MX9306178A - Bencimidazoles medicamentos que contienen estos compuestos yprocedimientos para su preparacion. - Google Patents
Bencimidazoles medicamentos que contienen estos compuestos yprocedimientos para su preparacion.Info
- Publication number
- MX9306178A MX9306178A MX9306178A MX9306178A MX9306178A MX 9306178 A MX9306178 A MX 9306178A MX 9306178 A MX9306178 A MX 9306178A MX 9306178 A MX9306178 A MX 9306178A MX 9306178 A MX9306178 A MX 9306178A
- Authority
- MX
- Mexico
- Prior art keywords
- compounds
- procedures
- bencimidazoles
- preparation
- medicines containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/08—Radicals containing only hydrogen and carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
El invento concierne a bencimidazoles de la fórmula general (I): en que Raa Rd están definidos como en la reivindicación 1, sus mezclas de isómeros1.3 y sus sales que presentan valiosas propiedades, a medicamentos quecontienen estos compuestos y a su empleo así como a procedimientos para supreparación. Los nuevos compuestos representan en particular antagonistasde angiotensina.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4233590A DE4233590A1 (de) | 1992-10-06 | 1992-10-06 | Benzimidazole, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung |
| DE4315349A DE4315349A1 (de) | 1992-10-06 | 1993-05-08 | Benzimidazole, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9306178A true MX9306178A (es) | 1995-01-31 |
Family
ID=25919224
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9306178A MX9306178A (es) | 1992-10-06 | 1993-10-05 | Bencimidazoles medicamentos que contienen estos compuestos yprocedimientos para su preparacion. |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US5521177A (es) |
| EP (1) | EP0591891A3 (es) |
| JP (1) | JPH06211807A (es) |
| KR (1) | KR940009160A (es) |
| CN (1) | CN1088202A (es) |
| CA (1) | CA2107604A1 (es) |
| CZ (1) | CZ207293A3 (es) |
| DE (1) | DE4315349A1 (es) |
| FI (1) | FI934343L (es) |
| HU (1) | HUT65300A (es) |
| IL (1) | IL107175A0 (es) |
| MX (1) | MX9306178A (es) |
| NO (1) | NO933558L (es) |
| NZ (1) | NZ248850A (es) |
| PL (1) | PL300585A1 (es) |
| SK (1) | SK106693A3 (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5565454A (en) * | 1995-05-31 | 1996-10-15 | Ergo Science, Incorporated | Method for preventing intervention-associated stenosis and other symptoms associated with stenosis of blood vessels following non-bypass, invasive interventions |
| EP1813286A3 (en) * | 1996-04-05 | 2008-04-16 | Takeda Pharmaceutical Company Limited | Pharmaceutical composition containing a compound having angiotensin II antagonistic activity in combination with another compound |
| US5955548A (en) * | 1997-05-07 | 1999-09-21 | Novo Nordisk A/S | Substituted 3, 3-diamino-2-propenenitriles, their preparation and use |
| CN1259119A (zh) * | 1997-05-07 | 2000-07-05 | 诺沃挪第克公司 | 取代的3,3-二氨基-2-丙烯腈,它们的制备及用途 |
| US6916813B2 (en) * | 2001-12-10 | 2005-07-12 | Bristol-Myers Squibb Co. | (1-phenyl-2-heteoaryl)ethyl-guanidine compounds as inhibitors of mitochondrial F1F0 ATP hydrolase |
| JPWO2005011736A1 (ja) * | 2003-07-30 | 2006-09-14 | 株式会社 東北テクノアーチ | アルツハイマー病の予防および/または治療剤 |
| CN101448778A (zh) * | 2006-05-26 | 2009-06-03 | 艾博特公司 | Polo样激酶的抑制剂 |
| WO2025207620A1 (en) * | 2024-03-27 | 2025-10-02 | Alterome Therapeutics, Inc. | Akt1 modulators |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0461039B1 (fr) * | 1990-06-08 | 1998-09-16 | Hoechst Marion Roussel | Dérivés du benzimidazole, leur procédé de préparation, les intermédiaires obtenus, leur application à titre de médicaments et les compositions pharmaceutiques les renfermant |
| SI9210098B (sl) * | 1991-02-06 | 2000-06-30 | Dr. Karl Thomae | Benzimidazoli, zdravila, ki te spojine vsebujejo, in postopek za njihovo pripravo |
-
1993
- 1993-05-08 DE DE4315349A patent/DE4315349A1/de not_active Ceased
- 1993-10-04 US US08/132,065 patent/US5521177A/en not_active Expired - Fee Related
- 1993-10-04 SK SK1066-93A patent/SK106693A3/sk unknown
- 1993-10-04 IL IL107175A patent/IL107175A0/xx unknown
- 1993-10-04 FI FI934343A patent/FI934343L/fi not_active Application Discontinuation
- 1993-10-04 CA CA002107604A patent/CA2107604A1/en not_active Abandoned
- 1993-10-04 EP EP19930115991 patent/EP0591891A3/de not_active Withdrawn
- 1993-10-04 NZ NZ248850A patent/NZ248850A/en unknown
- 1993-10-05 KR KR1019930020472A patent/KR940009160A/ko not_active Withdrawn
- 1993-10-05 NO NO933558A patent/NO933558L/no unknown
- 1993-10-05 CZ CZ932072A patent/CZ207293A3/cs unknown
- 1993-10-05 MX MX9306178A patent/MX9306178A/es unknown
- 1993-10-05 HU HU9302813A patent/HUT65300A/hu unknown
- 1993-10-05 PL PL93300585A patent/PL300585A1/xx unknown
- 1993-10-05 JP JP5248384A patent/JPH06211807A/ja active Pending
- 1993-10-06 CN CN93118625A patent/CN1088202A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| KR940009160A (ko) | 1994-05-20 |
| FI934343A0 (fi) | 1993-10-04 |
| NO933558L (no) | 1994-04-07 |
| FI934343A7 (fi) | 1994-04-07 |
| HUT65300A (en) | 1994-05-02 |
| JPH06211807A (ja) | 1994-08-02 |
| CA2107604A1 (en) | 1994-04-07 |
| EP0591891A2 (de) | 1994-04-13 |
| PL300585A1 (en) | 1994-05-16 |
| CN1088202A (zh) | 1994-06-22 |
| HU9302813D0 (en) | 1993-12-28 |
| NO933558D0 (no) | 1993-10-05 |
| US5521177A (en) | 1996-05-28 |
| NZ248850A (en) | 1995-12-21 |
| SK106693A3 (en) | 1994-08-10 |
| DE4315349A1 (de) | 1994-11-10 |
| IL107175A0 (en) | 1994-01-25 |
| FI934343L (fi) | 1994-04-07 |
| CZ207293A3 (en) | 1994-04-13 |
| EP0591891A3 (en) | 1994-07-20 |
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