NI201700066A - Antagonistas de a2a de dosis baja para tratamiento de tdah y la enfermedad de parkinson - Google Patents
Antagonistas de a2a de dosis baja para tratamiento de tdah y la enfermedad de parkinsonInfo
- Publication number
- NI201700066A NI201700066A NI201700066A NI201700066A NI201700066A NI 201700066 A NI201700066 A NI 201700066A NI 201700066 A NI201700066 A NI 201700066A NI 201700066 A NI201700066 A NI 201700066A NI 201700066 A NI201700066 A NI 201700066A
- Authority
- NI
- Nicaragua
- Prior art keywords
- parkinson
- treatment
- adhd
- antagonists
- disease
- Prior art date
Links
- 208000006096 Attention Deficit Disorder with Hyperactivity Diseases 0.000 title abstract 2
- 208000036864 Attention deficit/hyperactivity disease Diseases 0.000 title abstract 2
- 208000018737 Parkinson disease Diseases 0.000 title abstract 2
- 239000005557 antagonist Substances 0.000 title abstract 2
- 208000015802 attention deficit-hyperactivity disease Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4436—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Psychology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
Abstract
La presente invención se refiere a dosis específicas de un antagonista de A2A para utilizarlo como un medicamento y, en particular, que sean útiles para el tratamiento de enfermedades de Parkinson y del trastorno por déficit de atención con hiperactividad.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA201400704 | 2014-12-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NI201700066A true NI201700066A (es) | 2018-01-04 |
Family
ID=58731664
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NI201700066A NI201700066A (es) | 2014-12-03 | 2017-06-01 | Antagonistas de a2a de dosis baja para tratamiento de tdah y la enfermedad de parkinson |
Country Status (25)
| Country | Link |
|---|---|
| US (2) | US20160158211A1 (es) |
| EP (1) | EP3226863A1 (es) |
| JP (1) | JP2017536400A (es) |
| KR (1) | KR20170090430A (es) |
| CN (1) | CN106999480A (es) |
| AU (1) | AU2015357197A1 (es) |
| BR (1) | BR112017011777A2 (es) |
| CA (1) | CA2966582A1 (es) |
| CL (1) | CL2017001407A1 (es) |
| CO (1) | CO2017004785A2 (es) |
| CR (1) | CR20170221A (es) |
| DO (1) | DOP2017000121A (es) |
| EA (1) | EA201790973A1 (es) |
| EC (1) | ECSP17030050A (es) |
| IL (1) | IL252355A0 (es) |
| MA (1) | MA41090A (es) |
| MX (1) | MX2017007027A (es) |
| NI (1) | NI201700066A (es) |
| PE (1) | PE20170926A1 (es) |
| PH (1) | PH12017500923A1 (es) |
| SG (1) | SG11201704370XA (es) |
| SV (1) | SV2017005441A (es) |
| TN (1) | TN2017000174A1 (es) |
| TW (1) | TW201632186A (es) |
| WO (1) | WO2016087429A1 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL279829B2 (en) | 2018-07-05 | 2025-05-01 | Incyte Holdings Corp | Fused pyrazine derivatives as A2A/A2B inhibitors |
| JOP20210164A1 (ar) | 2019-01-11 | 2023-01-30 | Omeros Corp | طرق وتركيبات علاج السرطان |
| TWI829857B (zh) | 2019-01-29 | 2024-01-21 | 美商英塞特公司 | 作為a2a / a2b抑制劑之吡唑并吡啶及三唑并吡啶 |
| CN114917350B (zh) * | 2022-06-21 | 2023-06-13 | 重庆医科大学附属第二医院 | Cftr增强剂在注意缺陷与多动障碍中的应用及产品 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2004309279B2 (en) * | 2003-12-26 | 2010-07-15 | Kyowa Kirin Co., Ltd. | Thiazole derivative |
| CN102105168A (zh) * | 2008-07-23 | 2011-06-22 | 协和发酵麒麟株式会社 | 偏头痛治疗剂 |
| TWI548411B (zh) * | 2009-04-28 | 2016-09-11 | Kyowa Hakko Kirin Co Ltd | Exercise disorder treatment |
| UA113383C2 (xx) * | 2009-09-02 | 2017-01-25 | Терапевтичний агент для лікування тривожних розладів | |
| UA110097C2 (uk) * | 2009-09-02 | 2015-11-25 | Терапевтичний агент для лікування розладів настрою |
-
2015
- 2015-11-30 MA MA041090A patent/MA41090A/fr unknown
- 2015-12-01 BR BR112017011777A patent/BR112017011777A2/pt not_active Application Discontinuation
- 2015-12-01 TW TW104140137A patent/TW201632186A/zh unknown
- 2015-12-01 EP EP15802121.2A patent/EP3226863A1/en not_active Withdrawn
- 2015-12-01 JP JP2017529636A patent/JP2017536400A/ja not_active Withdrawn
- 2015-12-01 WO PCT/EP2015/078181 patent/WO2016087429A1/en not_active Ceased
- 2015-12-01 CA CA2966582A patent/CA2966582A1/en not_active Withdrawn
- 2015-12-01 SG SG11201704370XA patent/SG11201704370XA/en unknown
- 2015-12-01 CR CR20170221A patent/CR20170221A/es unknown
- 2015-12-01 AU AU2015357197A patent/AU2015357197A1/en not_active Withdrawn
- 2015-12-01 PE PE2017000864A patent/PE20170926A1/es not_active Application Discontinuation
- 2015-12-01 EA EA201790973A patent/EA201790973A1/ru unknown
- 2015-12-01 US US14/955,148 patent/US20160158211A1/en not_active Abandoned
- 2015-12-01 TN TN2017000174A patent/TN2017000174A1/en unknown
- 2015-12-01 KR KR1020177015211A patent/KR20170090430A/ko not_active Withdrawn
- 2015-12-01 MX MX2017007027A patent/MX2017007027A/es unknown
- 2015-12-01 CN CN201580064814.4A patent/CN106999480A/zh not_active Withdrawn
-
2017
- 2017-05-12 CO CONC2017/0004785A patent/CO2017004785A2/es unknown
- 2017-05-12 SV SV2017005441A patent/SV2017005441A/es unknown
- 2017-05-16 DO DO2017000121A patent/DOP2017000121A/es unknown
- 2017-05-16 EC ECIEPI201730050A patent/ECSP17030050A/es unknown
- 2017-05-17 IL IL252355A patent/IL252355A0/en unknown
- 2017-05-18 PH PH12017500923A patent/PH12017500923A1/en unknown
- 2017-06-01 NI NI201700066A patent/NI201700066A/es unknown
- 2017-06-02 CL CL2017001407A patent/CL2017001407A1/es unknown
- 2017-11-10 US US15/809,378 patent/US20180125835A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2966582A1 (en) | 2016-06-09 |
| DOP2017000121A (es) | 2017-07-15 |
| MA41090A (fr) | 2017-10-10 |
| PE20170926A1 (es) | 2017-07-13 |
| SG11201704370XA (en) | 2017-06-29 |
| MX2017007027A (es) | 2017-08-24 |
| US20180125835A1 (en) | 2018-05-10 |
| KR20170090430A (ko) | 2017-08-07 |
| CN106999480A (zh) | 2017-08-01 |
| CO2017004785A2 (es) | 2017-08-31 |
| TW201632186A (zh) | 2016-09-16 |
| EA201790973A1 (ru) | 2017-10-31 |
| CL2017001407A1 (es) | 2018-01-05 |
| IL252355A0 (en) | 2017-07-31 |
| AU2015357197A1 (en) | 2017-05-25 |
| TN2017000174A1 (en) | 2018-10-19 |
| CR20170221A (es) | 2017-10-05 |
| WO2016087429A1 (en) | 2016-06-09 |
| SV2017005441A (es) | 2017-08-25 |
| JP2017536400A (ja) | 2017-12-07 |
| US20160158211A1 (en) | 2016-06-09 |
| EP3226863A1 (en) | 2017-10-11 |
| BR112017011777A2 (pt) | 2018-02-20 |
| PH12017500923A1 (en) | 2017-11-20 |
| ECSP17030050A (es) | 2017-08-31 |
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