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MX9204342A - Indoles. - Google Patents

Indoles.

Info

Publication number
MX9204342A
MX9204342A MX9204342A MX9204342A MX9204342A MX 9204342 A MX9204342 A MX 9204342A MX 9204342 A MX9204342 A MX 9204342A MX 9204342 A MX9204342 A MX 9204342A MX 9204342 A MX9204342 A MX 9204342A
Authority
MX
Mexico
Prior art keywords
indoles
formula
present
provides compounds
pharmaceutical salts
Prior art date
Application number
MX9204342A
Other languages
English (en)
Inventor
Julian Blagg
Kelvin Cooper
Peter Lionel Spargo
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX9204342A publication Critical patent/MX9204342A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12Radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)

Abstract

La presente invención provee compuestos de la fórmula (I) y sales farmacéuticas aceptables de los mismos.
MX9204342A 1991-07-24 1992-07-23 Indoles. MX9204342A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919115951A GB9115951D0 (en) 1991-07-24 1991-07-24 Indoles

Publications (1)

Publication Number Publication Date
MX9204342A true MX9204342A (es) 1994-03-31

Family

ID=10698873

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9204342A MX9204342A (es) 1991-07-24 1992-07-23 Indoles.

Country Status (20)

Country Link
EP (2) EP0598754A1 (es)
JP (2) JPH06509336A (es)
CN (2) CN1068816A (es)
AU (2) AU655662B2 (es)
BR (1) BR9206306A (es)
CA (2) CA2112678A1 (es)
CZ (1) CZ13694A3 (es)
FI (2) FI940310A0 (es)
GB (1) GB9115951D0 (es)
HU (1) HU9400199D0 (es)
IE (2) IE922386A1 (es)
IL (2) IL102544A0 (es)
MX (1) MX9204342A (es)
NO (1) NO940237L (es)
NZ (1) NZ243687A (es)
PT (2) PT100717A (es)
SK (1) SK8494A3 (es)
TW (1) TW223060B (es)
WO (2) WO1993002050A1 (es)
ZA (2) ZA925547B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9204024D0 (en) * 1992-02-25 1992-04-08 Fujisawa Pharmaceutical Co Indole derivatives
GB9302577D0 (en) * 1993-02-10 1993-03-24 Fujisawa Pharmaceutical Co Indole derivatives
WO1994022821A1 (en) * 1993-04-05 1994-10-13 Fujisawa Pharmaceutical Co., Ltd. Indole derivatives as testosterone 5 alpha-reductase inhibitors
GB9310092D0 (en) * 1993-05-17 1993-06-30 Fujisawa Pharmaceutical Co Indole derivatives
GB9317096D0 (en) * 1993-08-17 1993-09-29 Pfizer Ltd Indoles
DE69521687T2 (de) * 1994-03-30 2001-10-25 Zeria Pharmaceutical Co., Ltd. 4-indol-1-yl-buttersäure derivate, deren herstellung und deren verwendung als inhibitoren für alpha1-adrenerge rezeptoren und testosteron 5alpha-reduktasen
GB9409583D0 (en) * 1994-05-13 1994-07-06 Pfizer Ltd Indoles
US5543417A (en) * 1994-10-21 1996-08-06 Merck & Co., Inc. Combination method of treating acne using 4-AZA-5α-cholestan-ones and 4-AZA-5α-androstan-ones as selective 5α-reductase inhibitors with anti-bacterial, keratolytic, or anti-inflammatory agents
CZ301985B6 (cs) 1997-05-14 2010-08-25 Atherogenics, Inc. Lécivo pro lécení kardiovaskulárního onemocnení na bázi monoesteru probukolu s jantarovou kyselinou
US6670398B2 (en) 1997-05-14 2003-12-30 Atherogenics, Inc. Compounds and methods for treating transplant rejection
US7417063B2 (en) 2004-04-13 2008-08-26 Bristol-Myers Squibb Company Bicyclic heterocycles useful as serine protease inhibitors
FR2893615B1 (fr) * 2005-11-18 2008-03-07 Sanofi Aventis Sa Derives de 3-acylindole, leur preparation et leur application en therapeutique
PE20090159A1 (es) 2007-03-08 2009-02-21 Plexxikon Inc COMPUESTOS DERIVADOS DE ACIDO INDOL-PROPIONICO COMO MODULADORES PPARs
WO2008118948A1 (en) 2007-03-26 2008-10-02 Atherogenics, Inc. Methods and compositions of derivatives of probucol for the treatment of diabetes
US10703969B2 (en) * 2016-09-27 2020-07-07 Kaohsiung Medical University Detection method for quaternary ammonium compound having γ-carboxyl group

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9011335D0 (en) * 1990-05-21 1990-07-11 Fujisawa Pharmaceutical Co Indolebutyric acid derivatives and process for preparation thereof
WO1993005020A1 (en) * 1991-09-06 1993-03-18 Merck & Co., Inc. Indoles as inhibitors of hiv reverse transcriptase

Also Published As

Publication number Publication date
FI940310A7 (fi) 1994-01-21
FI940311A7 (fi) 1994-01-21
IE922386A1 (en) 1993-01-27
BR9206306A (pt) 1994-11-08
HU9400199D0 (en) 1994-05-30
FI940311A0 (fi) 1994-01-21
EP0598754A1 (en) 1994-06-01
WO1993002051A1 (en) 1993-02-04
ZA925547B (en) 1994-01-24
JPH06509336A (ja) 1994-10-20
IL102545A0 (en) 1993-01-14
SK8494A3 (en) 1994-11-09
PT100717A (pt) 1993-08-31
NO940237D0 (no) 1994-01-24
ZA925546B (en) 1994-01-24
CZ13694A3 (en) 1994-07-13
IL102544A0 (en) 1993-01-14
FI940310A0 (fi) 1994-01-21
WO1993002050A1 (en) 1993-02-04
GB9115951D0 (en) 1991-09-11
NO940237L (no) 1994-01-24
EP0598750A1 (en) 1994-06-01
TW223060B (es) 1994-05-01
PT100718A (pt) 1993-08-31
IE922387A1 (en) 1993-01-27
JPH06511483A (ja) 1994-12-22
AU655662B2 (en) 1995-01-05
CA2112689A1 (en) 1993-02-04
AU2327092A (en) 1993-02-23
AU2327192A (en) 1993-02-23
CA2112678A1 (en) 1993-02-04
NZ243687A (en) 1994-12-22
CN1068816A (zh) 1993-02-10
CN1068817A (zh) 1993-02-10

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