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MXPA05001581A - Algunas imidazopiridinas novedosas y su uso. - Google Patents

Algunas imidazopiridinas novedosas y su uso.

Info

Publication number
MXPA05001581A
MXPA05001581A MXPA05001581A MXPA05001581A MXPA05001581A MX PA05001581 A MXPA05001581 A MX PA05001581A MX PA05001581 A MXPA05001581 A MX PA05001581A MX PA05001581 A MXPA05001581 A MX PA05001581A MX PA05001581 A MXPA05001581 A MX PA05001581A
Authority
MX
Mexico
Prior art keywords
formula
disclosed
compounds
imidazopyridines
novel
Prior art date
Application number
MXPA05001581A
Other languages
English (en)
Inventor
Peter Storm
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of MXPA05001581A publication Critical patent/MXPA05001581A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pulmonology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Se describe el uso de compuestos de la formula (1)en donde R1, R3, R10, m y Ar son como se define en la especificacion y sales farmaceuticamente aceptables de los mismos en la manufactura de un medicamento para el tratamiento o profilaxis de enfermedades o condiciones en las cuales la inhibicion de la actividad Itk de la cinasa es benefica. Tambien se describen ciertos compuestos novedosos de la formula (1), junto con los procesos para su preparacion, composiciones que los contienen y su uso en la terapia.
MXPA05001581A 2002-08-14 2003-08-13 Algunas imidazopiridinas novedosas y su uso. MXPA05001581A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0202462A SE0202462D0 (sv) 2002-08-14 2002-08-14 Novel use
PCT/SE2003/001279 WO2004016611A1 (en) 2002-08-14 2003-08-13 Use of and some novel imidazopyridines

Publications (1)

Publication Number Publication Date
MXPA05001581A true MXPA05001581A (es) 2005-04-25

Family

ID=20288750

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA05001581A MXPA05001581A (es) 2002-08-14 2003-08-13 Algunas imidazopiridinas novedosas y su uso.

Country Status (18)

Country Link
US (1) US7410966B2 (es)
EP (1) EP1539759B1 (es)
JP (1) JP2006503010A (es)
KR (1) KR20060005333A (es)
CN (1) CN100358893C (es)
AT (1) ATE370138T1 (es)
AU (1) AU2003251272A1 (es)
BR (1) BR0313461A (es)
CA (1) CA2495511A1 (es)
DE (1) DE60315674T2 (es)
ES (1) ES2290538T3 (es)
IL (1) IL166413A0 (es)
MX (1) MXPA05001581A (es)
NO (1) NO20051265L (es)
NZ (1) NZ538156A (es)
SE (1) SE0202462D0 (es)
WO (1) WO2004016611A1 (es)
ZA (1) ZA200500887B (es)

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Also Published As

Publication number Publication date
DE60315674T2 (de) 2008-06-19
NO20051265L (no) 2005-05-12
CA2495511A1 (en) 2004-02-26
US7410966B2 (en) 2008-08-12
WO2004016611A1 (en) 2004-02-26
DE60315674D1 (de) 2007-09-27
CN1684964A (zh) 2005-10-19
ZA200500887B (en) 2006-02-22
CN100358893C (zh) 2008-01-02
ATE370138T1 (de) 2007-09-15
EP1539759A1 (en) 2005-06-15
ES2290538T3 (es) 2008-02-16
SE0202462D0 (sv) 2002-08-14
US20050261333A1 (en) 2005-11-24
NZ538156A (en) 2006-09-29
EP1539759B1 (en) 2007-08-15
JP2006503010A (ja) 2006-01-26
IL166413A0 (en) 2006-01-15
KR20060005333A (ko) 2006-01-17
BR0313461A (pt) 2005-07-05
AU2003251272A1 (en) 2004-03-03

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