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MXPA03005270A - Derivados de piperazina. - Google Patents

Derivados de piperazina.

Info

Publication number
MXPA03005270A
MXPA03005270A MXPA03005270A MXPA03005270A MXPA03005270A MX PA03005270 A MXPA03005270 A MX PA03005270A MX PA03005270 A MXPA03005270 A MX PA03005270A MX PA03005270 A MXPA03005270 A MX PA03005270A MX PA03005270 A MXPA03005270 A MX PA03005270A
Authority
MX
Mexico
Prior art keywords
piperazine derivatives
piperazine
derivatives
Prior art date
Application number
MXPA03005270A
Other languages
English (en)
Inventor
Jacques Mizrahi
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MXPA03005270A publication Critical patent/MXPA03005270A/es

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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
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    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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MXPA03005270A 2000-12-15 2001-12-06 Derivados de piperazina. MXPA03005270A (es)

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GBGB0030710.8A GB0030710D0 (en) 2000-12-15 2000-12-15 Piperazine derivatives
PCT/EP2001/014343 WO2002048124A2 (en) 2000-12-15 2001-12-06 Piperazine derivatives

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ES2306736T3 (es) 2008-11-16
EP1343775A2 (en) 2003-09-17
EP1343775B1 (en) 2008-06-04
CA2430601A1 (en) 2002-06-20
JP2004519438A (ja) 2004-07-02
UY27075A1 (es) 2002-07-31
PE20020667A1 (es) 2002-07-27
PA8534801A1 (es) 2002-08-26
AU2962602A (en) 2002-06-24
JP4047724B2 (ja) 2008-02-13
BR0116201A (pt) 2004-03-02
WO2002048124A2 (en) 2002-06-20
KR20030072563A (ko) 2003-09-15
ZA200304346B (en) 2004-09-03
CA2430601C (en) 2008-05-06
US20040235859A1 (en) 2004-11-25
AR035517A1 (es) 2004-06-02
ATE397595T1 (de) 2008-06-15
KR100623833B1 (ko) 2006-09-18
US20020143020A1 (en) 2002-10-03
CN1533382A (zh) 2004-09-29
DE60134338D1 (de) 2008-07-17
US7022707B2 (en) 2006-04-04
CN1277824C (zh) 2006-10-04
GB0030710D0 (en) 2001-01-31
WO2002048124A3 (en) 2003-06-05

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