MXPA03009647A - Heterociclildicarbamidas como inhibidores de caspasa. - Google Patents
Heterociclildicarbamidas como inhibidores de caspasa.Info
- Publication number
- MXPA03009647A MXPA03009647A MXPA03009647A MXPA03009647A MXPA03009647A MX PA03009647 A MXPA03009647 A MX PA03009647A MX PA03009647 A MXPA03009647 A MX PA03009647A MX PA03009647 A MXPA03009647 A MX PA03009647A MX PA03009647 A MXPA03009647 A MX PA03009647A
- Authority
- MX
- Mexico
- Prior art keywords
- heterocyclyldicarbamides
- caspase inhibitors
- caspase
- inhibitors
- Prior art date
Links
- 102000011727 Caspases Human genes 0.000 title 1
- 108010076667 Caspases Proteins 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US28505101P | 2001-04-19 | 2001-04-19 | |
| PCT/US2002/012638 WO2002085899A1 (en) | 2001-04-19 | 2002-04-19 | Heterocyclyldicarbamides as caspase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA03009647A true MXPA03009647A (es) | 2004-01-29 |
Family
ID=23092531
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03009647A MXPA03009647A (es) | 2001-04-19 | 2002-04-19 | Heterociclildicarbamidas como inhibidores de caspasa. |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US20030096737A1 (es) |
| EP (1) | EP1381602A1 (es) |
| JP (2) | JP4676676B2 (es) |
| CA (1) | CA2443600A1 (es) |
| MX (1) | MXPA03009647A (es) |
| WO (1) | WO2002085899A1 (es) |
Families Citing this family (45)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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| US6204261B1 (en) | 1995-12-20 | 2001-03-20 | Vertex Pharmaceuticals Incorporated | Inhibitors of interleukin-1β Converting enzyme inhibitors |
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| WO1999018781A1 (en) | 1997-10-10 | 1999-04-22 | Cytovia, Inc. | Dipeptide apoptosis inhibitors and the use thereof |
| DE69925268T2 (de) | 1998-03-16 | 2006-03-23 | Cytovia, Inc., San Diego | Dipeptid-Caspase-Inhibitoren und deren Verwendung |
| US6242422B1 (en) | 1998-10-22 | 2001-06-05 | Idun Pharmacueticals, Inc. | (Substituted)Acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases |
| AU4213500A (en) | 1999-04-09 | 2000-11-14 | Cytovia, Inc. | Caspase inhibitors and the use thereof |
| WO2001044214A1 (en) * | 1999-12-03 | 2001-06-21 | Ono Pharmaceutical Co., Ltd. | Oxadiazole derivatives and drugs containing these derivatives as the active ingredient |
| US6800619B2 (en) * | 2000-09-13 | 2004-10-05 | Vertex Pharmaceuticals Incorporated | Caspase inhibitors and uses thereof |
| AU2003211052A1 (en) * | 2002-02-11 | 2003-09-04 | Vertex Pharmaceuticals Incorporated | Phospholipids as caspase inhibitor prodrugs |
-
2002
- 2002-04-19 WO PCT/US2002/012638 patent/WO2002085899A1/en not_active Ceased
- 2002-04-19 EP EP02723934A patent/EP1381602A1/en not_active Withdrawn
- 2002-04-19 US US10/127,324 patent/US20030096737A1/en not_active Abandoned
- 2002-04-19 JP JP2002583426A patent/JP4676676B2/ja not_active Expired - Fee Related
- 2002-04-19 MX MXPA03009647A patent/MXPA03009647A/es not_active Application Discontinuation
- 2002-04-19 CA CA002443600A patent/CA2443600A1/en not_active Abandoned
-
2006
- 2006-09-14 US US11/522,375 patent/US7807659B2/en not_active Expired - Fee Related
-
2010
- 2010-03-19 JP JP2010065250A patent/JP2010202652A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| JP2004527548A (ja) | 2004-09-09 |
| US20030096737A1 (en) | 2003-05-22 |
| WO2002085899A1 (en) | 2002-10-31 |
| EP1381602A1 (en) | 2004-01-21 |
| JP2010202652A (ja) | 2010-09-16 |
| US7807659B2 (en) | 2010-10-05 |
| CA2443600A1 (en) | 2002-10-31 |
| US20070010457A1 (en) | 2007-01-11 |
| JP4676676B2 (ja) | 2011-04-27 |
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| Date | Code | Title | Description |
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| FA | Abandonment or withdrawal |