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MX2024012473A - Formulaciones farmaceuticas de liberacion modificada que comprenden deferiprona - Google Patents

Formulaciones farmaceuticas de liberacion modificada que comprenden deferiprona

Info

Publication number
MX2024012473A
MX2024012473A MX2024012473A MX2024012473A MX2024012473A MX 2024012473 A MX2024012473 A MX 2024012473A MX 2024012473 A MX2024012473 A MX 2024012473A MX 2024012473 A MX2024012473 A MX 2024012473A MX 2024012473 A MX2024012473 A MX 2024012473A
Authority
MX
Mexico
Prior art keywords
deferiprone
pharmaceutical formulations
modified release
release pharmaceutical
directed
Prior art date
Application number
MX2024012473A
Other languages
English (en)
Inventor
Marisa Pertile
Andrea Gazzaniga
Matteo Cerea
Micol Cirilli
Original Assignee
Chiesi Farm Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US17/717,913 external-priority patent/US12016850B2/en
Application filed by Chiesi Farm Spa filed Critical Chiesi Farm Spa
Publication of MX2024012473A publication Critical patent/MX2024012473A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A61K9/2036Silicones; Polysiloxanes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención se dirige a composiciones farmacéuticas para administración oral que comprenden deferiprona. En particular, la invención también se dirige a comprimidos de liberación retardada adecuados para administración dos veces al día o una vez al día. La invención también se dirige a métodos de fabricación y uso de los mismos.
MX2024012473A 2022-04-11 2024-10-08 Formulaciones farmaceuticas de liberacion modificada que comprenden deferiprona MX2024012473A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17/717,913 US12016850B2 (en) 2022-04-11 2022-04-11 Modified release pharmaceutical formulations comprising deferiprone
EP22167557 2022-04-11
PCT/EP2023/059304 WO2023198641A1 (en) 2022-04-11 2023-04-07 Modified release pharmaceutical formulations comprising deferiprone

Publications (1)

Publication Number Publication Date
MX2024012473A true MX2024012473A (es) 2024-11-08

Family

ID=86099807

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2024012473A MX2024012473A (es) 2022-04-11 2024-10-08 Formulaciones farmaceuticas de liberacion modificada que comprenden deferiprona

Country Status (8)

Country Link
EP (1) EP4507678A1 (es)
JP (1) JP2025512012A (es)
KR (1) KR20250002399A (es)
CN (1) CN119300809A (es)
AU (1) AU2023254403A1 (es)
CA (1) CA3248497A1 (es)
MX (1) MX2024012473A (es)
WO (1) WO2023198641A1 (es)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8268352B2 (en) * 2002-08-05 2012-09-18 Torrent Pharmaceuticals Limited Modified release composition for highly soluble drugs
AU2003280818A1 (en) 2002-11-18 2004-06-15 Nippon Unicar Company Limited Odorless polyether-modified polysiloxane composition, process for the production thereof, and cosmetics containing the same
CA3172668A1 (en) 2017-10-25 2019-05-02 Chiesi Farmaceutici S.P.A. Delayed release deferiprone tablets and methods of using the same

Also Published As

Publication number Publication date
CN119300809A (zh) 2025-01-10
KR20250002399A (ko) 2025-01-07
CA3248497A1 (en) 2023-10-19
EP4507678A1 (en) 2025-02-19
JP2025512012A (ja) 2025-04-16
WO2023198641A1 (en) 2023-10-19
AU2023254403A1 (en) 2024-11-21

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