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MX2022014094A - Formulaciones farmaceuticas y sus preparaciones para el tratamiento del cancer. - Google Patents

Formulaciones farmaceuticas y sus preparaciones para el tratamiento del cancer.

Info

Publication number
MX2022014094A
MX2022014094A MX2022014094A MX2022014094A MX2022014094A MX 2022014094 A MX2022014094 A MX 2022014094A MX 2022014094 A MX2022014094 A MX 2022014094A MX 2022014094 A MX2022014094 A MX 2022014094A MX 2022014094 A MX2022014094 A MX 2022014094A
Authority
MX
Mexico
Prior art keywords
treatment
preparations
cancer
formulation
pharmaceutical formulations
Prior art date
Application number
MX2022014094A
Other languages
English (en)
Inventor
Mahesh Kandula
Original Assignee
Cellix Bio Private Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cellix Bio Private Ltd filed Critical Cellix Bio Private Ltd
Publication of MX2022014094A publication Critical patent/MX2022014094A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La presente invención se refiere a una formulación farmacéutica de derivados de 5-fluoropirimidina o una sal, solvato o hidrato de los mismos para su administración oral, en donde la formulación es una composición simple que se ingiere de manera simple, más segura, conveniente, no invasiva, con versatilidad y en donde lo más importante es la conformidad del paciente para su administración oral con una conformidad, seguridad y biodisponibilidad mejoradas. Además, se divulga un proceso para la preparación, composición y métodos de administración, dosificaciones de la formulación y su uso para el tratamiento de cánceres y sus complicaciones asociadas.
MX2022014094A 2020-05-19 2021-05-17 Formulaciones farmaceuticas y sus preparaciones para el tratamiento del cancer. MX2022014094A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN202041020998 2020-05-19
PCT/IB2021/054199 WO2021234532A1 (en) 2020-05-19 2021-05-17 Pharmaceutical formulations and their preparations for treatment of cancer

Publications (1)

Publication Number Publication Date
MX2022014094A true MX2022014094A (es) 2022-12-08

Family

ID=78707794

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022014094A MX2022014094A (es) 2020-05-19 2021-05-17 Formulaciones farmaceuticas y sus preparaciones para el tratamiento del cancer.

Country Status (11)

Country Link
US (1) US20250186435A1 (es)
EP (1) EP4153137A4 (es)
JP (1) JP2023528266A (es)
KR (1) KR20230012572A (es)
AU (1) AU2021275620A1 (es)
BR (1) BR112022022796A2 (es)
CA (1) CA3178648A1 (es)
IL (1) IL298204A (es)
MX (1) MX2022014094A (es)
WO (1) WO2021234532A1 (es)
ZA (1) ZA202212702B (es)

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5968914A (en) * 1987-10-28 1999-10-19 Pro-Neuron, Inc. Treatment of chemotherapeutic agent and antiviral agent toxicity with acylated pyrimidine nucleosides
ATE540679T1 (de) * 2004-04-29 2012-01-15 Taiho Pharmaceutical Co Ltd Verfahren zur verringerung der gastrointestinalen toxizität durch verabreichung von tegafur
US20080085310A1 (en) * 2006-10-06 2008-04-10 Maria Oksana Bachynsky Capecitabine rapidly disintegrating tablets
US20110027374A1 (en) * 2008-12-16 2011-02-03 Maria Oksana Bachynsky Capecitabine rapidly disintegrating tablets
CN103156877B (zh) * 2011-12-13 2015-11-25 深圳海王药业有限公司 一种卡培他滨速释微丸及其制备方法
CA2958332A1 (en) * 2014-09-26 2016-03-31 Intas Pharmaceuticals Ltd. Pharmaceutical composition having improved content uniformity
CN104739800A (zh) * 2015-02-03 2015-07-01 吉林修正药业新药开发有限公司 一种卡培他滨片组合物及其制备方法
US20200054659A1 (en) * 2015-06-13 2020-02-20 Intas Pharmaceuticals Ltd. Extended release capecitabine capsules
CN109414438A (zh) * 2016-06-28 2019-03-01 塞尔利克斯生物私人有限公司 用于治疗癌症的组合物和方法
IN201817045551A (es) * 2018-12-03 2018-12-28

Also Published As

Publication number Publication date
AU2021275620A1 (en) 2022-12-08
WO2021234532A1 (en) 2021-11-25
EP4153137A1 (en) 2023-03-29
IL298204A (en) 2023-01-01
JP2023528266A (ja) 2023-07-04
BR112022022796A2 (pt) 2022-12-13
US20250186435A1 (en) 2025-06-12
EP4153137A4 (en) 2024-07-10
KR20230012572A (ko) 2023-01-26
ZA202212702B (en) 2023-04-26
CA3178648A1 (en) 2021-11-25

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