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MX9300412A - Derivados de 1h-bencimidazol sustituidos con pirroloimidazolilo e imadazopiridinilo - Google Patents

Derivados de 1h-bencimidazol sustituidos con pirroloimidazolilo e imadazopiridinilo

Info

Publication number
MX9300412A
MX9300412A MX9300412A MX9300412A MX9300412A MX 9300412 A MX9300412 A MX 9300412A MX 9300412 A MX9300412 A MX 9300412A MX 9300412 A MX9300412 A MX 9300412A MX 9300412 A MX9300412 A MX 9300412A
Authority
MX
Mexico
Prior art keywords
substituted
pyroloimidazolyl
imadazopyridinyl
bencimidazole
derivatives
Prior art date
Application number
MX9300412A
Other languages
English (en)
Inventor
Marcel August Constant Janssen
Alfons Herman
Margaretha R Eddy
Jean Edgard Freyne
Michael Nicholas Greco
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of MX9300412A publication Critical patent/MX9300412A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02EREDUCTION OF GREENHOUSE GAS [GHG] EMISSIONS, RELATED TO ENERGY GENERATION, TRANSMISSION OR DISTRIBUTION
    • Y02E50/00Technologies for the production of fuel of non-fossil origin
    • Y02E50/10Biofuels, e.g. bio-diesel

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

Derivados de 1H-bencimidazol sustituidos con pirroloimidazolilo e imidazopiridinilo, que tienen la fórmula (I). Composiciones que se contienen dichos compuestos de la fórmula (I), preparaciones de dichos compuestos y composiciones y su uso para tratar mamíferos que sufren de desórdenes provocados por la hormona sexual.
MX9300412A 1992-01-27 1993-01-26 Derivados de 1h-bencimidazol sustituidos con pirroloimidazolilo e imadazopiridinilo MX9300412A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US82656492A 1992-01-27 1992-01-27

Publications (1)

Publication Number Publication Date
MX9300412A true MX9300412A (es) 1993-07-01

Family

ID=25246906

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9300412A MX9300412A (es) 1992-01-27 1993-01-26 Derivados de 1h-bencimidazol sustituidos con pirroloimidazolilo e imadazopiridinilo

Country Status (20)

Country Link
EP (1) EP0625155B1 (es)
JP (1) JPH07503242A (es)
KR (1) KR100263412B1 (es)
CN (2) CN1036007C (es)
AT (1) ATE203992T1 (es)
AU (1) AU668708B2 (es)
CA (1) CA2127689A1 (es)
DE (1) DE69330557T2 (es)
DK (1) DK0625155T3 (es)
ES (1) ES2161714T3 (es)
FI (1) FI106462B (es)
GR (1) GR3036545T3 (es)
HU (1) HU222117B1 (es)
IL (1) IL104498A (es)
MX (1) MX9300412A (es)
NO (1) NO301118B1 (es)
PT (1) PT625155E (es)
TW (1) TW221690B (es)
WO (1) WO1993015079A1 (es)
ZA (1) ZA93561B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6015796A (en) * 1995-06-14 1997-01-15 Yamanouchi Pharmaceutical Co., Ltd. Fused imidazole derivatives and medicinal composition thereof
CA2429133C (en) 2000-11-17 2009-08-18 Takeda Chemical Industries, Ltd. Novel imidazole derivatives, production method thereof and use thereof
WO2005000795A2 (en) * 2003-06-10 2005-01-06 Smithkline Beecham Corporation Aniline derivatived androgen-, glucocorticoid-, mineralcorticoid- and progesterone- receptor modulators
CN100496525C (zh) * 2004-04-02 2009-06-10 李嫦梅 从洋蓟根、茎、叶中提取活性成份的方法及其应用
AR049125A1 (es) * 2004-05-28 2006-06-28 Speedel Experimenta Ag Heterociclos biciclicos nitrogenados inhibidores de la aromatasa.
WO2005118541A2 (en) * 2004-05-28 2005-12-15 Speedel Experimenta Ag Heterocyclic compounds and their use as aldosterone synthase inhibitors
CA2568165A1 (en) * 2004-05-28 2005-12-15 Speedel Experimenta Ag Heterocyclic compounds and their use as aldosterone synthase inhibitors
AR049667A1 (es) * 2004-07-09 2006-08-23 Speedel Experimenta Ag Heterociclos condensados conteniendo n como inhibidores de aromatasa y procedimiento para prepararlos
US8828429B2 (en) 2005-03-03 2014-09-09 Takeda Pharmaceutical Company Limited Release-control composition
GT200600381A (es) * 2005-08-25 2007-03-28 Compuestos organicos
CN101250559B (zh) * 2008-03-14 2010-12-29 厦门大学 一种利用天然抗菌剂防治酒精发酵染菌的方法
JP5749410B2 (ja) 2012-01-17 2015-07-15 ノバルティス アーゲー ジヒドロピロロ[1,2−c]イミダゾリルアルドステロンシンターゼまたはアロマターゼ阻害薬の新たな形態および塩
CN106665636A (zh) * 2015-11-07 2017-05-17 郑州明德生物科技有限公司 采用月桂酰精氨酸乙酯抑制酒精发酵污染微生物的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4426450A (en) * 1981-08-24 1984-01-17 Fermentec Corporation Fermentation process and apparatus
GB8820730D0 (en) * 1988-09-02 1988-10-05 Erba Carlo Spa Substituted 5 6 7 8-tetrahydroimidazo/1.5-a/pyridines & process for their preparation
CA2026792A1 (en) * 1989-11-01 1991-05-02 Michael N. Greco (6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-5-yl)- and (5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-5-yl) substituted 1h-benzotriazole derivatives
US5059431A (en) * 1990-12-07 1991-10-22 State Of Oregon Acting By And Through The State Board Of Higher Education On Behalf Of Oregon State University Process for deacidifying wine

Also Published As

Publication number Publication date
ATE203992T1 (de) 2001-08-15
PT625155E (pt) 2002-01-30
FI943511A7 (fi) 1994-07-26
HUT70853A (en) 1995-11-28
AU668708B2 (en) 1996-05-16
DE69330557T2 (de) 2002-06-20
DK0625155T3 (da) 2001-11-12
JPH07503242A (ja) 1995-04-06
FI943511A0 (fi) 1994-07-26
AU3450593A (en) 1993-09-01
ZA93561B (en) 1994-07-26
NO942748L (no) 1994-09-26
NO942748D0 (no) 1994-07-22
CN1036007C (zh) 1997-10-01
FI106462B (fi) 2001-02-15
CA2127689A1 (en) 1993-08-05
KR100263412B1 (ko) 2000-08-01
IL104498A (en) 1996-07-23
IL104498A0 (en) 1993-05-13
HU222117B1 (hu) 2003-04-28
CN1049687C (zh) 2000-02-23
ES2161714T3 (es) 2001-12-16
GR3036545T3 (en) 2001-12-31
HU9402208D0 (en) 1994-09-28
DE69330557D1 (de) 2001-09-13
WO1993015079A1 (en) 1993-08-05
CN1074907A (zh) 1993-08-04
EP0625155A1 (en) 1994-11-23
CN1095415A (zh) 1994-11-23
EP0625155B1 (en) 2001-08-08
TW221690B (es) 1994-03-11
NO301118B1 (no) 1997-09-15

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