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NO151201C - PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ANTIGENDATIVE DERIVATIVES - Google Patents

PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ANTIGENDATIVE DERIVATIVES

Info

Publication number
NO151201C
NO151201C NO79790626A NO790626A NO151201C NO 151201 C NO151201 C NO 151201C NO 79790626 A NO79790626 A NO 79790626A NO 790626 A NO790626 A NO 790626A NO 151201 C NO151201 C NO 151201C
Authority
NO
Norway
Prior art keywords
antigendative
derivatives
procedure
preparation
therapeutically effective
Prior art date
Application number
NO79790626A
Other languages
Norwegian (no)
Other versions
NO790626L (en
NO151201B (en
Inventor
Gerhard Baschang
Felix M Dietrich
Roland Gisler
Jaroslav Stanek
Albert Hartmann
Lajos Tarcsay
Original Assignee
Ciba Geigy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27173419&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO151201(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ciba Geigy filed Critical Ciba Geigy
Publication of NO790626L publication Critical patent/NO790626L/en
Publication of NO151201B publication Critical patent/NO151201B/en
Publication of NO151201C publication Critical patent/NO151201C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H9/00Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical
    • C07H9/02Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical the hetero ring containing only oxygen as ring hetero atoms
    • C07H9/04Cyclic acetals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K39/385Haptens or antigens, bound to carriers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H23/00Compounds containing boron, silicon or a metal, e.g. chelates or vitamin B12
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/001Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence having less than 12 amino acids and not being part of a ring structure
    • C07K9/005Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence having less than 12 amino acids and not being part of a ring structure containing within the molecule the substructure with m, n > 0 and m+n > 0, A, B, D, E being heteroatoms; X being a bond or a chain, e.g. muramylpeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/555Medicinal preparations containing antigens or antibodies characterised by a specific combination antigen/adjuvant
    • A61K2039/55511Organic adjuvants
    • A61K2039/55583Polysaccharides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/60Medicinal preparations containing antigens or antibodies characteristics by the carrier linked to the antigen
    • A61K2039/6031Proteins
    • A61K2039/6062Muramyl peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Immunology (AREA)
  • Public Health (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Peptides Or Proteins (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO79790626A 1978-02-24 1979-02-23 PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ANTIGENDATIVE DERIVATIVES NO151201C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH203578 1978-02-24
CH377778 1978-04-07
CH539478 1978-05-18

Publications (3)

Publication Number Publication Date
NO790626L NO790626L (en) 1979-08-27
NO151201B NO151201B (en) 1984-11-19
NO151201C true NO151201C (en) 1985-02-27

Family

ID=27173419

Family Applications (2)

Application Number Title Priority Date Filing Date
NO79790626A NO151201C (en) 1978-02-24 1979-02-23 PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ANTIGENDATIVE DERIVATIVES
NO79793993A NO151088C (en) 1978-02-24 1979-12-07 ANALOGY PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICALLY EFFECTIVE SILYL-GLUCOSAMINE DERIVATIVES

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO79793993A NO151088C (en) 1978-02-24 1979-12-07 ANALOGY PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICALLY EFFECTIVE SILYL-GLUCOSAMINE DERIVATIVES

Country Status (20)

Country Link
EP (1) EP0003833B2 (en)
JP (1) JPS54141718A (en)
AR (1) AR223833A1 (en)
AT (1) AT364718B (en)
AU (1) AU527549B2 (en)
CA (1) CA1138436A (en)
DD (1) DD141616A5 (en)
DK (1) DK161026C (en)
ES (2) ES477977A1 (en)
FI (1) FI66878C (en)
GB (1) GB2015534A (en)
GR (1) GR77615B (en)
HU (1) HU182011B (en)
IL (1) IL56724A (en)
NO (2) NO151201C (en)
NZ (1) NZ189756A (en)
PL (1) PL123315B1 (en)
PT (1) PT69281A (en)
SU (1) SU1055312A3 (en)
ZA (1) ZA79893B (en)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54130516A (en) * 1978-03-31 1979-10-09 Yuuichi Yamamura Acyllnnacetylmuramylpeptide derivativeeantigen combination
FR2428051A1 (en) * 1978-06-05 1980-01-04 Anvar NOVEL MURAMYL-PEPTIDE COMPOUNDS AND MEDICAMENTS CONTAINING THEM
FR2428050A1 (en) * 1978-06-05 1980-01-04 Anvar OLIGOMERS OF MURAMYL-PEPTIDE COMPOUNDS AND DRUGS CONTAINING THEM
EP0013856B1 (en) 1978-12-22 1983-03-09 ANVAR Agence Nationale de Valorisation de la Recherche New compounds associating peptidyl or aminoacyl residues to lipophilic groups and pharmaceutical compositions containing said new compounds
FR2446292A1 (en) * 1979-01-12 1980-08-08 Anvar MURAMYL-PEPTIDES FIXED ON PEPTIDE POLYMERS AND MEDICAMENTS CONTAINING THEM
FR2449697A1 (en) 1979-02-20 1980-09-19 Anvar NOVEL MURAMYL-PEPTIDES SUBSTITUTED ON PEPTIDE NITROGEN AND MEDICAMENTS CONTAINING THEM
JPS5618996A (en) * 1979-06-21 1981-02-23 Dai Ichi Seiyaku Co Ltd Muramyldipeptide derivative
DK156252C (en) * 1979-07-31 1989-12-18 Fujisawa Pharmaceutical Co METHOD OF ANALOGUE FOR THE PREPARATION OF DI, TRIAL OR TETRAPEPTIDE DERIVATIVES OR SALTS THEREOF
US4406889A (en) * 1980-02-15 1983-09-27 Ciba-Geigy Corporation Derivatives of aldohexoses, intermediates, processes for their manufacture, preparations containing such compounds, and their use
EP0038153A3 (en) * 1980-04-15 1982-12-22 Beecham Group Plc Modified allergens
US4368190A (en) * 1980-04-17 1983-01-11 Merck & Co., Inc. Immunologically active dipeptidyl 4-O-,6-O-acyl-2-amino-2-deoxy-D-glucose derivatives and methods for their preparation
US4497729A (en) * 1980-12-01 1985-02-05 Fujisawa Pharmaceutical Co., Ltd. Peptide, process for preparation thereof and use thereof
FR2522967B1 (en) * 1982-03-15 1986-03-07 Anvar CONJUGATES OF HAPTENES AND MURAMYL-PEPTIDES, WITH IMMUNOGENIC ACTIVITY AND COMPOSITIONS CONTAINING THEM
US4587046A (en) * 1982-05-18 1986-05-06 The Regents Of The University Of California Drug-carrier conjugates
FR2558165B1 (en) * 1984-01-17 1986-07-04 Anvar NOVEL CONJUGATES OF OLIGO-MURAMYLPEPTIDES AND BIOLOGICAL COMPOSITIONS CONTAINING THEM FOR THE ACTIVATION OF MACROPHAGES
FR2569984B1 (en) * 1984-09-12 1987-08-14 Anvar SYNTHETIC MOLECULE CONTAINING A PLURALITY OF SEPARATE EPITOPES, PROCESS FOR OBTAINING SAME AND APPLICATION TO THE PRODUCTION OF POLYVACCINES
CN116077439A (en) 2016-04-29 2023-05-09 西奈山伊坎医学院 Targeting the innate immune system to induce long-term tolerance and address macrophage accumulation in atherosclerosis
EP3636656A4 (en) 2017-06-09 2021-04-14 Chugai Seiyaku Kabushiki Kaisha PROCESS FOR SYNTHESIS OF A PEPTIDE CONTAINING AN N-SUBSTITUTED AMINO ACID
EP3889164A4 (en) * 2018-11-30 2022-11-02 Chugai Seiyaku Kabushiki Kaisha METHOD FOR DEPROTECTION AND METHOD FOR RESIN REMOVAL IN A SOLID PHASE REACTION OF A PEPTIDE COMPOUND OR AN AMIDE COMPOUND, AND METHOD FOR PRODUCTION OF A PEPTIDE COMPOUND
IL306006A (en) 2021-03-19 2023-11-01 Trained Therapeutix Discovery Inc Compounds for regulating trained immunity, and their methods of use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH564031A5 (en) * 1968-03-29 1975-07-15 Anvar
US4186194A (en) * 1973-10-23 1980-01-29 Agence Nationale De Valorisation De La Recherche (Anvar) Water soluble agents effective as immunological adjuvants for stimulating, in the host the immune response to various antigens and compositions, notably vaccines containing said water soluble agents
CH613709A5 (en) * 1975-12-10 1979-10-15 Ciba Geigy Ag Process for the preparation of glucosamine derivatives
FR2343482A1 (en) * 1976-03-10 1977-10-07 Anvar LA 2- (2-ACETAMIDO-2-DEOXY-3-O-D-GLUCOPYRANOSYL) -D-PROPIONYL-L-SERYL-D-ISOGLUTAMINE AND MEDICINES CONTAINING IT
JPS52139018A (en) * 1976-03-10 1977-11-19 Anvar Immuno adjuvant and antiinfection adjuvant composed of mainly nnacetyll muramiccllalanyllddglutamic ester or nnacetyllmuramiccllalanylldd isoglutamic ester

Also Published As

Publication number Publication date
FI790584A7 (en) 1979-08-25
EP0003833A2 (en) 1979-09-05
NO151088B (en) 1984-10-29
NO151088C (en) 1985-02-06
SU1055312A3 (en) 1983-11-15
JPS54141718A (en) 1979-11-05
FI66878B (en) 1984-08-31
ZA79893B (en) 1980-03-26
AR223833A1 (en) 1981-09-30
DK79779A (en) 1979-08-25
DK161026C (en) 1991-10-28
ATA142079A (en) 1981-04-15
PL123315B1 (en) 1982-10-30
ES483558A1 (en) 1980-04-16
JPH0130809B2 (en) 1989-06-22
GR77615B (en) 1984-09-25
ES477977A1 (en) 1980-01-16
HU182011B (en) 1983-12-28
NO790626L (en) 1979-08-27
PT69281A (en) 1979-03-01
AU4454679A (en) 1979-08-30
NO793993L (en) 1979-08-27
DK161026B (en) 1991-05-21
EP0003833B2 (en) 1990-12-19
DD141616A5 (en) 1980-05-14
IL56724A (en) 1982-12-31
GB2015534A (en) 1979-09-12
EP0003833B1 (en) 1983-07-20
AU527549B2 (en) 1983-03-10
NO151201B (en) 1984-11-19
PL213696A1 (en) 1980-07-14
NZ189756A (en) 1982-05-31
EP0003833A3 (en) 1980-02-06
FI66878C (en) 1984-12-10
IL56724A0 (en) 1979-05-31
CA1138436A (en) 1982-12-28
AT364718B (en) 1981-11-10

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