NI200700039A - Derivados de triazolopiridinilsulfanilo como inhibidores de quinasa map p38. - Google Patents
Derivados de triazolopiridinilsulfanilo como inhibidores de quinasa map p38.Info
- Publication number
- NI200700039A NI200700039A NI200700039A NI200700039A NI200700039A NI 200700039 A NI200700039 A NI 200700039A NI 200700039 A NI200700039 A NI 200700039A NI 200700039 A NI200700039 A NI 200700039A NI 200700039 A NI200700039 A NI 200700039A
- Authority
- NI
- Nicaragua
- Prior art keywords
- triazolopiridinilsulfanilo
- quinasa
- inhibitors
- map
- derivatives
- Prior art date
Links
- 239000012826 P38 inhibitor Substances 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 2
- 208000035475 disorder Diseases 0.000 abstract 2
- 230000001404 mediated effect Effects 0.000 abstract 2
- 210000002345 respiratory system Anatomy 0.000 abstract 2
- 208000006545 Chronic Obstructive Pulmonary Disease Diseases 0.000 abstract 1
- 208000026935 allergic disease Diseases 0.000 abstract 1
- 230000000172 allergic effect Effects 0.000 abstract 1
- 208000010668 atopic eczema Diseases 0.000 abstract 1
- 208000027866 inflammatory disease Diseases 0.000 abstract 1
- 230000000414 obstructive effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Un compuesto de fórmula (I), o un sal y/o solvato (incluyendo un hidrato) farmacéuticamente aceptable del mismo; y el uso de un compuesto de fórmula (I) en el tratamiento de una enfermedad, trastorno o afección mediada por TNF, o una enfermedad, trastorno o afección mediada por p38, en particular las enfermedades alérgicas y no alérgicas de las vías respiratorias, más particularmente enfermedades obstructivas o inflamatorias de las vías respiratorias, preferiblemente la enfermedad pulmonar obstructiva crónica.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0418015A GB0418015D0 (en) | 2004-08-12 | 2004-08-12 | New compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NI200700039A true NI200700039A (es) | 2008-03-07 |
Family
ID=33017410
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NI200700039A NI200700039A (es) | 2004-08-12 | 2007-02-09 | Derivados de triazolopiridinilsulfanilo como inhibidores de quinasa map p38. |
Country Status (9)
| Country | Link |
|---|---|
| CN (1) | CN101006087B (es) |
| GB (1) | GB0418015D0 (es) |
| ME (1) | ME01360B (es) |
| NI (1) | NI200700039A (es) |
| PE (1) | PE20060618A1 (es) |
| RS (1) | RS50642B (es) |
| TW (1) | TWI295926B (es) |
| UA (1) | UA93032C2 (es) |
| ZA (1) | ZA200700923B (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK2303267T3 (da) * | 2008-02-04 | 2013-09-02 | Pfizer Ltd | Polymorf form af et [1,2,4]-triazolo-[4,3-a]pyridinderivat til behandling af inflammatoriske sygdomme |
| JP2012517992A (ja) * | 2009-02-17 | 2012-08-09 | チェシ ファーマスーティシ エス.ピー.エイ. | P38mapキナーゼインヒビターとしてのトリアゾロピリジン誘導体 |
| GB201009731D0 (en) * | 2010-06-10 | 2010-07-21 | Pulmagen Therapeutics Inflamma | Kinase inhibitors |
| PT2788349T (pt) * | 2011-12-09 | 2017-02-02 | Chiesi Farm Spa | Inibidores de cinase |
| CN105693716A (zh) * | 2016-03-01 | 2016-06-22 | 孙霖 | 晶型a及制备方法 |
| CN105646484A (zh) * | 2016-03-01 | 2016-06-08 | 孙霖 | 晶型b及制备方法 |
-
2004
- 2004-08-12 GB GB0418015A patent/GB0418015D0/en not_active Ceased
-
2005
- 2005-08-09 CN CN2005800274566A patent/CN101006087B/zh not_active Expired - Fee Related
- 2005-08-09 PE PE2005000916A patent/PE20060618A1/es not_active Application Discontinuation
- 2005-08-09 RS RSP-2008/0599A patent/RS50642B/sr unknown
- 2005-08-09 ME MEP-2008-934A patent/ME01360B/me unknown
- 2005-08-09 TW TW94126968A patent/TWI295926B/zh not_active IP Right Cessation
- 2005-08-09 UA UAA200701488A patent/UA93032C2/uk unknown
-
2007
- 2007-01-31 ZA ZA200700923A patent/ZA200700923B/xx unknown
- 2007-02-09 NI NI200700039A patent/NI200700039A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN101006087B (zh) | 2010-09-29 |
| PE20060618A1 (es) | 2006-07-14 |
| TWI295926B (en) | 2008-04-21 |
| ME01360B (me) | 2010-06-30 |
| CN101006087A (zh) | 2007-07-25 |
| TW200610529A (en) | 2006-04-01 |
| GB0418015D0 (en) | 2004-09-15 |
| RS50642B (sr) | 2010-06-30 |
| UA93032C2 (uk) | 2011-01-10 |
| ZA200700923B (en) | 2008-09-25 |
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