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MXPA02005103A - Ligandos selectivos del receptor de canabinoide (cb2) perifericos. - Google Patents

Ligandos selectivos del receptor de canabinoide (cb2) perifericos.

Info

Publication number
MXPA02005103A
MXPA02005103A MXPA02005103A MXPA02005103A MXPA02005103A MX PA02005103 A MXPA02005103 A MX PA02005103A MX PA02005103 A MXPA02005103 A MX PA02005103A MX PA02005103 A MXPA02005103 A MX PA02005103A MX PA02005103 A MXPA02005103 A MX PA02005103A
Authority
MX
Mexico
Prior art keywords
cannabinoid receptor
selective ligands
peripheral cannabinoid
peripheral
ligands
Prior art date
Application number
MXPA02005103A
Other languages
English (en)
Inventor
Alexandros Makriyannis
Original Assignee
Alexipharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alexipharma Inc filed Critical Alexipharma Inc
Publication of MXPA02005103A publication Critical patent/MXPA02005103A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
MXPA02005103A 1999-10-18 2000-10-18 Ligandos selectivos del receptor de canabinoide (cb2) perifericos. MXPA02005103A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US16014699P 1999-10-18 1999-10-18
PCT/US2000/028818 WO2001028329A1 (en) 1999-10-18 2000-10-18 Peripheral cannabinoid receptor (cb2) selective ligands

Publications (1)

Publication Number Publication Date
MXPA02005103A true MXPA02005103A (es) 2003-09-25

Family

ID=22575729

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA02005103A MXPA02005103A (es) 1999-10-18 2000-10-18 Ligandos selectivos del receptor de canabinoide (cb2) perifericos.

Country Status (9)

Country Link
US (1) US6995187B1 (es)
EP (1) EP1223808B1 (es)
JP (1) JP2003511469A (es)
AU (1) AU778159B2 (es)
CA (1) CA2387764A1 (es)
DE (1) DE60033834T2 (es)
MX (1) MXPA02005103A (es)
WO (1) WO2001028329A1 (es)
ZA (1) ZA200203908B (es)

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US7897598B2 (en) 1998-06-09 2011-03-01 Alexandros Makriyannis Inhibitors of the anandamide transporter
US7276613B1 (en) 1998-11-24 2007-10-02 University Of Connecticut Retro-anandamides, high affinity and stability cannabinoid receptor ligands
US7161016B1 (en) 1998-11-24 2007-01-09 University Of Connecticut Cannabimimetic lipid amides as useful medications
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US7393842B2 (en) 2001-08-31 2008-07-01 University Of Connecticut Pyrazole analogs acting on cannabinoid receptors
US6943266B1 (en) * 1999-10-18 2005-09-13 University Of Connecticut Bicyclic cannabinoid agonists for the cannabinoid receptor
US7119108B1 (en) * 1999-10-18 2006-10-10 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US8084467B2 (en) * 1999-10-18 2011-12-27 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US7741365B2 (en) * 1999-10-18 2010-06-22 University Of Connecticut Peripheral cannabinoid receptor (CB2) selective ligands
US7329651B2 (en) 2001-01-26 2008-02-12 University Of Connecticut Cannabimimetic ligands
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Also Published As

Publication number Publication date
WO2001028329A1 (en) 2001-04-26
US6995187B1 (en) 2006-02-07
AU1213601A (en) 2001-04-30
AU778159B2 (en) 2004-11-18
DE60033834T2 (de) 2007-11-15
JP2003511469A (ja) 2003-03-25
DE60033834D1 (de) 2007-04-19
ZA200203908B (en) 2004-12-29
EP1223808A1 (en) 2002-07-24
CA2387764A1 (en) 2001-04-26
EP1223808A4 (en) 2003-04-02
EP1223808B1 (en) 2007-03-07

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