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MX9307810A - Heterociclicos no aromaticos sustituidos con aminometileno. - Google Patents

Heterociclicos no aromaticos sustituidos con aminometileno.

Info

Publication number
MX9307810A
MX9307810A MX9307810A MX9307810A MX9307810A MX 9307810 A MX9307810 A MX 9307810A MX 9307810 A MX9307810 A MX 9307810A MX 9307810 A MX9307810 A MX 9307810A MX 9307810 A MX9307810 A MX 9307810A
Authority
MX
Mexico
Prior art keywords
aminomethylene
aromatic hetero
hetero cycles
substituted
new
Prior art date
Application number
MX9307810A
Other languages
English (en)
Inventor
Harry R Howard
Brian T O'neill
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX9307810A publication Critical patent/MX9307810A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Anesthesiology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

La presente invención se refiere a nuevos heterociclos no aromáticos sustituidos con aminometileno y, más específicamente, a compuestos correspondientes a la fórmula Ia, Ib, donde W, R1, R2, R3, A, X', Y' y Z' se definen como en la memoria descriptiva, y se refiere además a productos intermedios utilizados en la síntesis de tales compuestos. Los nuevos compuestos correspondientes a las fórmulas Ia y Ib resultan útiles en el tratamiento de enfermedades inflamatorias y trastornos del sistema nervioso central, además de otras enfermedades.
MX9307810A 1992-12-10 1993-12-09 Heterociclicos no aromaticos sustituidos con aminometileno. MX9307810A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US98865392A 1992-12-10 1992-12-10

Publications (1)

Publication Number Publication Date
MX9307810A true MX9307810A (es) 1994-07-29

Family

ID=25534364

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9307810A MX9307810A (es) 1992-12-10 1993-12-09 Heterociclicos no aromaticos sustituidos con aminometileno.

Country Status (15)

Country Link
EP (2) EP0675886B1 (es)
JP (2) JP2722279B2 (es)
CN (1) CN1092771A (es)
AT (1) ATE194340T1 (es)
AU (1) AU5169693A (es)
CA (1) CA2150123C (es)
DE (1) DE69328975T2 (es)
DK (1) DK0675886T3 (es)
ES (1) ES2147759T3 (es)
FI (1) FI935529L (es)
GR (1) GR3034329T3 (es)
IL (1) IL107843A0 (es)
MX (1) MX9307810A (es)
PT (1) PT675886E (es)
WO (1) WO1994013663A1 (es)

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Also Published As

Publication number Publication date
GR3034329T3 (en) 2000-12-29
FI935529A7 (fi) 1994-06-11
CN1092771A (zh) 1994-09-28
JPH1095780A (ja) 1998-04-14
AU5169693A (en) 1994-07-04
ES2147759T3 (es) 2000-10-01
DE69328975D1 (de) 2000-08-10
FI935529A0 (fi) 1993-12-09
WO1994013663A1 (en) 1994-06-23
PT675886E (pt) 2000-12-29
EP0675886B1 (en) 2000-07-05
JP3165401B2 (ja) 2001-05-14
IL107843A0 (en) 1994-04-12
EP0675886A1 (en) 1995-10-11
DE69328975T2 (de) 2000-11-09
CA2150123A1 (en) 1994-06-23
ATE194340T1 (de) 2000-07-15
FI935529L (fi) 1994-06-11
DK0675886T3 (da) 2000-09-18
JPH07509490A (ja) 1995-10-19
JP2722279B2 (ja) 1998-03-04
EP0806423A1 (en) 1997-11-12
CA2150123C (en) 2004-12-07

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