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MXPA01011287A - Derivados de ciclotiocarbamato como moduladores de receptor de progesterona. - Google Patents

Derivados de ciclotiocarbamato como moduladores de receptor de progesterona.

Info

Publication number
MXPA01011287A
MXPA01011287A MXPA01011287A MXPA01011287A MXPA01011287A MX PA01011287 A MXPA01011287 A MX PA01011287A MX PA01011287 A MXPA01011287 A MX PA01011287A MX PA01011287 A MXPA01011287 A MX PA01011287A MX PA01011287 A MXPA01011287 A MX PA01011287A
Authority
MX
Mexico
Prior art keywords
alkyl
optionally substituted
aryl
ring
groups
Prior art date
Application number
MXPA01011287A
Other languages
English (en)
Inventor
P Edwards James
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/552,354 external-priority patent/US6436929B1/en
Application filed by American Home Prod filed Critical American Home Prod
Publication of MXPA01011287A publication Critical patent/MXPA01011287A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Chemical Or Physical Treatment Of Fibers (AREA)
  • Detergent Compositions (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MXPA01011287A 1999-05-04 2000-05-01 Derivados de ciclotiocarbamato como moduladores de receptor de progesterona. MXPA01011287A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18301399P 1999-05-04 1999-05-04
US09/552,354 US6436929B1 (en) 1999-05-04 2000-04-19 Cyclothiocarbamate derivatives as progesterone receptor modulators
PCT/US2000/011749 WO2000066570A1 (en) 1999-05-04 2000-05-01 Cyclothiocarbamate derivatives as progesterone receptor modulators

Publications (1)

Publication Number Publication Date
MXPA01011287A true MXPA01011287A (es) 2003-07-14

Family

ID=26878649

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA01011287A MXPA01011287A (es) 1999-05-04 2000-05-01 Derivados de ciclotiocarbamato como moduladores de receptor de progesterona.

Country Status (24)

Country Link
EP (1) EP1175411B1 (es)
JP (2) JP4958338B2 (es)
KR (1) KR100732692B1 (es)
CN (1) CN1131856C (es)
AT (1) ATE386729T1 (es)
AU (1) AU766801B2 (es)
BG (1) BG65277B1 (es)
BR (1) BR0010214A (es)
CA (1) CA2371712C (es)
CZ (1) CZ20013952A3 (es)
DE (1) DE60038108T2 (es)
DK (1) DK1175411T3 (es)
EA (1) EA004511B1 (es)
ES (1) ES2301482T3 (es)
GE (1) GEP20043181B (es)
HU (1) HUP0203332A3 (es)
IL (1) IL146298A0 (es)
MX (1) MXPA01011287A (es)
NO (1) NO321370B1 (es)
NZ (1) NZ515353A (es)
PL (1) PL351083A1 (es)
SG (1) SG120970A1 (es)
SK (1) SK15922001A3 (es)
TR (1) TR200103285T2 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK15922001A3 (sk) * 1999-05-04 2002-09-10 American Home Products Corporation Deriváty cyklotiokarbamátu ako modulátory receptora pre progesterón
US6407101B1 (en) * 1999-05-04 2002-06-18 American Home Products Corporation Cyanopyrroles
WO2005100346A1 (en) * 2004-04-08 2005-10-27 Wyeth Thioamide derivatives as progesterone receptor modulators
CN1938298B (zh) * 2004-04-08 2013-02-06 惠氏公司 减少硫代酰胺杂质的方法
CN1953967B (zh) 2004-04-27 2013-03-13 惠氏公司 孕酮受体调节剂的纯化
PL1756095T3 (pl) * 2004-04-27 2008-10-31 Wyeth Corp Cyjanopirole zawierające cykliczne karbaminianowe i tiokarbaminianowe biaryle oraz sposoby ich wytwarzania
TW200603813A (en) * 2004-07-07 2006-02-01 Wyeth Corp Cyclic progestin regimens and kits
CA2575737C (en) 2004-08-13 2013-09-24 Wyeth Tanaproget derivatives, metabolites, and uses thereof
ATE461701T1 (de) 2005-04-28 2010-04-15 Wyeth Corp Mikronisiertes tanaproget und zusammensetzungen damit
BRPI0610438A2 (pt) * 2005-04-28 2012-10-23 Wyeth Corp composição farmacêutica, cápsula, conjunto farmacêutico, e, processo para preparar uma composição
CN101166736B (zh) * 2005-04-28 2013-02-06 惠氏公司 他那普戈特的多晶型ⅱ
AR053595A1 (es) * 2005-04-28 2007-05-09 Wyeth Corp Forma purificada de tanaproget
PL1896034T3 (pl) 2005-04-28 2010-07-30 Wyeth Llc Mikronizowane kompozycje tanaprogetu i sposoby ich wytwarzania
BRPI0611250A2 (pt) * 2005-06-09 2011-02-15 Wyeth Corp composto, enanciÈmeros, diastereoisÈmeros do mesmo ou um sal farmaceuticamente aceitável do mesmo, composição farmacêutica, e, uso de um composto

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0510235A1 (en) * 1991-04-26 1992-10-28 Dong-A Pharm. Co., Ltd. Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same
JPH0510235A (ja) * 1991-07-05 1993-01-19 Nippondenso Co Ltd 内燃機関の点火時期制御装置
AU1694295A (en) * 1994-01-28 1995-08-15 Merck & Co., Inc. Benzoxazinones as inhibitors of hiv reverse transcriptase
US5696133A (en) * 1994-12-22 1997-12-09 Ligand Pharmaceuticals Incorporated Steroid receptor modulator compounds and methods
JPH10510840A (ja) * 1994-12-22 1998-10-20 リガンド・ファーマシューティカルズ・インコーポレイテッド ステロイド受容体モジュレーター化合物および方法
EP0929533B1 (en) * 1996-10-02 2003-09-03 Bristol-Myers Squibb Pharma Company 4,4-disubstituted-1,4-dihydro-2h-3,1-benzoxazin-2-ones useful as hiv reverse transcriptase inhibitors and intermediates and processes for making the same
SK15922001A3 (sk) * 1999-05-04 2002-09-10 American Home Products Corporation Deriváty cyklotiokarbamátu ako modulátory receptora pre progesterón
ATE461701T1 (de) * 2005-04-28 2010-04-15 Wyeth Corp Mikronisiertes tanaproget und zusammensetzungen damit
BRPI0611250A2 (pt) * 2005-06-09 2011-02-15 Wyeth Corp composto, enanciÈmeros, diastereoisÈmeros do mesmo ou um sal farmaceuticamente aceitável do mesmo, composição farmacêutica, e, uso de um composto

Also Published As

Publication number Publication date
CN1349516A (zh) 2002-05-15
NO20015381D0 (no) 2001-11-02
NO321370B1 (no) 2006-05-02
JP2012087129A (ja) 2012-05-10
NO20015381L (no) 2002-01-03
BR0010214A (pt) 2002-02-13
GEP20043181B (en) 2004-02-25
EP1175411B1 (en) 2008-02-20
CN1131856C (zh) 2003-12-24
SK15922001A3 (sk) 2002-09-10
CA2371712A1 (en) 2000-11-09
AU766801B2 (en) 2003-10-23
DK1175411T3 (da) 2008-06-09
AU4811900A (en) 2000-11-17
JP2002543192A (ja) 2002-12-17
BG65277B1 (bg) 2007-11-30
EP1175411A1 (en) 2002-01-30
TR200103285T2 (tr) 2002-02-21
NZ515353A (en) 2004-03-26
CZ20013952A3 (cs) 2002-05-15
KR100732692B1 (ko) 2007-06-27
ATE386729T1 (de) 2008-03-15
CA2371712C (en) 2009-12-22
DE60038108T2 (de) 2009-02-12
KR20020000170A (ko) 2002-01-04
HUP0203332A3 (en) 2004-12-28
DE60038108D1 (de) 2008-04-03
JP5523430B2 (ja) 2014-06-18
ES2301482T3 (es) 2008-07-01
SG120970A1 (en) 2006-04-26
HUP0203332A2 (hu) 2003-01-28
JP4958338B2 (ja) 2012-06-20
EA004511B1 (ru) 2004-04-29
EA200101181A1 (ru) 2002-04-25
PL351083A1 (en) 2003-03-10
BG106080A (en) 2002-05-31
IL146298A0 (en) 2002-07-25

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