MX9504245A - Composicion para suministro de un farmaco. - Google Patents
Composicion para suministro de un farmaco.Info
- Publication number
- MX9504245A MX9504245A MX9504245A MX9504245A MX9504245A MX 9504245 A MX9504245 A MX 9504245A MX 9504245 A MX9504245 A MX 9504245A MX 9504245 A MX9504245 A MX 9504245A MX 9504245 A MX9504245 A MX 9504245A
- Authority
- MX
- Mexico
- Prior art keywords
- composition
- std
- bioadhesive
- sexually transmitted
- irritation
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S424/00—Drug, bio-affecting and body treating compositions
- Y10S424/14—Topical contraceptives and spermacides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Gynecology & Obstetrics (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Oncology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invencion proporciona una composicion y uso de una composicion que comprende una formulacion de polímero de ácido policarboxílico reticulado, bioadhesivo que permite el uso de cantidades relativamente bajas de agentes anti-STD, tales como N-9 para utilizarse para prevenir la infeccion por las STD sin provocar la irritacion al tejido genital que con frecuencia acompaña a las dosis elevadas de anti-STD. El polímero bioadhesivo mantiene e infeccioso durante un período de tiempo mucho mayor, permitiendo que una concentracion menor actue más tiempo sobre el agente infeccioso, cuando se compara con las aplicaciones comerciales actualmente disponibles que contienen N-9. Tal suministro permitirá una disminucion segura y sin irritacion en el riesgo de infeccion con las STD, incluyendo el VIH.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/319,495 US5667492A (en) | 1994-10-07 | 1994-10-07 | Use and composition of an anti-sexually transmitted diseases formulation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9504245A true MX9504245A (es) | 1997-01-31 |
Family
ID=23242477
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9504245A MX9504245A (es) | 1994-10-07 | 1995-10-06 | Composicion para suministro de un farmaco. |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US5667492A (es) |
| EP (1) | EP0784466B1 (es) |
| JP (1) | JPH10507178A (es) |
| KR (1) | KR970705976A (es) |
| AT (1) | ATE213623T1 (es) |
| AU (1) | AU704836B2 (es) |
| BR (1) | BR9509280A (es) |
| CA (1) | CA2201872A1 (es) |
| CO (1) | CO4480018A1 (es) |
| DE (1) | DE69525634T2 (es) |
| DK (1) | DK0784466T3 (es) |
| ES (1) | ES2173203T3 (es) |
| FI (1) | FI971440A0 (es) |
| HU (1) | HUT77527A (es) |
| IL (1) | IL115495A0 (es) |
| MA (1) | MA23687A1 (es) |
| MX (1) | MX9504245A (es) |
| NO (1) | NO971491L (es) |
| NZ (1) | NZ295947A (es) |
| PE (1) | PE46996A1 (es) |
| PT (1) | PT784466E (es) |
| RU (1) | RU2157184C2 (es) |
| WO (1) | WO1996010989A1 (es) |
| ZA (1) | ZA958434B (es) |
Families Citing this family (37)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6596777B1 (en) | 1997-05-29 | 2003-07-22 | Mcneil-Ppc, Inc. | Moisture containing compositions that are spreadable onto and adherable to biomembranes |
| US6440980B1 (en) * | 1996-09-17 | 2002-08-27 | Avanir Pharmaceuticals | Synergistic inhibition of viral replication by long-chain hydrocarbons and nucleoside analogs |
| US5942243A (en) * | 1996-11-12 | 1999-08-24 | Polytherapeutics, Inc. | Mucoadhesive compositions for administration of biologically active agents to animal tissue |
| WO1998051273A1 (en) * | 1997-05-12 | 1998-11-19 | Sage Pharmaceuticals, Inc. | Topical spray for burn treatment and anti-infection |
| US8765177B2 (en) * | 1997-09-12 | 2014-07-01 | Columbia Laboratories, Inc. | Bioadhesive progressive hydration tablets |
| DE69819748T2 (de) * | 1997-09-12 | 2004-09-30 | Columbia Laboratories (Bermuda) Ltd. | Arzneimittel zur behandlung von dysmenorrhöe und verfrühten wehen |
| US20040234606A1 (en) * | 1997-09-12 | 2004-11-25 | Levine Howard L. | Localized vaginal delivery without detrimental blood levels |
| EP1356806A1 (en) * | 1997-09-12 | 2003-10-29 | Columbia Laboratories (Bermuda) Limited | A pharmaceutical composition for treating dysmenorrhea and premature labor |
| JP2002518351A (ja) | 1998-06-19 | 2002-06-25 | オキシバイオ・インコーポレイテッド | 抗感染および避妊特性を有する医療装置 |
| AU4489399A (en) * | 1998-06-23 | 2000-01-10 | Notax Holding Gesellschaft M.B.H. | Use of nonoxynol-9 as lubricant and method for its production |
| US6159491A (en) * | 1999-02-12 | 2000-12-12 | Biovector Technologies, Inc. | Prolonged release bioadhesive vaginal gel dosage form |
| RU2310474C2 (ru) | 1999-10-05 | 2007-11-20 | Колумбия Лабораториз (Бермуда) Лимитед | Способ лечения эндометриоза или бесплодия или улучшение способности к воспроизведению потомства и фармацевтическая композиция для его осуществления |
| US6479045B2 (en) | 1999-12-22 | 2002-11-12 | Columbia Laboratories, Inc. | Vaginal pH buffering for preventing miscarriage and premature labor, by treating or preventing bacterial vaginosis |
| PL202918B1 (pl) | 2000-03-07 | 2009-08-31 | Rush Presbyterian St Luke | Przeciwbakteryjna i antykoncepcyjna kompozycja oraz jej zastosowanie |
| US7547433B2 (en) * | 2001-02-15 | 2009-06-16 | Access Pharmaceuticals, Inc. | Liquid formulations for the prevention and treatment of mucosal diseases and disorders |
| US7544348B2 (en) * | 2001-02-15 | 2009-06-09 | Access Pharmaceuticals, Inc. | Liquid formulations for the prevention and treatment of mucosal diseases and disorders |
| US20060073174A1 (en) * | 2001-08-16 | 2006-04-06 | Access Pharmaceuticals, Inc. | Adherent and erodible film to treat a moist surface of a body tissue |
| US6585997B2 (en) | 2001-08-16 | 2003-07-01 | Access Pharmaceuticals, Inc. | Mucoadhesive erodible drug delivery device for controlled administration of pharmaceuticals and other active compounds |
| JP2005519868A (ja) * | 2001-10-16 | 2005-07-07 | アバニール・ファーマシューティカルズ | n−ドコサノールによるウイルス阻害 |
| CN101327326A (zh) * | 2001-10-29 | 2008-12-24 | 哥伦比亚实验室(百慕大群岛)有限公司 | 阴道给药治疗骨盆痛和不孕症的抗节律障碍剂 |
| US7709026B2 (en) * | 2001-10-29 | 2010-05-04 | Columbia Laboratories, Inc. | Low concentration of peroxide for treating or preventing vaginal infections |
| US20030114394A1 (en) * | 2001-10-29 | 2003-06-19 | Levine Howard L. | Vaginally administered anti-dysrhythmic agents for treating pelvic pain |
| US20080182841A1 (en) * | 2001-10-29 | 2008-07-31 | Levine Howard L | Vaginally administered anti-dysrhythmic agents for treating pelvic pain |
| US8425892B2 (en) | 2001-10-29 | 2013-04-23 | Columbia Laboratories, Inc. | Extended, controlled-release pharmaceutical compositions using charged polymers |
| RU2200571C1 (ru) * | 2002-02-26 | 2003-03-20 | Быков Валерий Алексеевич | Комплекс природных соединений растительного происхождения, активный в отношении вирусных и других инфекций, передаваемых половым путем |
| RU2200570C1 (ru) * | 2002-02-26 | 2003-03-20 | Быков Валерий Алексеевич | Комплекс природных соединений растительного происхождения, обладающий сперматоцидным эффектом и активностью в отношении инфекций, передаваемых половым путем |
| RU2200572C1 (ru) * | 2002-02-26 | 2003-03-20 | Быков Валерий Алексеевич | Комплекс природных соединений растительного происхождения, обладающий противоинфекционным действием в отношении инфекций, передаваемых половым путем |
| NZ541902A (en) * | 2003-02-07 | 2008-12-24 | Janssen Pharmaceutica Nv | Pyrimidine derivatives for the prevention of HIV infection |
| ES2237298B1 (es) * | 2003-07-16 | 2006-11-01 | Italfarmaco, S.A. | Formulaciones mucoadhesivas semisolidas. |
| ITMI20031640A1 (it) | 2003-08-08 | 2005-02-09 | Mipharm S P A | Base per gel bioadesivi. |
| US12011423B2 (en) | 2007-11-06 | 2024-06-18 | Foraviset Ltd. | S-alkylisothiouronium derivatives for treating uterine hypercontractility disorders |
| ES2344673B1 (es) | 2008-08-07 | 2011-05-03 | Italfarmaco, S.A. | Uso de estriol en la preparacion de una formulacion farmaceutica parael tratamiento de atrofia vaginal en mujeres con riesgo de potologiatumoral. |
| ES2344675B1 (es) | 2008-12-19 | 2011-04-28 | Italfarmaco, S.A. | Uso de estriol en la preparacion de una formulacion farrmaceutica para el tratamiento de atrofia vaginal en mujeres con riesgo de patologiacardiovascular. |
| HK1208809A1 (en) * | 2012-06-13 | 2016-03-18 | 伊沃菲姆股份有限公司 | Compositions and methods for enhancing the efficacy of contraceptive microbicides |
| KR102407408B1 (ko) | 2013-12-19 | 2022-06-10 | 에보펨 인코포레이티드 | 알긴산계 항균성 화합물을 사용하는 염증 및 질병을 억제하기 위한 조성물 및 방법 |
| CA2897038C (en) * | 2014-07-14 | 2016-10-04 | Novicol International Holding Inc. | Microbicidal composition comprising an octoxynol and a quinolizidine alkaloid compound or a source thereof |
| EP3522879A4 (en) | 2016-10-04 | 2020-06-03 | Evofem, Inc. | Method of treatment and prevention of bacterial vaginosis |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL265428A (es) * | 1960-06-06 | |||
| US4286593A (en) * | 1980-05-05 | 1981-09-01 | Place Virgil A | Vaginal contraceptive shield |
| EP0077063B1 (en) * | 1981-10-13 | 1988-03-16 | Exovir, Inc. | Interferon-containing compositions and the use of these compositions in the treatment of herpetic infections, pre-malignant skin lesions, skin malignancies and psoriasis |
| WO1985002092A1 (en) * | 1983-11-14 | 1985-05-23 | Bio-Mimetics Inc. | Bioadhesive compositions and methods of treatment therewith |
| US4983393A (en) * | 1987-07-21 | 1991-01-08 | Maximed Corporation | Intra-vaginal device and method for sustained drug release |
| NO178843C (no) * | 1988-07-11 | 1996-06-19 | Sspl Sa Safe Sex Prod Licens | Fremgangsmåte for fremstilling av et farmasöytisk preparat for å forhindre seksuelt overförbare sykdommer |
| US5000749A (en) * | 1988-10-13 | 1991-03-19 | Leveen Harry H | Iodine contraceptive sponge |
| BR9007807A (pt) * | 1989-10-31 | 1992-09-29 | Columbia Lab Inc | Composicao e metodo para umedecimento de tecido |
| ES2050096T3 (es) * | 1989-10-31 | 1995-01-16 | Columbia Lab Inc | Composicion humidificante del tejido vaginal. |
| DK0429156T3 (da) * | 1989-10-31 | 1995-01-16 | Columbia Lab Inc | Fremgangsmåde til fugtiggørelse af væv og præparat hertil |
| US5380523A (en) * | 1993-08-17 | 1995-01-10 | University Of Kentucky Research Foundation | High energy coprecipitate of nonoxynol oligomer, PVP and iodine having contraceptive and potent anti-HIV properties |
-
1994
- 1994-10-07 US US08/319,495 patent/US5667492A/en not_active Expired - Fee Related
-
1995
- 1995-10-02 IL IL11549595A patent/IL115495A0/xx unknown
- 1995-10-06 PT PT95937526T patent/PT784466E/pt unknown
- 1995-10-06 MA MA24032A patent/MA23687A1/fr unknown
- 1995-10-06 KR KR1019970702233A patent/KR970705976A/ko not_active Ceased
- 1995-10-06 HU HU9701492A patent/HUT77527A/hu unknown
- 1995-10-06 BR BR9509280A patent/BR9509280A/pt not_active Application Discontinuation
- 1995-10-06 WO PCT/US1995/013424 patent/WO1996010989A1/en not_active Ceased
- 1995-10-06 EP EP95937526A patent/EP0784466B1/en not_active Expired - Lifetime
- 1995-10-06 AU AU39612/95A patent/AU704836B2/en not_active Ceased
- 1995-10-06 ES ES95937526T patent/ES2173203T3/es not_active Expired - Lifetime
- 1995-10-06 DE DE69525634T patent/DE69525634T2/de not_active Expired - Fee Related
- 1995-10-06 AT AT95937526T patent/ATE213623T1/de not_active IP Right Cessation
- 1995-10-06 MX MX9504245A patent/MX9504245A/es unknown
- 1995-10-06 CA CA002201872A patent/CA2201872A1/en not_active Abandoned
- 1995-10-06 FI FI971440A patent/FI971440A0/fi unknown
- 1995-10-06 CO CO95046725A patent/CO4480018A1/es unknown
- 1995-10-06 NZ NZ295947A patent/NZ295947A/xx unknown
- 1995-10-06 RU RU97107333/14A patent/RU2157184C2/ru active
- 1995-10-06 DK DK95937526T patent/DK0784466T3/da active
- 1995-10-06 PE PE1995280984A patent/PE46996A1/es not_active Application Discontinuation
- 1995-10-06 JP JP8512743A patent/JPH10507178A/ja active Pending
- 1995-10-06 ZA ZA958434A patent/ZA958434B/xx unknown
-
1997
- 1997-04-02 NO NO971491A patent/NO971491L/no unknown
- 1997-06-06 US US08/870,653 patent/US20010006667A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR970705976A (ko) | 1997-11-03 |
| CA2201872A1 (en) | 1996-04-18 |
| EP0784466A1 (en) | 1997-07-23 |
| FI971440L (fi) | 1997-04-07 |
| ATE213623T1 (de) | 2002-03-15 |
| MA23687A1 (fr) | 1996-07-01 |
| US20010006667A1 (en) | 2001-07-05 |
| IL115495A0 (en) | 1996-01-19 |
| US5667492A (en) | 1997-09-16 |
| FI971440A7 (fi) | 1997-04-07 |
| PE46996A1 (es) | 1996-11-23 |
| CO4480018A1 (es) | 1997-07-09 |
| WO1996010989A1 (en) | 1996-04-18 |
| JPH10507178A (ja) | 1998-07-14 |
| ZA958434B (en) | 1996-05-08 |
| NO971491D0 (no) | 1997-04-02 |
| BR9509280A (pt) | 1997-11-18 |
| EP0784466B1 (en) | 2002-02-27 |
| NZ295947A (en) | 1999-02-25 |
| ES2173203T3 (es) | 2002-10-16 |
| AU3961295A (en) | 1996-05-02 |
| HUT77527A (hu) | 1998-05-28 |
| DE69525634T2 (de) | 2002-08-29 |
| DE69525634D1 (de) | 2002-04-04 |
| PT784466E (pt) | 2002-06-28 |
| NO971491L (no) | 1997-06-09 |
| FI971440A0 (fi) | 1997-04-07 |
| RU2157184C2 (ru) | 2000-10-10 |
| AU704836B2 (en) | 1999-05-06 |
| DK0784466T3 (da) | 2002-04-22 |
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