MX9708057A - Sulfonamidas que contienen thf inhibidoras de la aspartilproteasa. - Google Patents
Sulfonamidas que contienen thf inhibidoras de la aspartilproteasa.Info
- Publication number
- MX9708057A MX9708057A MX9708057A MX9708057A MX9708057A MX 9708057 A MX9708057 A MX 9708057A MX 9708057 A MX9708057 A MX 9708057A MX 9708057 A MX9708057 A MX 9708057A MX 9708057 A MX9708057 A MX 9708057A
- Authority
- MX
- Mexico
- Prior art keywords
- hiv
- thf
- aspartyl protease
- compounds
- relates
- Prior art date
Links
- 108010017640 Aspartic Acid Proteases Proteins 0.000 title abstract 2
- 102000004580 Aspartic Acid Proteases Human genes 0.000 title abstract 2
- 229940124530 sulfonamide Drugs 0.000 title abstract 2
- 150000003456 sulfonamides Chemical class 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 241000713772 Human immunodeficiency virus 1 Species 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 2
- 230000002401 inhibitory effect Effects 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 241000725303 Human immunodeficiency virus Species 0.000 abstract 1
- 108010016183 Human immunodeficiency virus 1 p16 protease Proteins 0.000 abstract 1
- 241000713340 Human immunodeficiency virus 2 Species 0.000 abstract 1
- 108010016191 Human immunodeficiency virus 2 p16 protease Proteins 0.000 abstract 1
- 239000003443 antiviral agent Substances 0.000 abstract 1
- 239000003696 aspartic proteinase inhibitor Substances 0.000 abstract 1
Landscapes
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invencion se relaciona con una clase de sulfonamidas que contienen THF, las cuales son inhibidoras de las aspartil proteasa. Esta invencion de relaciona con las composiciones farmacéuticas que comprenden estos compuestos. Los compuestos y composiciones farmacéuticas de esta invencion son particularmente muy adecuadas para inhibir la actividad de la proteasa VIH-1 y VIH-2 por consiguiente, pueden ser utilizados ventajosamente como agentes antivirales contra los virus VIH-1 VIH-2. Esta invencion también se relaciona con métodos para inhibir de la aspartilproteasa VIH utilizando los compuestos de esta invencion.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/US1996/005475 WO1996033184A1 (en) | 1995-04-19 | 1996-04-18 | Thf-containing sulfonamide inhibitors of aspartyl protease |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9708057A true MX9708057A (es) | 1998-01-31 |
Family
ID=39165679
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9708057A MX9708057A (es) | 1996-04-18 | 1996-04-18 | Sulfonamidas que contienen thf inhibidoras de la aspartilproteasa. |
Country Status (1)
| Country | Link |
|---|---|
| MX (1) | MX9708057A (es) |
-
1996
- 1996-04-18 MX MX9708057A patent/MX9708057A/es unknown
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