NI201400004A - 4 - IMIDAZOPYRIDAZIN - 1 - IL - BENZAMIDES AND 4 - IMIDAZOTRIAZIN - 1 - IL - BENZAMIDES AS BTK INHIBITORS - Google Patents
4 - IMIDAZOPYRIDAZIN - 1 - IL - BENZAMIDES AND 4 - IMIDAZOTRIAZIN - 1 - IL - BENZAMIDES AS BTK INHIBITORSInfo
- Publication number
- NI201400004A NI201400004A NI201400004A NI201400004A NI201400004A NI 201400004 A NI201400004 A NI 201400004A NI 201400004 A NI201400004 A NI 201400004A NI 201400004 A NI201400004 A NI 201400004A NI 201400004 A NI201400004 A NI 201400004A
- Authority
- NI
- Nicaragua
- Prior art keywords
- benzamides
- imidazotriazin
- imidazopyridazin
- btk inhibitors
- formula
- Prior art date
Links
- 229940054066 benzamide antipsychotics Drugs 0.000 title 2
- 229940124291 BTK inhibitor Drugs 0.000 title 1
- 102000001714 Agammaglobulinaemia Tyrosine Kinase Human genes 0.000 abstract 2
- 108010029445 Agammaglobulinaemia Tyrosine Kinase Proteins 0.000 abstract 2
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical group C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere a compuestos de anillos de piridina fusionados de 5-6 miembros según la fórmula I o una sal farmacéuticamente aceptable de los mismos o a composiciones farmacéuticas que comprenden estos compuestos y a su uso en terapia. En particular, la presente invención se refiere al uso de compuestos de anillos de piridina fusionados de 5-6 miembros según la fórmula I en el tratamiento de trastornos mediados por tirosina cinasa de Bruton (BK).The present invention relates to 5-6 membered fused pyridine ring compounds according to formula I or a pharmaceutically acceptable salt thereof or to pharmaceutical compositions comprising these compounds and their use in therapy. In particular, the present invention relates to the use of 5-6 membered fused pyridine ring compounds according to formula I in the treatment of disorders mediated by Bruton's tyrosine kinase (BK).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161509397P | 2011-07-19 | 2011-07-19 | |
| EP11174578 | 2011-07-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NI201400004A true NI201400004A (en) | 2014-10-10 |
Family
ID=67956153
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NI201400004A NI201400004A (en) | 2011-07-19 | 2014-01-17 | 4 - IMIDAZOPYRIDAZIN - 1 - IL - BENZAMIDES AND 4 - IMIDAZOTRIAZIN - 1 - IL - BENZAMIDES AS BTK INHIBITORS |
Country Status (8)
| Country | Link |
|---|---|
| CY (1) | CY1121174T1 (en) |
| LT (2) | LT3689878T (en) |
| ME (1) | ME03310B (en) |
| NI (1) | NI201400004A (en) |
| NL (1) | NL301097I2 (en) |
| NO (1) | NO2021016I1 (en) |
| PT (1) | PT2734522T (en) |
| TR (1) | TR201901013T4 (en) |
-
2012
- 2012-07-11 LT LTEP19215783.2T patent/LT3689878T/en unknown
- 2012-07-11 ME MEP-2019-4A patent/ME03310B/en unknown
- 2012-07-11 PT PT12733505T patent/PT2734522T/en unknown
- 2012-07-11 TR TR2019/01013T patent/TR201901013T4/en unknown
-
2014
- 2014-01-17 NI NI201400004A patent/NI201400004A/en unknown
-
2019
- 2019-01-22 CY CY20191100084T patent/CY1121174T1/en unknown
-
2021
- 2021-03-22 NL NL301097C patent/NL301097I2/en unknown
- 2021-03-24 LT LTPA2021004C patent/LTC2734522I2/en unknown
- 2021-04-09 NO NO2021016C patent/NO2021016I1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| LTPA2021004I1 (en) | 2021-04-12 |
| TR201901013T4 (en) | 2019-02-21 |
| NL301097I1 (en) | 2021-03-24 |
| CY1121174T1 (en) | 2020-05-29 |
| LTC2734522I2 (en) | 2022-09-26 |
| LT3689878T (en) | 2021-11-25 |
| ME03310B (en) | 2019-10-20 |
| PT2734522T (en) | 2019-02-04 |
| NO2021016I1 (en) | 2021-04-09 |
| NL301097I2 (en) | 2021-04-12 |
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