MX9806036A - Compuestos para inhibir tumores en el colon. - Google Patents
Compuestos para inhibir tumores en el colon.Info
- Publication number
- MX9806036A MX9806036A MX9806036A MX9806036A MX9806036A MX 9806036 A MX9806036 A MX 9806036A MX 9806036 A MX9806036 A MX 9806036A MX 9806036 A MX9806036 A MX 9806036A MX 9806036 A MX9806036 A MX 9806036A
- Authority
- MX
- Mexico
- Prior art keywords
- methods
- colon tumors
- inhibiting colon
- inhibiting
- hexamethyleneimino
- Prior art date
Links
- 208000029742 colonic neoplasm Diseases 0.000 title abstract 2
- 230000002401 inhibitory effect Effects 0.000 title abstract 2
- RWRDLPDLKQPQOW-UHFFFAOYSA-N tetrahydropyrrole Natural products C1CCNC1 RWRDLPDLKQPQOW-UHFFFAOYSA-N 0.000 abstract 2
- 206010009944 Colon cancer Diseases 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- -1 hexamethyleneimino Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000000587 piperidin-1-yl group Chemical group [H]C1([H])N(*)C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
- 125000000719 pyrrolidinyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4535—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Gastroenterology & Hepatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Pyrrole Compounds (AREA)
Abstract
Un método para inhibir el cáncer de colon que comprende la administracion a un mamífero que necesita del mismo, una cantidad efectiva de un compuesto que tiene la formula (I, en donde R1 y R3 son independientemente hidrogeno, -CH3, (a), o (b), en donde Ar es fenilo opcionalmente sustituido; R2 se selecciona del grupo que consiste de pirrolidina, hexametilenimino y piperidino; o una sal farmacéuticamente aceptable o solvato del mismo.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1077296P | 1996-01-29 | 1996-01-29 | |
| GBGB9603150.5A GB9603150D0 (en) | 1996-02-15 | 1996-02-15 | Methods of inhibiting colon tumors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9806036A true MX9806036A (es) | 1998-11-29 |
Family
ID=26308709
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9806036A MX9806036A (es) | 1996-01-29 | 1998-07-27 | Compuestos para inhibir tumores en el colon. |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP0921799A4 (es) |
| JP (1) | JP2000503994A (es) |
| KR (1) | KR19990082054A (es) |
| CN (1) | CN1209745A (es) |
| AR (1) | AR010978A1 (es) |
| AU (1) | AU707892B2 (es) |
| BR (1) | BR9700778A (es) |
| CO (1) | CO4761062A1 (es) |
| CZ (1) | CZ235498A3 (es) |
| EA (1) | EA001104B1 (es) |
| ID (1) | ID15917A (es) |
| IL (1) | IL125521A (es) |
| MX (1) | MX9806036A (es) |
| NO (1) | NO983451L (es) |
| NZ (1) | NZ331105A (es) |
| PL (1) | PL328147A1 (es) |
| TW (1) | TW446560B (es) |
| WO (1) | WO1997026877A1 (es) |
| YU (1) | YU2397A (es) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW366342B (en) * | 1992-07-28 | 1999-08-11 | Lilly Co Eli | The use of 2-phenyl-3-aroylbenzothiophenes in inhibiting bone loss |
| IL111287A0 (en) * | 1993-10-15 | 1994-12-29 | Lilly Co Eli | Methods for treating resistant neoplasms |
| US5574047A (en) * | 1993-12-21 | 1996-11-12 | Eli Lilly And Company | Methods of inhibiting imperfect tissue repair |
-
1997
- 1997-01-22 ID IDP970182A patent/ID15917A/id unknown
- 1997-01-24 YU YU2397A patent/YU2397A/sr unknown
- 1997-01-24 AR ARP970100300A patent/AR010978A1/es unknown
- 1997-01-25 TW TW086100832A patent/TW446560B/zh not_active IP Right Cessation
- 1997-01-27 CN CN97191791A patent/CN1209745A/zh active Pending
- 1997-01-27 PL PL97328147A patent/PL328147A1/xx unknown
- 1997-01-27 EP EP97906587A patent/EP0921799A4/en not_active Withdrawn
- 1997-01-27 IL IL12552197A patent/IL125521A/en not_active IP Right Cessation
- 1997-01-27 JP JP9527132A patent/JP2000503994A/ja active Pending
- 1997-01-27 NZ NZ331105A patent/NZ331105A/en unknown
- 1997-01-27 AU AU21239/97A patent/AU707892B2/en not_active Ceased
- 1997-01-27 EA EA199800677A patent/EA001104B1/ru not_active IP Right Cessation
- 1997-01-27 WO PCT/US1997/002286 patent/WO1997026877A1/en not_active Ceased
- 1997-01-27 CZ CZ982354A patent/CZ235498A3/cs unknown
- 1997-01-27 KR KR1019980705775A patent/KR19990082054A/ko not_active Ceased
- 1997-01-27 BR BR9700778A patent/BR9700778A/pt active Search and Examination
- 1997-01-28 CO CO97003856A patent/CO4761062A1/es unknown
-
1998
- 1998-07-27 MX MX9806036A patent/MX9806036A/es unknown
- 1998-07-27 NO NO983451A patent/NO983451L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| NZ331105A (en) | 2000-06-23 |
| IL125521A (en) | 2001-11-25 |
| CN1209745A (zh) | 1999-03-03 |
| TW446560B (en) | 2001-07-21 |
| NO983451D0 (no) | 1998-07-27 |
| EP0921799A4 (en) | 2002-03-13 |
| AU2123997A (en) | 1997-08-20 |
| YU2397A (en) | 1999-11-22 |
| CO4761062A1 (es) | 1999-04-27 |
| EA001104B1 (ru) | 2000-10-30 |
| NO983451L (no) | 1998-07-27 |
| ID15917A (id) | 1997-08-21 |
| WO1997026877A1 (en) | 1997-07-31 |
| EP0921799A1 (en) | 1999-06-16 |
| AR010978A1 (es) | 2000-08-02 |
| IL125521A0 (en) | 1999-03-12 |
| EA199800677A1 (ru) | 1999-02-25 |
| PL328147A1 (en) | 1999-01-18 |
| KR19990082054A (ko) | 1999-11-15 |
| BR9700778A (pt) | 1998-10-06 |
| CZ235498A3 (cs) | 1999-02-17 |
| AU707892B2 (en) | 1999-07-22 |
| JP2000503994A (ja) | 2000-04-04 |
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