en) |
| MY (3) | MY8500451A (en) |
| NL (1) | NL7805935A (en) |
| NO (3) | NO152214C (en) |
| NZ (1) | NZ187376A (en) |
| SE (3) | SE443784B (en) |
| SG (1) | SG8584G (en) |
| YU (4) | YU129778A (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS568352A (en) * | 1979-07-03 | 1981-01-28 | Shionogi & Co Ltd | Aminoalkylvenzene derivative |
| US4339439A (en) * | 1981-01-19 | 1982-07-13 | Bristol-Myers Company | Pharmaceutical methods and compositions |
| JPS6018010U (en) * | 1983-07-18 | 1985-02-07 | 日産自動車株式会社 | Temperature adjustment mechanism of vehicle air conditioner |
| JPS60113211U (en) * | 1984-01-06 | 1985-07-31 | 松下電器産業株式会社 | Automotive air conditioner |
| ES2007948A6 (en) * | 1988-07-06 | 1989-07-01 | Vinas Lab | Propargylguanidine derivatives and process for the preparation thereof. |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1338169A (en) * | 1971-03-09 | 1973-11-21 | Smith Kline French Lab | Ureas thioureas and guanidines |
| US4024271A (en) * | 1971-03-09 | 1977-05-17 | Smith Kline & French Laboratories Limited | Pharmacologically active guanidine compounds |
| GB1397436A (en) * | 1972-09-05 | 1975-06-11 | Smith Kline French Lab | Heterocyclic n-cyanoguinidines |
| GB1531231A (en) * | 1974-09-02 | 1978-11-08 | Smith Kline French Lab | Process for the production of cyanoguanidine derivatives |
| GB1531221A (en) * | 1974-09-02 | 1978-11-08 | Smith Kline French Lab | Process for preparing guanidine derivatives |
| GB1533380A (en) * | 1974-09-02 | 1978-11-22 | Smith Kline French Lab | Process for the preparation of heterocyclic substituted thioureas and h-cyanoguanidines |
-
1978
- 1978-05-25 NZ NZ187376A patent/NZ187376A/en unknown
- 1978-05-25 CA CA304,045A patent/CA1110251A/en not_active Expired
- 1978-05-26 CY CY1231A patent/CY1231A/en unknown
- 1978-05-26 GB GB18923/80A patent/GB1598630A/en not_active Expired
- 1978-05-26 GB GB23611/78A patent/GB1598628A/en not_active Expired
- 1978-05-26 CY CY1229A patent/CY1229A/en unknown
- 1978-05-26 CY CY1230A patent/CY1230A/en unknown
- 1978-05-26 GB GB27637/79A patent/GB1598629A/en not_active Expired
- 1978-05-29 GR GR56374A patent/GR73860B/el unknown
- 1978-05-29 LU LU79725A patent/LU79725A1/en unknown
- 1978-05-31 IL IL54819A patent/IL54819A/en unknown
- 1978-05-31 YU YU01297/78A patent/YU129778A/en unknown
- 1978-05-31 AR AR272401A patent/AR222797A1/en active
- 1978-05-31 NL NL7805935A patent/NL7805935A/en not_active Application Discontinuation
- 1978-05-31 FI FI781737A patent/FI69069C/en not_active IP Right Cessation
- 1978-05-31 DK DK243178A patent/DK243178A/en not_active Application Discontinuation
- 1978-06-01 DE DE19782824066 patent/DE2824066A1/en not_active Withdrawn
- 1978-06-02 IE IE1112/78A patent/IE47543B1/en unknown
- 1978-06-02 SE SE7806525A patent/SE443784B/en unknown
- 1978-06-02 HU HU811135A patent/HU186766B/en unknown
- 1978-06-02 NO NO781928A patent/NO152214C/en unknown
- 1978-06-02 FR FR7816601A patent/FR2401143A1/en active Granted
- 1978-06-02 JP JP6590078A patent/JPS543067A/en active Granted
- 1978-06-02 ES ES470474A patent/ES470474A1/en not_active Expired
- 1978-06-02 CH CH609278A patent/CH641167A5/en not_active IP Right Cessation
- 1978-06-05 DD DD78205794A patent/DD140038A5/en unknown
-
1979
- 1979-03-01 ES ES478203A patent/ES478203A1/en not_active Expired
- 1979-03-01 ES ES478202A patent/ES478202A1/en not_active Expired
- 1979-03-05 YU YU530/79A patent/YU41620B/en unknown
- 1979-05-16 NO NO791637A patent/NO791637L/en unknown
- 1979-10-26 AR AR278645A patent/AR222503A1/en active
- 1979-11-23 FR FR7928943A patent/FR2436138A1/en active Granted
-
1982
- 1982-09-27 YU YU2154/82A patent/YU40624B/en unknown
- 1982-09-27 YU YU2155/82A patent/YU40625B/en unknown
-
1983
- 1983-09-12 NO NO833255A patent/NO151824C/en unknown
- 1983-10-07 CH CH549283A patent/CH644591A5/en not_active IP Right Cessation
-
1984
- 1984-01-30 SG SG85/84A patent/SG8584G/en unknown
- 1984-02-10 KE KE3373A patent/KE3373A/en unknown
- 1984-03-16 SE SE8401492A patent/SE8401492D0/en not_active Application Discontinuation
- 1984-03-16 SE SE8401491A patent/SE8401491L/en not_active Application Discontinuation
- 1984-05-03 HK HK380/84A patent/HK38084A/en unknown
- 1984-05-03 HK HK382/84A patent/HK38284A/en unknown
- 1984-05-03 HK HK381/84A patent/HK38184A/en unknown
-
1985
- 1985-12-30 MY MY451/85A patent/MY8500451A/en unknown
- 1985-12-30 MY MY452/85A patent/MY8500452A/en unknown
- 1985-12-30 MY MY453/85A patent/MY8500453A/en unknown
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