MXPA02002712A - Profarmacos anfifilicos. - Google Patents
Profarmacos anfifilicos.Info
- Publication number
- MXPA02002712A MXPA02002712A MXPA02002712A MXPA02002712A MXPA02002712A MX PA02002712 A MXPA02002712 A MX PA02002712A MX PA02002712 A MXPA02002712 A MX PA02002712A MX PA02002712 A MXPA02002712 A MX PA02002712A MX PA02002712 A MXPA02002712 A MX PA02002712A
- Authority
- MX
- Mexico
- Prior art keywords
- amphiphilic prodrugs
- amphiphilic
- prodrugs
- Prior art date
Links
- 229940002612 prodrug Drugs 0.000 title 1
- 239000000651 prodrug Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
- A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
- A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US15364999P | 1999-09-13 | 1999-09-13 | |
| US09/474,915 US6713454B1 (en) | 1999-09-13 | 1999-12-31 | Prodrugs of etoposide and etoposide analogs |
| PCT/US2000/024520 WO2001019406A2 (en) | 1999-09-13 | 2000-09-07 | Amphiphilic prodrugs |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA02002712A true MXPA02002712A (es) | 2003-10-14 |
Family
ID=26850733
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA02002712A MXPA02002712A (es) | 1999-09-13 | 2000-09-07 | Profarmacos anfifilicos. |
Country Status (17)
| Country | Link |
|---|---|
| US (3) | US6713454B1 (es) |
| EP (1) | EP1212099A2 (es) |
| JP (1) | JP2003509385A (es) |
| KR (1) | KR20020059398A (es) |
| CN (1) | CN1390143A (es) |
| AU (1) | AU7575600A (es) |
| BR (1) | BR0013948A (es) |
| CA (1) | CA2384645A1 (es) |
| CZ (1) | CZ2002928A3 (es) |
| HU (1) | HUP0204110A3 (es) |
| IL (1) | IL148558A0 (es) |
| MX (1) | MXPA02002712A (es) |
| NO (1) | NO20021213L (es) |
| NZ (1) | NZ517681A (es) |
| PL (1) | PL354261A1 (es) |
| RU (1) | RU2002109595A (es) |
| WO (1) | WO2001019406A2 (es) |
Families Citing this family (62)
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|---|---|---|---|---|
| US6703381B1 (en) * | 1998-08-14 | 2004-03-09 | Nobex Corporation | Methods for delivery therapeutic compounds across the blood-brain barrier |
| US6541508B2 (en) | 1999-09-13 | 2003-04-01 | Nobex Corporation | Taxane prodrugs |
| US6713454B1 (en) * | 1999-09-13 | 2004-03-30 | Nobex Corporation | Prodrugs of etoposide and etoposide analogs |
| US6380405B1 (en) | 1999-09-13 | 2002-04-30 | Nobex Corporation | Taxane prodrugs |
| KR100619612B1 (ko) * | 1999-10-04 | 2006-09-01 | 넥타르 테라퓨틱스 에이엘, 코포레이션 | 폴리머 안정화 신경펩타이드 |
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| US7632866B2 (en) | 2002-10-21 | 2009-12-15 | Ramot At Tel Aviv University | Derivatives of N-phenylanthranilic acid and 2-benzimidazolone as potassium channel and/or neuron activity modulators |
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| ES2744225T3 (es) | 2005-07-15 | 2020-02-24 | Angiochem Inc | Uso de polipéptidos de aprotinina como portadores en conjugados farmacéuticos |
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| US6703381B1 (en) | 1998-08-14 | 2004-03-09 | Nobex Corporation | Methods for delivery therapeutic compounds across the blood-brain barrier |
| EP1176985A2 (en) | 1999-04-28 | 2002-02-06 | Vectramed, Inc. | Enzymatically activated polymeric drug conjugates |
| US6309633B1 (en) | 1999-06-19 | 2001-10-30 | Nobex Corporation | Amphiphilic drug-oligomer conjugates with hydroyzable lipophile components and methods for making and using the same |
| EP1210121A2 (en) | 1999-08-24 | 2002-06-05 | Cellgate Inc. | Enhancing drug delivery across and into epithelial tissues using oligo arginine moieties |
| US6541508B2 (en) | 1999-09-13 | 2003-04-01 | Nobex Corporation | Taxane prodrugs |
| US6380405B1 (en) * | 1999-09-13 | 2002-04-30 | Nobex Corporation | Taxane prodrugs |
| US6713454B1 (en) | 1999-09-13 | 2004-03-30 | Nobex Corporation | Prodrugs of etoposide and etoposide analogs |
-
1999
- 1999-12-31 US US09/474,915 patent/US6713454B1/en not_active Expired - Fee Related
-
2000
- 2000-09-07 CN CN00815508A patent/CN1390143A/zh active Pending
- 2000-09-07 NZ NZ517681A patent/NZ517681A/en unknown
- 2000-09-07 IL IL14855800A patent/IL148558A0/xx unknown
- 2000-09-07 PL PL00354261A patent/PL354261A1/xx not_active Application Discontinuation
- 2000-09-07 HU HU0204110A patent/HUP0204110A3/hu unknown
- 2000-09-07 CA CA002384645A patent/CA2384645A1/en not_active Abandoned
- 2000-09-07 RU RU2002109595/14A patent/RU2002109595A/ru not_active Application Discontinuation
- 2000-09-07 BR BR0013948-3A patent/BR0013948A/pt not_active IP Right Cessation
- 2000-09-07 CZ CZ2002928A patent/CZ2002928A3/cs unknown
- 2000-09-07 JP JP2001523037A patent/JP2003509385A/ja active Pending
- 2000-09-07 KR KR1020027003276A patent/KR20020059398A/ko not_active Withdrawn
- 2000-09-07 AU AU75756/00A patent/AU7575600A/en not_active Abandoned
- 2000-09-07 WO PCT/US2000/024520 patent/WO2001019406A2/en not_active Ceased
- 2000-09-07 EP EP00964949A patent/EP1212099A2/en not_active Withdrawn
- 2000-09-07 MX MXPA02002712A patent/MXPA02002712A/es unknown
-
2002
- 2002-03-12 NO NO20021213A patent/NO20021213L/no not_active Application Discontinuation
-
2004
- 2004-03-24 US US10/808,044 patent/US7119074B2/en not_active Expired - Fee Related
- 2004-03-29 US US10/811,760 patent/US20040253206A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US6713454B1 (en) | 2004-03-30 |
| NO20021213L (no) | 2002-05-13 |
| US20040180840A1 (en) | 2004-09-16 |
| BR0013948A (pt) | 2002-05-14 |
| PL354261A1 (en) | 2003-12-29 |
| CA2384645A1 (en) | 2001-03-22 |
| US20040253206A1 (en) | 2004-12-16 |
| CN1390143A (zh) | 2003-01-08 |
| US7119074B2 (en) | 2006-10-10 |
| HUP0204110A2 (hu) | 2003-04-28 |
| RU2002109595A (ru) | 2003-11-27 |
| IL148558A0 (en) | 2002-09-12 |
| HUP0204110A3 (en) | 2003-08-28 |
| AU7575600A (en) | 2001-04-17 |
| WO2001019406A3 (en) | 2002-01-17 |
| EP1212099A2 (en) | 2002-06-12 |
| JP2003509385A (ja) | 2003-03-11 |
| NO20021213D0 (no) | 2002-03-12 |
| CZ2002928A3 (cs) | 2002-09-11 |
| WO2001019406A2 (en) | 2001-03-22 |
| NZ517681A (en) | 2004-01-30 |
| KR20020059398A (ko) | 2002-07-12 |
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