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MX9710403A - Uso de ritonavir (abt-538) para mejorar la farmacocinetica de farmacos metabolizados a traves de citrocromo p450 en un metodo para el tratamiento del sida. - Google Patents

Uso de ritonavir (abt-538) para mejorar la farmacocinetica de farmacos metabolizados a traves de citrocromo p450 en un metodo para el tratamiento del sida.

Info

Publication number
MX9710403A
MX9710403A MX9710403A MX9710403A MX9710403A MX 9710403 A MX9710403 A MX 9710403A MX 9710403 A MX9710403 A MX 9710403A MX 9710403 A MX9710403 A MX 9710403A MX 9710403 A MX9710403 A MX 9710403A
Authority
MX
Mexico
Prior art keywords
cytochrome
pharmacokinetics
improving
ritonavir
abt
Prior art date
Application number
MX9710403A
Other languages
English (en)
Other versions
MXPA97010403A (es
Inventor
Daniel W Norbeck
Dale J Kempf
John M Leonard
Richard J Bertz
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26667933&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX9710403(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of MX9710403A publication Critical patent/MX9710403A/es
Publication of MXPA97010403A publication Critical patent/MXPA97010403A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/453Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/341Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/05Dipeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/06Tripeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/55Protease inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)

Abstract

Se describe un método para mejorar la farmacocinética de un fármaco, el cual es metabolizado a través de monooxigenadas de citocromo P450.
MXPA/A/1997/010403A 1995-06-29 1997-12-18 Uso de ritonavir (abt-538) para mejorar la farmacocinetica de farmacos metabolizados a traves de citocromo p450 en un metodo para el tratamiento del sida MXPA97010403A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US000654 1987-01-06
US003849 1987-01-14
US65495P 1995-06-29 1995-06-29
US384995P 1995-09-15 1995-09-15
PCT/US1996/011015 WO1997001349A1 (en) 1995-06-29 1996-06-28 Use of ritonavir (abt-538) for improving the pharmacokinetics of drugs metabolized by cytochrome p450 in a method of treating aids

Publications (2)

Publication Number Publication Date
MX9710403A true MX9710403A (es) 1998-07-31
MXPA97010403A MXPA97010403A (es) 1998-11-09

Family

ID=

Also Published As

Publication number Publication date
EP1210941A2 (en) 2002-06-05
EP0871465A1 (en) 1998-10-21
JP5364871B2 (ja) 2013-12-11
EP1273298A2 (en) 2003-01-08
CA2224738A1 (en) 1997-01-16
DE69624136D1 (de) 2002-11-07
EP2295052B1 (en) 2014-01-08
AU6342096A (en) 1997-01-30
EP1273298A3 (en) 2003-03-19
JP2012111775A (ja) 2012-06-14
PT871465E (pt) 2003-02-28
EP0871465B1 (en) 2002-10-02
HK1053782A1 (en) 2003-11-07
PT1293207E (pt) 2009-08-11
WO1997001349A1 (en) 1997-01-16
CA2224738C (en) 2002-08-27
US6037157A (en) 2000-03-14
KR100824547B1 (ko) 2008-11-04
ES2328559T3 (es) 2009-11-16
EP1210941A3 (en) 2002-07-31
ES2186787T3 (es) 2003-05-16
US20020039998A1 (en) 2002-04-04
EP1293207B1 (en) 2009-07-22
DE69637511D1 (de) 2008-06-05
DK1293207T3 (da) 2009-10-05
PT2295052E (pt) 2014-01-23
ATE225186T1 (de) 2002-10-15
HK1016088A1 (en) 1999-10-29
IL122546A (en) 2012-01-31
EP1284140B1 (en) 2008-04-23
JP4023823B2 (ja) 2007-12-19
DE69637511T2 (de) 2009-06-04
PT1284140E (pt) 2008-05-14
US6703403B2 (en) 2004-03-09
HK1049103A1 (en) 2003-05-02
EP1284140A3 (en) 2003-03-19
ATE392895T1 (de) 2008-05-15
ES2441736T3 (es) 2014-02-06
KR19990028407A (ko) 1999-04-15
EP1284140A2 (en) 2003-02-19
DK0871465T3 (da) 2003-02-03
DK1284140T3 (da) 2008-08-18
DE69624136T2 (de) 2003-08-14
HK1053783A1 (en) 2003-11-07
EP1293207A1 (en) 2003-03-19
JP2015013878A (ja) 2015-01-22
AU722812B2 (en) 2000-08-10
KR20070120619A (ko) 2007-12-24
IL122546A0 (en) 1998-06-15
EP2130534A1 (en) 2009-12-09
DE69637976D1 (de) 2009-09-03
DK2295052T3 (da) 2014-01-20
JPH11508884A (ja) 1999-08-03
EP2295052A1 (en) 2011-03-16
JP2007291131A (ja) 2007-11-08
ES2304416T3 (es) 2008-10-16

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