NL169877B - METHOD FOR THE PREPARATION OR MANUFACTURE OF PREPARATIONS WITH ANTI-INFLAMMATORIC, ANALGETIC AND ANTI-RHEUMATIC PROPERTIES CONTAINING AN CARBOZOLIC DERIVATIVE AS AN ACTIVE SUBSTANCE. - Google Patents
METHOD FOR THE PREPARATION OR MANUFACTURE OF PREPARATIONS WITH ANTI-INFLAMMATORIC, ANALGETIC AND ANTI-RHEUMATIC PROPERTIES CONTAINING AN CARBOZOLIC DERIVATIVE AS AN ACTIVE SUBSTANCE.Info
- Publication number
- NL169877B NL169877B NLAANVRAGE7310275,A NL7310275A NL169877B NL 169877 B NL169877 B NL 169877B NL 7310275 A NL7310275 A NL 7310275A NL 169877 B NL169877 B NL 169877B
- Authority
- NL
- Netherlands
- Prior art keywords
- carbozolic
- inflammatoric
- analgetic
- preparations
- derivative
- Prior art date
Links
- 238000002360 preparation method Methods 0.000 title 2
- 239000013543 active substance Substances 0.000 title 1
- 230000000202 analgesic effect Effects 0.000 title 1
- 230000003110 anti-inflammatory effect Effects 0.000 title 1
- 230000003356 anti-rheumatic effect Effects 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- C07D209/82—Carbazoles; Hydrogenated carbazoles
- C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- C07D209/82—Carbazoles; Hydrogenated carbazoles
- C07D209/86—Carbazoles; Hydrogenated carbazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the ring system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pain & Pain Management (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27414272A | 1972-07-24 | 1972-07-24 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NL7310275A NL7310275A (en) | 1974-01-28 |
| NL169877B true NL169877B (en) | 1982-04-01 |
| NL169877C NL169877C (en) | 1982-09-01 |
Family
ID=23046965
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NLAANVRAGE7310275,A NL169877C (en) | 1972-07-24 | 1973-07-24 | METHOD FOR THE PREPARATION OR MANUFACTURE OF PREPARATIONS WITH ANTI-INFLAMMATORIC, ANALGETIC AND ANTI-RHEUMATIC PROPERTIES CONTAINING AN CARBOZOLIC DERIVATIVE AS AN ACTIVE SUBSTANCE. |
Country Status (26)
| Country | Link |
|---|---|
| JP (1) | JPS5740144B2 (en) |
| KR (1) | KR780000289B1 (en) |
| AR (1) | AR205331A1 (en) |
| AT (1) | AT325607B (en) |
| AU (1) | AU475534B2 (en) |
| BE (1) | BE802596A (en) |
| CA (1) | CA1026348A (en) |
| CH (1) | CH587819A5 (en) |
| DD (1) | DD107681A5 (en) |
| DE (1) | DE2337340C2 (en) |
| DK (1) | DK138537B (en) |
| FI (1) | FI59244C (en) |
| FR (1) | FR2193611B1 (en) |
| GB (1) | GB1385620A (en) |
| HK (1) | HK49878A (en) |
| HU (1) | HU167611B (en) |
| IE (1) | IE37942B1 (en) |
| IL (1) | IL42799A (en) |
| KE (1) | KE2847A (en) |
| LU (1) | LU68071A1 (en) |
| MY (1) | MY7800315A (en) |
| NL (1) | NL169877C (en) |
| NO (1) | NO142865C (en) |
| SE (2) | SE402283B (en) |
| SU (1) | SU509220A3 (en) |
| ZA (1) | ZA734047B (en) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4146542A (en) * | 1978-06-12 | 1979-03-27 | Hoffmann-La Roche Inc. | Dihydrocarbazole acetic acid and esters thereof |
| US4150031A (en) * | 1978-06-26 | 1979-04-17 | Hoffmann-La Roche Inc. | Hydroxy methyl carbazole acetic acid and esters |
| US4158007A (en) * | 1978-08-21 | 1979-06-12 | Hoffmann-La Roche Inc. | Carbazole methyl malonates |
| US4501908A (en) * | 1981-03-12 | 1985-02-26 | Hoffmann-La Roche Inc. | 2,3-Isopropylidene ribonic acid, 1,4-lactones |
| JPS6040256U (en) * | 1983-08-25 | 1985-03-20 | 伊東 璋 | Container cleaning machine |
| EP0234708B1 (en) * | 1986-01-23 | 1991-02-27 | Merck Frosst Canada Inc. | Tetrahydrocarbazole 1-alkanoic acids |
| DE3786030T2 (en) | 1986-03-27 | 1993-12-02 | Merck Frosst Canada Inc | Tetrahydrocarbazole esters. |
| EP0307077A1 (en) * | 1987-07-21 | 1989-03-15 | Merck Frosst Canada Inc. | Tetrahydrocarbazoles for the improvement of cyclosporin therapy |
| CA1326030C (en) * | 1987-07-21 | 1994-01-11 | John W. Gillard | Cyclohept[b]indolealkanoic acids |
| PT95692A (en) * | 1989-10-27 | 1991-09-13 | American Home Prod | PROCESS FOR THE PREPARATION OF INDOLE-, INDENO-, PYRANOINDOLE- AND TETRA-HYDROCARBAZOLE-ALCANOIC ACID DERIVATIVES, OR WHICH ARE USEFUL AS PLA2 INHIBITORS AND LIPOXIGENASE |
| US6013808A (en) * | 1998-06-16 | 2000-01-11 | Pfizer Inc. | Method of purifying carbazole ester precursors of 6-chloro-α-methyl-carbazole-2-acetic acid |
| JP2004010601A (en) * | 2002-06-11 | 2004-01-15 | Nippon Steel Chem Co Ltd | Process for producing indole derivative and useful intermediate therefor |
| AU2004206796A1 (en) | 2003-01-14 | 2004-08-05 | Merck & Co., Inc. | Geminally di-substituted NSAID derivatives as Abeta 42 lowering agents |
| KR101121819B1 (en) * | 2003-05-06 | 2012-03-21 | 에어프로덕츠앤드케미칼스,인코포레이티드 | Hydrogen storage by reversible hydrogenation of pi-conjugated substrates |
| CA2535497A1 (en) * | 2003-08-15 | 2005-02-24 | Universite Laval | Monomers, oligomers and polymers of 2-functionalized and 2,7-difunctionalized carbazoles |
| US7601856B2 (en) | 2006-07-27 | 2009-10-13 | Wyeth | Benzofurans as potassium ion channel modulators |
| US7662831B2 (en) | 2006-07-27 | 2010-02-16 | Wyeth Llc | Tetracyclic indoles as potassium channel modulators |
| KR101986272B1 (en) * | 2011-11-15 | 2019-06-05 | 이섬 리서치 디벨러프먼트 컴파니 오브 더 히브루 유니버시티 오브 예루살렘 엘티디. | Tricyclic compounds, compositions comprising them and uses thereof |
| JP5940036B2 (en) * | 2013-10-08 | 2016-06-29 | テックフィールズ バイオケム カンパニー リミテッド | Positively charged water-soluble prodrugs of aryl- and heteroarylpropionic acids with very fast skin permeability |
| CN114787130A (en) * | 2020-03-25 | 2022-07-22 | 捷恩智株式会社 | Compound, liquid crystal composition and liquid crystal display element |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DD70880A (en) * | ||||
| US3580926A (en) * | 1969-11-10 | 1971-05-25 | Parke Davis & Co | Carbazole-4-alkanoic acids and tetrahydrocarbazole-4-alkanoic acids |
| ZA715217B (en) * | 1970-08-20 | 1972-04-26 | Org Nv | Anti-inflammatory preparations |
-
1973
- 1973-01-01 AR AR249230A patent/AR205331A1/en active
- 1973-06-14 ZA ZA734047A patent/ZA734047B/en unknown
- 1973-06-15 CH CH871673A patent/CH587819A5/xx not_active IP Right Cessation
- 1973-07-20 IL IL42799A patent/IL42799A/en unknown
- 1973-07-20 HU HUHO1597A patent/HU167611B/hu unknown
- 1973-07-20 KR KR7301174A patent/KR780000289B1/en not_active Expired
- 1973-07-20 BE BE133691A patent/BE802596A/en not_active IP Right Cessation
- 1973-07-23 AT AT649773A patent/AT325607B/en not_active IP Right Cessation
- 1973-07-23 CA CA177,061A patent/CA1026348A/en not_active Expired
- 1973-07-23 DE DE2337340A patent/DE2337340C2/en not_active Expired
- 1973-07-23 DK DK405973AA patent/DK138537B/en not_active IP Right Cessation
- 1973-07-23 IE IE1252/73A patent/IE37942B1/en unknown
- 1973-07-23 GB GB3496873A patent/GB1385620A/en not_active Expired
- 1973-07-23 NO NO2975/73A patent/NO142865C/en unknown
- 1973-07-23 LU LU68071A patent/LU68071A1/xx unknown
- 1973-07-23 SE SE7310244A patent/SE402283B/en unknown
- 1973-07-23 JP JP48081008A patent/JPS5740144B2/ja not_active Expired
- 1973-07-23 DD DD172456A patent/DD107681A5/xx unknown
- 1973-07-23 AU AU58390/73A patent/AU475534B2/en not_active Expired
- 1973-07-23 FI FI2311/73A patent/FI59244C/en active
- 1973-07-24 FR FR7327020A patent/FR2193611B1/fr not_active Expired
- 1973-07-24 SU SU1950151A patent/SU509220A3/en active
- 1973-07-24 NL NLAANVRAGE7310275,A patent/NL169877C/en not_active IP Right Cessation
-
1976
- 1976-05-21 SE SE7605813A patent/SE7605813L/en unknown
-
1978
- 1978-06-13 KE KE2847A patent/KE2847A/en unknown
- 1978-08-31 HK HK498/78A patent/HK49878A/en unknown
- 1978-12-30 MY MY315/78A patent/MY7800315A/en unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| SNR | Assignments of patents or rights arising from examined patent applications |
Owner name: F. HOFFMANN-LA ROCHE AG |
|
| V4 | Discontinued because of reaching the maximum lifetime of a patent |