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MX2022007671A - Compuestos antihelminticos que comprenden una estructura de azaindoles. - Google Patents

Compuestos antihelminticos que comprenden una estructura de azaindoles.

Info

Publication number
MX2022007671A
MX2022007671A MX2022007671A MX2022007671A MX2022007671A MX 2022007671 A MX2022007671 A MX 2022007671A MX 2022007671 A MX2022007671 A MX 2022007671A MX 2022007671 A MX2022007671 A MX 2022007671A MX 2022007671 A MX2022007671 A MX 2022007671A
Authority
MX
Mexico
Prior art keywords
azaindoles
anthelmintic compounds
compounds
dirofilaria
anthelmintic
Prior art date
Application number
MX2022007671A
Other languages
English (en)
Inventor
Michael Berger
Michael Linder
Carolin Schneider
Janina Tänzler
Ulrich Sondern
Original Assignee
Intervet Int Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Intervet Int Bv filed Critical Intervet Int Bv
Publication of MX2022007671A publication Critical patent/MX2022007671A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P5/00—Nematocides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Dentistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agronomy & Crop Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente invención se refiere a nuevos compuestos antihelmínticos. Estos compuestos se pueden usar por ejemplo en el tratamiento del tipo de helmintiasis causados por helmintos tal como Dirofilaria, en particular Dirofilaria immitis.
MX2022007671A 2019-12-18 2020-12-17 Compuestos antihelminticos que comprenden una estructura de azaindoles. MX2022007671A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP19217671 2019-12-18
EP20213299 2020-12-11
PCT/EP2020/086660 WO2021122906A1 (en) 2019-12-18 2020-12-17 Anthelmintic compounds comprising azaindoles structure

Publications (1)

Publication Number Publication Date
MX2022007671A true MX2022007671A (es) 2022-07-19

Family

ID=74106031

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022007671A MX2022007671A (es) 2019-12-18 2020-12-17 Compuestos antihelminticos que comprenden una estructura de azaindoles.

Country Status (9)

Country Link
US (1) US12479841B2 (es)
EP (1) EP4077322A1 (es)
JP (1) JP7644121B2 (es)
CN (1) CN114846014B (es)
AU (1) AU2020404100A1 (es)
BR (1) BR112022012130A2 (es)
CA (1) CA3164104A1 (es)
MX (1) MX2022007671A (es)
WO (1) WO2021122906A1 (es)

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CA3183100A1 (en) 2020-05-29 2021-12-02 Boehringer Ingelheim Pharma Gmbh & Co. Kg Anthelmintic heterocyclic compounds
AR127495A1 (es) 2021-11-01 2024-01-31 Boehringer Ingelheim Vetmedica Gmbh Compuestos de pirrolopiridazina como antihelmínticos
WO2023208174A1 (zh) * 2022-04-28 2023-11-02 杭州普济远成生物医药科技有限公司 去泛素化酶抑制剂及其应用
WO2024213752A1 (en) 2023-04-14 2024-10-17 Elanco Animal Health Gmbh Long-term prevention and/or treatment of a disease by slo-1 inhibitors

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Also Published As

Publication number Publication date
AU2020404100A1 (en) 2022-06-09
WO2021122906A1 (en) 2021-06-24
US12479841B2 (en) 2025-11-25
CN114846014A (zh) 2022-08-02
CA3164104A1 (en) 2021-06-24
JP7644121B2 (ja) 2025-03-11
JP2023506303A (ja) 2023-02-15
CN114846014B (zh) 2025-06-13
US20230110397A1 (en) 2023-04-13
EP4077322A1 (en) 2022-10-26
BR112022012130A2 (pt) 2022-08-30

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