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MXPA02003114A - Dispersiones para formular ingredientes activos ligeramente o poco solubles. - Google Patents

Dispersiones para formular ingredientes activos ligeramente o poco solubles.

Info

Publication number
MXPA02003114A
MXPA02003114A MXPA02003114A MXPA02003114A MXPA02003114A MX PA02003114 A MXPA02003114 A MX PA02003114A MX PA02003114 A MXPA02003114 A MX PA02003114A MX PA02003114 A MXPA02003114 A MX PA02003114A MX PA02003114 A MXPA02003114 A MX PA02003114A
Authority
MX
Mexico
Prior art keywords
slightly
formulate
dispersions
active ingredients
little active
Prior art date
Application number
MXPA02003114A
Other languages
English (en)
Inventor
Helmut M Ller Rainer
Original Assignee
Pharmasol Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7650573&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MXPA02003114(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmasol Gmbh filed Critical Pharmasol Gmbh
Publication of MXPA02003114A publication Critical patent/MXPA02003114A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Virology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Colloid Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invencion se refiere a una dispersion que comprende una fase aceitosa y una fase acuosa en la forma de una emulsion aceite/agua o una solucion agua/aceite, por lo menos un ingrediente activo el cual es ligeramente o poco soluble en fases aceitosas y acuosas, ademas de uno o mas emulsificadores y/o estabilizadores opcionales. La dispersion esta desprovista de solventes organicos cuestionables toxicologicamente y contiene una cantidad disuelta de dicho ingrediente activo que es mayor que la cantidad de aditivo obtenida por su solubilidad maxima, tanto en la fase aceitosa como la fase acuosa de la emulsion.
MXPA02003114A 2000-07-28 2001-07-27 Dispersiones para formular ingredientes activos ligeramente o poco solubles. MXPA02003114A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10036871A DE10036871A1 (de) 2000-07-28 2000-07-28 Dispersionen zur Formulierung wenig oder schwer löslicher Wirkstoffe
PCT/EP2001/008726 WO2002009667A2 (de) 2000-07-28 2001-07-27 Dispersionen zur formulierung wenig oder schwer löslicher wirkstoffe

Publications (1)

Publication Number Publication Date
MXPA02003114A true MXPA02003114A (es) 2003-04-10

Family

ID=7650573

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA02003114A MXPA02003114A (es) 2000-07-28 2001-07-27 Dispersiones para formular ingredientes activos ligeramente o poco solubles.

Country Status (15)

Country Link
US (2) US7060285B2 (es)
EP (1) EP1305006B1 (es)
JP (1) JP2004505032A (es)
KR (1) KR20020063869A (es)
CN (1) CN1620283A (es)
AT (1) ATE401055T1 (es)
AU (1) AU8976801A (es)
BR (1) BR0107042A (es)
CA (1) CA2388550A1 (es)
DE (2) DE10036871A1 (es)
ES (1) ES2307644T3 (es)
MX (1) MXPA02003114A (es)
PL (1) PL365874A1 (es)
RU (1) RU2002111336A (es)
WO (1) WO2002009667A2 (es)

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AU2002214233A1 (en) * 2001-11-01 2003-07-09 Novagali Pharma Sa Method and composition for dry eye treatment
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US20040022820A1 (en) * 2001-11-28 2004-02-05 David Anderson Reversed liquid crystalline phases with non-paraffin hydrophobes
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Also Published As

Publication number Publication date
US7060285B2 (en) 2006-06-13
KR20020063869A (ko) 2002-08-05
BR0107042A (pt) 2002-06-04
US20030059470A1 (en) 2003-03-27
US20060188534A1 (en) 2006-08-24
US7744909B2 (en) 2010-06-29
WO2002009667A3 (de) 2002-11-07
ES2307644T3 (es) 2008-12-01
ATE401055T1 (de) 2008-08-15
WO2002009667A9 (de) 2002-02-28
AU8976801A (en) 2002-02-13
EP1305006A2 (de) 2003-05-02
PL365874A1 (pl) 2005-01-10
CN1620283A (zh) 2005-05-25
EP1305006B1 (de) 2008-07-16
JP2004505032A (ja) 2004-02-19
DE10036871A1 (de) 2002-02-14
RU2002111336A (ru) 2003-11-20
CA2388550A1 (en) 2002-02-07
WO2002009667A2 (de) 2002-02-07
DE50114130D1 (de) 2008-08-28

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