MX9308188A - Glucomanano de konjac facilmente disponible, como un excipiente de liberacion sostenida. - Google Patents
Glucomanano de konjac facilmente disponible, como un excipiente de liberacion sostenida.Info
- Publication number
- MX9308188A MX9308188A MX9308188A MX9308188A MX9308188A MX 9308188 A MX9308188 A MX 9308188A MX 9308188 A MX9308188 A MX 9308188A MX 9308188 A MX9308188 A MX 9308188A MX 9308188 A MX9308188 A MX 9308188A
- Authority
- MX
- Mexico
- Prior art keywords
- konjac
- excipient
- glucomanane
- easily available
- sustained liberation
- Prior art date
Links
- 241001312219 Amorphophallus konjac Species 0.000 title abstract 5
- 235000001206 Amorphophallus rivieri Nutrition 0.000 title abstract 5
- 229920002752 Konjac Polymers 0.000 title abstract 5
- 235000010485 konjac Nutrition 0.000 title abstract 5
- 239000000252 konjac Substances 0.000 title abstract 5
- 239000000546 pharmaceutical excipient Substances 0.000 title abstract 3
- 230000002459 sustained effect Effects 0.000 title 1
- LUEWUZLMQUOBSB-FSKGGBMCSA-N (2s,3s,4s,5s,6r)-2-[(2r,3s,4r,5r,6s)-6-[(2r,3s,4r,5s,6s)-4,5-dihydroxy-2-(hydroxymethyl)-6-[(2r,4r,5s,6r)-4,5,6-trihydroxy-2-(hydroxymethyl)oxan-3-yl]oxyoxan-3-yl]oxy-4,5-dihydroxy-2-(hydroxymethyl)oxan-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol Chemical compound O[C@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]1O[C@@H]1[C@@H](CO)O[C@@H](O[C@@H]2[C@H](O[C@@H](OC3[C@H](O[C@@H](O)[C@@H](O)[C@H]3O)CO)[C@@H](O)[C@H]2O)CO)[C@H](O)[C@H]1O LUEWUZLMQUOBSB-FSKGGBMCSA-N 0.000 abstract 1
- 229920002581 Glucomannan Polymers 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 229940046240 glucomannan Drugs 0.000 abstract 1
- 230000000887 hydrating effect Effects 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000000843 powder Substances 0.000 abstract 1
- 239000007909 solid dosage form Substances 0.000 abstract 1
- 238000013268 sustained release Methods 0.000 abstract 1
- 239000012730 sustained-release form Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
Abstract
Una forma de dosis sólida, tal como una tableta farmacéutica, que contiene un glucomanano de konjac que se hidrata rápidamente, como excipiente de liberación sostenida, tal como konjac clarificado, konjac triturado criogénicamente y konjac plastificado. El método para elaborar las tabletas mediante la compresión del excipiente y el ingrediente farmacéuticamente activo, como polvos secos.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US99833592A | 1992-12-30 | 1992-12-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9308188A true MX9308188A (es) | 1994-06-30 |
Family
ID=25545069
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9308188A MX9308188A (es) | 1992-12-30 | 1993-12-17 | Glucomanano de konjac facilmente disponible, como un excipiente de liberacion sostenida. |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US5486364A (es) |
| EP (1) | EP0676967A4 (es) |
| JP (1) | JP2628231B2 (es) |
| AU (1) | AU5745394A (es) |
| CA (1) | CA2152795C (es) |
| MX (1) | MX9308188A (es) |
| WO (1) | WO1994015643A1 (es) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1996016639A1 (en) * | 1994-12-01 | 1996-06-06 | Cibus Pharmaceutical, Inc. | Nsaid delivery employing a powdered hydrocolloid gum obtainable from higher plants |
| AU709413B2 (en) * | 1994-12-01 | 1999-08-26 | Amarin Development Ab | Sustained-release drug delivery employing a powdered hydrocolloid gum obtainable from higher plants |
| FR2729857B1 (fr) | 1995-01-27 | 1997-04-04 | Rhone Poulenc Chimie | Compositions pharmaceutiques sous forme de comprimes a liberation prolongee a base de granules en polysaccharides de haut poids moleculaire |
| US5811388A (en) * | 1995-06-07 | 1998-09-22 | Cibus Pharmaceutical, Inc. | Delivery of drugs to the lower GI tract |
| US6893664B1 (en) * | 1996-06-17 | 2005-05-17 | Powderject Research Limited | Particle delivery techniques |
| GB9613470D0 (en) | 1996-06-27 | 1996-08-28 | Ciba Geigy Ag | Small solid oral dosage form |
| JPH10114682A (ja) * | 1996-10-11 | 1998-05-06 | Shimizu Kagaku Kk | グルコマンナン配合持効性内服用薬剤 |
| US6537318B1 (en) * | 1998-04-06 | 2003-03-25 | Konjac Technologies, Llc | Use of glucomannan hydrocolloid as filler material in prostheses |
| US6497157B1 (en) * | 1999-11-29 | 2002-12-24 | Distek, Inc. | Intrinsic dissolution apparatus with stationary sample holder |
| US6955821B2 (en) | 2000-04-28 | 2005-10-18 | Adams Laboratories, Inc. | Sustained release formulations of guaifenesin and additional drug ingredients |
| US7985420B2 (en) * | 2000-04-28 | 2011-07-26 | Reckitt Benckiser Inc. | Sustained release of guaifenesin combination drugs |
| US7838032B2 (en) * | 2000-04-28 | 2010-11-23 | Reckitt Benckiser Inc. | Sustained release of guaifenesin |
| US8012504B2 (en) * | 2000-04-28 | 2011-09-06 | Reckitt Benckiser Inc. | Sustained release of guaifenesin combination drugs |
| US7326404B2 (en) * | 2000-05-31 | 2008-02-05 | Vuksan Holdings Inc. | Konjac-mannan and ginseng compositions and methods and uses thereof |
| SE0003125D0 (sv) * | 2000-09-05 | 2000-09-05 | Astrazeneca Ab | Modified polymers |
| CN1325050C (zh) * | 2002-04-26 | 2007-07-11 | 霍夫曼-拉罗奇有限公司 | 包含脂肪酶抑制剂和葡甘露聚糖的药物组合物 |
| DE10247910A1 (de) * | 2002-10-14 | 2004-04-22 | Beisel, Günther | Mittel zur Erzeugung eines langanhaltenden Sättigungseffektes |
| US8003152B1 (en) * | 2006-03-30 | 2011-08-23 | Vitalico LLC | Fast-hydratable konjac composition |
| SI2178870T1 (sl) | 2007-08-17 | 2018-11-30 | Lg Chem, Ltd. | Indolne in indazolne spojine kot inhibitor celične nekroze |
| CN101780400B (zh) * | 2009-01-21 | 2011-11-09 | 西南科技大学 | 热塑性葡甘聚糖阳离子吸附材料及其制备方法 |
| JP5903250B2 (ja) * | 2011-11-16 | 2016-04-13 | 清水化学株式会社 | 徐放性組成物 |
| CA2791206A1 (en) | 2012-09-28 | 2014-03-28 | Pharmascience Inc. | Abuse deterrent pharmaceutical formulation |
| US9114091B2 (en) | 2013-07-05 | 2015-08-25 | Shimizu Chemical Corporation | Sustained release solid dosage preparations |
| EP2826464A1 (en) * | 2013-07-19 | 2015-01-21 | Shimizu Chemical Corporation | Sustained release solid dosage preparations |
| CA2953396C (en) | 2014-07-03 | 2022-11-08 | Mallinckrodt Llc | Abuse deterrent immediate release formulations comprising non-cellulose polysaccharides |
| GB201506755D0 (en) | 2015-04-21 | 2015-06-03 | Reckitt Benckiser Llc | Novel pharmaceutical formulation |
| CA3001337C (en) | 2015-10-09 | 2023-12-12 | Reckitt Benckiser Llc | Pharmaceutical formulation |
| WO2018195267A1 (en) | 2017-04-20 | 2018-10-25 | Dow Global Technologies Llc | Fast hydratable konjac flour |
| WO2018195271A1 (en) * | 2017-04-20 | 2018-10-25 | Dow Global Technologies Llc | Fast hydratable konjac flour |
| WO2020023396A1 (en) | 2018-07-23 | 2020-01-30 | Nutragenom, Llc | Composition and methods for generating and sustaining molecular hydrogen (h2) in aqueous systems |
| WO2020068510A1 (en) | 2018-09-25 | 2020-04-02 | SpecGx LLC | Abuse deterrent immediate release capsule dosage forms |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR901111A (fr) * | 1943-08-31 | 1945-07-18 | Perfectionnement aux dispositifs de réglage de terrage des charruesbascules | |
| US3928322A (en) * | 1970-12-30 | 1975-12-23 | Shimizu Manzo Shoten Kk | Konjac mannan |
| JPS57185216A (en) * | 1981-05-11 | 1982-11-15 | Chiyoda Yakuhin Kk | Preparation of glucomannan tablet |
| FR2523446A1 (fr) * | 1982-03-19 | 1983-09-23 | Dietlin Francois | Nouveau procede d'obtention de formes pharmaceutiques a liberation programmee |
| FR2531339A1 (fr) * | 1982-08-04 | 1984-02-10 | Dietlin Francois | Nouveau procede d'obtention de formes pharmaceutiques a liberation programmee |
| JPS60219238A (ja) * | 1984-04-14 | 1985-11-01 | Hayashibara Biochem Lab Inc | 徐崩性プルラン含有成形物とその製法 |
| BE901111A (fr) * | 1984-11-22 | 1985-03-15 | Benfar Representee Par Vanderl | Composition pharmaceutiques a liberation prolongee, leur procede de preparation et leur utilisation. |
| GB8431699D0 (en) * | 1984-12-14 | 1985-01-30 | Mars G B Ltd | Gel system |
| GB8601204D0 (en) * | 1986-01-18 | 1986-02-19 | Boots Co Plc | Therapeutic agents |
| GB8616669D0 (en) * | 1986-07-09 | 1986-08-13 | Merk Sharpe & Dohme Ltd | Pharmaceutical compositions |
| GB8710704D0 (en) * | 1987-05-06 | 1987-06-10 | Mars G B Ltd | Edible gels |
| US4994276A (en) * | 1988-09-19 | 1991-02-19 | Edward Mendell Co., Inc. | Directly compressible sustained release excipient |
| US5096714A (en) * | 1988-06-28 | 1992-03-17 | Hauser-Kuhrts, Inc. | Prolonged release drug tablet formulations |
| JPH0443819A (ja) * | 1990-06-09 | 1992-02-13 | Yamaha Motor Co Ltd | 2サイクルエンジンの吸気用ロータリバルブ装置 |
-
1993
- 1993-12-09 EP EP94903550A patent/EP0676967A4/en not_active Withdrawn
- 1993-12-09 CA CA002152795A patent/CA2152795C/en not_active Expired - Fee Related
- 1993-12-09 JP JP6515521A patent/JP2628231B2/ja not_active Expired - Lifetime
- 1993-12-09 WO PCT/US1993/011970 patent/WO1994015643A1/en not_active Ceased
- 1993-12-09 AU AU57453/94A patent/AU5745394A/en not_active Abandoned
- 1993-12-17 MX MX9308188A patent/MX9308188A/es not_active Application Discontinuation
-
1994
- 1994-08-15 US US08/290,457 patent/US5486364A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2628231B2 (ja) | 1997-07-09 |
| US5486364A (en) | 1996-01-23 |
| EP0676967A4 (en) | 1996-10-02 |
| JPH08504214A (ja) | 1996-05-07 |
| CA2152795A1 (en) | 1994-07-21 |
| WO1994015643A1 (en) | 1994-07-21 |
| CA2152795C (en) | 1999-02-16 |
| EP0676967A1 (en) | 1995-10-18 |
| AU5745394A (en) | 1994-08-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |