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MX2022006569A - Proceso para la sintesis de una 2-tioalquilpirimidina. - Google Patents

Proceso para la sintesis de una 2-tioalquilpirimidina.

Info

Publication number
MX2022006569A
MX2022006569A MX2022006569A MX2022006569A MX2022006569A MX 2022006569 A MX2022006569 A MX 2022006569A MX 2022006569 A MX2022006569 A MX 2022006569A MX 2022006569 A MX2022006569 A MX 2022006569A MX 2022006569 A MX2022006569 A MX 2022006569A
Authority
MX
Mexico
Prior art keywords
formula
sup
compound
synthesis
thioalkyl
Prior art date
Application number
MX2022006569A
Other languages
English (en)
Inventor
Junbae Hong
Original Assignee
Fmc Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fmc Corp filed Critical Fmc Corp
Publication of MX2022006569A publication Critical patent/MX2022006569A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un método para preparar un compuesto de Fórmula 1 y compuestos a partir de él, que comprende tratar un compuesto de Fórmula 2 con un compuesto de Fórmula 3 y hacer reaccionar el intermedio resultante de Fórmula 4 con un compuesto de Fórmula 5 (o una sal de este). (ver Fórmula) El compuesto de Fórmula 1, preparado mediante el método anterior, se puede utilizar para preparar un compuesto de Fórmula 8 (ver Fórmula) donde R2, R3, R4, m y r son como se definen en la memoria descriptiva.
MX2022006569A 2019-12-02 2020-12-02 Proceso para la sintesis de una 2-tioalquilpirimidina. MX2022006569A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962942490P 2019-12-02 2019-12-02
PCT/US2020/062779 WO2021113282A1 (en) 2019-12-02 2020-12-02 Process for synthesis of a 2-thioalkyl pyrimidine

Publications (1)

Publication Number Publication Date
MX2022006569A true MX2022006569A (es) 2022-07-01

Family

ID=74046154

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022006569A MX2022006569A (es) 2019-12-02 2020-12-02 Proceso para la sintesis de una 2-tioalquilpirimidina.

Country Status (12)

Country Link
US (1) US12516045B2 (es)
EP (1) EP4069679A1 (es)
JP (1) JP2023503573A (es)
KR (1) KR20220109428A (es)
CN (1) CN114761384A (es)
AU (1) AU2020395117A1 (es)
BR (1) BR112022010520A2 (es)
CA (1) CA3162102A1 (es)
IL (1) IL292898A (es)
MX (1) MX2022006569A (es)
TW (1) TW202130623A (es)
WO (1) WO2021113282A1 (es)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7326715B2 (en) * 2005-09-23 2008-02-05 N.V. Organon 4-Phenyl-6-substituted-pyrimidine-2-carbonitrile derivatives
JP5163125B2 (ja) 2005-10-14 2013-03-13 旭硝子株式会社 塩基性陰イオン交換樹脂の再生方法
UY31774A (es) * 2008-04-22 2009-12-14 Astrazeneca Ab Compuestos de 2-pirimidin-5- ilcarboxamida sustituidos
US8080566B1 (en) 2008-06-11 2011-12-20 Kalypsys, Inc Carbazole inhibitors of histamine receptors for the treatment of disease
SG11201604813YA (en) * 2014-01-16 2016-07-28 Du Pont Pyrimidinyloxy benzene derivatives as herbicides
CN107250134B (zh) * 2015-03-18 2021-04-09 Fmc公司 作为除草剂的取代的嘧啶氧基吡啶衍生物
TWI828952B (zh) * 2015-06-05 2024-01-11 美商艾佛艾姆希公司 作為除草劑之嘧啶氧基苯衍生物

Also Published As

Publication number Publication date
CN114761384A (zh) 2022-07-15
US20230068064A1 (en) 2023-03-02
IL292898A (en) 2022-07-01
WO2021113282A1 (en) 2021-06-10
CA3162102A1 (en) 2021-06-10
EP4069679A1 (en) 2022-10-12
JP2023503573A (ja) 2023-01-31
US12516045B2 (en) 2026-01-06
KR20220109428A (ko) 2022-08-04
AU2020395117A1 (en) 2022-06-16
BR112022010520A2 (pt) 2022-08-16
TW202130623A (zh) 2021-08-16

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